Fredrik Björkling

Fredrik Björkling

Emeritus

ORCID: 0000-0001-7018-8334

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  1. Published

    [18F]FLT and [18F]FDG PET for non-invasive treatment monitoring of the nicotinamide phosphoribosyltransferase inhibitor APO866 in human xenografts

    Erichsen, K. D., Johnbeck, C. B., Björkling, Fredrik, Madsen, J., Bzorek, M., Jensen, Peter, Højgaard, Liselotte, Sehested, M., Kjær, Andreas & Wessel, Mette Munk, 2013, In: P L o S One. 8, 1, p. 1-8 9 p., e53410.

    Research output: Contribution to journal › Journal article › Research › peer-review

  2. Published

    [18F]FLT PET for Non-Invasive Assessment of Tumor Sensitivity to Chemotherapy: Studies with Experimental Chemotherapy TP202377 in Human Cancer Xenografts in Mice: studies with experimental chemotherapy TP202377 in human cancer xenografts in mice

    Wessel, Mette Munk, Erichsen, K. D., Björkling, Fredrik, Madsen, J., Jensen, P. B., Sehested, M., Højgaard, Liselotte & Kjær, Andreas, 2012, In: P L o S One. 7, 11, p. e50618 e50618.

    Research output: Contribution to journal › Journal article › Research › peer-review

  3. Published

    [18F]FDG and [18F]FLT positron emission tomography imaging following treatment with belinostat in human ovary cancer xenografts in mice

    Wessel, Mette Munk, Erichsen, K. D., Johnbeck, C. B., Björkling, Fredrik, Madsen, J., Jensen, Peter, Sehested, M., Højgaard, Liselotte & Kjær, Andreas, 2013, In: B M C Cancer. 13, p. 1-9 10 p., 168.

    Research output: Contribution to journal › Journal article › Research › peer-review

  4. Published

    Triphenylcarbenium Tetrafluoroborate as an Efficient Catalyst in the Regioselective Reductive Ring Opening of Benzylidene Acetals of Carbohydrates

    Thota, N., Björkling, Fredrik & Kankala, S., 2019, In: ChemistrySelect. 4, 27, p. 7976-7980

    Research output: Contribution to journal › Journal article › Research › peer-review

  5. Published

    Target enzyme mutations are the molecular basis for resistance towards pharmacological inhibition of nicotinamide phosphoribosyltransferase

    Olesen, U. H., Petersen, J. G., Garten, A., Kiess, W., Yoshino, J., Imai, S., Christensen, M. K., Fristrup, P., Thougaard, A. V., Björkling, Fredrik, Jensen, P. B., Nielsen, S. J. & Sehested, M., 10 Dec 2010, In: BMC Cancer. 10, p. 677 13 p.

    Research output: Contribution to journal › Journal article › Research › peer-review

  6. Published

    Synthesis of thiazole linked chalcones and their pyrimidine analogues as anticancer agents

    Kesari, C., Rama, K. R., Sedighi, K., Stenvang, Jan, Björkling, Fredrik, Kankala, S. & Thota, N., 2021, In: Synthetic Communications. 51, 9, p. 1406-1416 11 p.

    Research output: Contribution to journal › Journal article › Research › peer-review

  7. Published

    Synthesis of novel fluorophenylpyrazole-picolinamide derivatives and determination of their anticancer activity

    Kankala, S., Rama, K. R., Kesari, C., Björkling, Fredrik, Nerella, S., Gundepaka, P., Guguloth, H. & Thota, N., 2020, In: Synthetic Communications. 50, 19, p. 2997-3006 10 p.

    Research output: Contribution to journal › Journal article › Research › peer-review

  8. Published

    Synthesis and antitumor effect in vitro and in vivo of substituted 1,3-dihydroindole-2-ones

    Christensen, M. K., Erichsen, K. D., Trojel-Hansen, C., Tjørnelund, J., Nielsen, S. J., Frydenvang, Karla Andrea, Johansen, Tommy Nørskov, Nielsen, Birgitte, Sehested, M., Jensen, P. B., Ikaunieks, M., Zaichenko, A., Loza, E., Kalvinsh, I. & Björkling, Fredrik, 14 Oct 2010, In: Journal of Medicinal Chemistry. 53, 19, p. 7140-7145 6 p.

    Research output: Contribution to journal › Journal article › Research › peer-review

  9. Published

    Synthesis and Structure–Activity Relationships of Novel Non-Steroidal CYP17A1 Inhibitors as Potential Prostate Cancer Agents

    Wróbel, T. M., Rogova, O., Sharma, K., Velazquez, M. N. R., Pandey, A. V., Jørgensen, Flemming Steen, Arendrup, Frederic Schrøder, Andersen, Kasper Langebjerg & Björkling, Fredrik, 2022, In: Biomolecules. 12, 2, 165.

    Research output: Contribution to journal › Journal article › Research › peer-review

  10. Published

    Studies of antibacterial activity (in vitro and in vivo) and mode of action for des-acyl tridecaptins (DATs)

    Couturier, C., Ronzon, Q., Lattanzi, G., Lingard, I., Coyne, S., Cazals, V., Dubarry, N., Yvon, S., Leroi-Geissler, C., Gracia, O. R., Teague, J., Sordello, S., Corbett, D., Bauch, C., Monlong, C., Payne, L., Taillier, T., Fuchs, H., Broenstrup, M., Harrison, P. H. & 10 others, Moynié, L., Lakshminarayanan, A., Gianga, T. M., Hussain, R., Naismith, J. H., Mourez, M., Bacqué, E., Björkling, Fredrik, Sabuco, J. F. & Franzyk, Henrik, 2024, In: European Journal of Medicinal Chemistry. 265, 20 p., 116097.

    Research output: Contribution to journal › Journal article › Research › peer-review

  11. Published

    Structure-activity study of oncocin: On-resin guanidinylation and incorporation of homoarginine, 4-hydroxyproline or 4,4-difluoroproline residues

    Shaikh, Ashif Yasin, Björkling, Fredrik, Zabicka, D., Tomczak, M., Urbas, M., Domraceva, I., Kreicberga, A. & Franzyk, Henrik, 2023, In: Bioorganic Chemistry. 141, 11 p., 106876.

    Research output: Contribution to journal › Journal article › Research › peer-review

  12. Published

    Structural Basis of Metallo-β-lactamase Inhibition by N-Sulfamoylpyrrole-2-carboxylates

    Farley, A. J. M., Ermolovich, Y., Calvopiña, K., Rabe, P., Panduwawala, T., Brem, J., Björkling, Fredrik & Schofield, C. J., 2021, In: ACS Infectious Diseases. 7, 6, p. 1809–1817

    Research output: Contribution to journal › Journal article › Research › peer-review

  13. Published

    Silver carbene complexes: An emerging class of anticancer agents

    Kankala, S., Thota, N., Björkling, Fredrik, Taylor, M. K., Vadde, R. & Balusu, R., Mar 2019, In: Drug Development Research. 80, 2, p. 188-199

    Research output: Contribution to journal › Journal article › Research › peer-review

  14. Published

    Selected strategies to fight pathogenic bacteria

    Plotniece, A., Sobolev, A., Supuran, C. T., Carta, F., Björkling, Fredrik, Franzyk, Henrik, Yli-Kauhaluoma, J., Augustyns, K., Cos, P., De Vooght, L., Govaerts, M., Aizawa, J., Tammela, P. & Žalubovskis, R., 2023, In: Journal of Enzyme Inhibition and Medicinal Chemistry. 38, 1, 27 p., 2155816.

    Research output: Contribution to journal › Review › Research › peer-review

  15. Published

    Prediction of drug efficacy for cancer treatment based on comparative analysis of chemosensitivity and gene expression data

    Wan, P., Li, Q., Larsen, J. E. P., Eklund, A. C., Parlesak, A., Rigina, O., Nielsen, S. J., Björkling, Fredrik & Jonsdottir, S. O., 2012, In: Bioorganic & Medicinal Chemistry. 20, 1, p. 167-176 9 p.

    Research output: Contribution to journal › Journal article › Research › peer-review

  16. Published

    Polymyxins with Potent Antibacterial Activity against Colistin-Resistant Pathogens: Fine-Tuning Hydrophobicity with Unnatural Amino Acids

    Jørgensen, Johan Storm, Harifi Mood, Elnaz, Knap, A. S. H., Nielsen, S. E., Nielsen, Peter E., Żabicka, D., Matias, C., Domraceva, I., Björkling, Fredrik & Franzyk, Henrik, 2024, In: Journal of Medicinal Chemistry. 67, 2, p. 1370–1383

    Research output: Contribution to journal › Journal article › Research › peer-review

  17. Published

    Peptide/β-Peptoid Hybrids with Ultrashort PEG-Like Moieties: Effects on Hydrophobicity, Antibacterial Activity and Hemolytic Properties

    Frederiksen, N., Louka, S., Mudaliar, C., Domraceva, I., Kreicberga, A., Pugovics, O., Żabicka, D., Tomczak, M., Wygoda, W., Björkling, Fredrik & Franzyk, Henrik, 2021, In: International Journal of Molecular Sciences. 22, 13, 17 p., 7041.

    Research output: Contribution to journal › Journal article › Research › peer-review

  18. Published

    Peptide/Peptoid Hybrid Oligomers: The Influence of Hydrophobicity and Relative Side-Chain Length on Antibacterial Activity and Cell Selectivity

    Frederiksen, N., Hansen, Paul Robert, Björkling, Fredrik & Franzyk, Henrik, 4 Dec 2019, In: Molecules (Print Archive Edition). 24, 18 p., 4429.

    Research output: Contribution to journal › Journal article › Research › peer-review

  19. Published

    Optimized Synthesis of Fmoc/Boc-Protected PNA Monomers and their Assembly into PNA Oligomers.

    Shaikh, Ashif Yasin, Björkling, Fredrik, Nielsen, Peter E. & Franzyk, Henrik, 2021, In: European Journal of Organic Chemistry. 2021, 19, p. 2792-2801 10 p.

    Research output: Contribution to journal › Journal article › Research › peer-review

  20. Published

    Novel Agonist Bioisosteres and Common Structure-Activity Relationships for The Orphan G Protein-Coupled Receptor GPR139

    Shehata, M. A., Jensen, A. C. N., Lissa, D., Bisig, C., Isberg, V., Andersen, K. B., Harpsøe, Kasper, Björkling, Fredrik, Bräuner, Hans & Gloriam, David E., 10 Nov 2016, In: Scientific Reports. 6, p. 1-13 13 p., 36681.

    Research output: Contribution to journal › Journal article › Research › peer-review

  21. Published

    Non-steroidal CYP17A1 Inhibitors: Discovery and Assessment

    Wróbel, T. M., Jørgensen, Flemming Steen, Pandey, A. V., Grudzińska, A., Sharma, K., Yakubu, J. & Björkling, Fredrik, 2023, In: Journal of Medicinal Chemistry. 66, 10, p. 6542–6566

    Research output: Contribution to journal › Review › Research › peer-review

  22. Published

    Non-natural Amino Acid and Peptoid Building Blocks for Optimization of the Cell-Penetrating (R-X-R)n Motif

    Wester, A., Björkling, Fredrik, Nieslen, P. & Franzyk, Henrik, Sep 2018, In: Journal of Peptide Science. 24, p. S94-S94

    Research output: Contribution to journal › Conference abstract in journal › Research › peer-review

  23. Published

    Microwave-assisted solid-phase synthesis of antisense acpP peptide nucleic acid-peptide conjugates active against colistin- and tigecycline-resistant E. coli and K. pneumoniae

    Hansen, A. M., Bonke, G., Hogendorf, W. F. J., Björkling, Fredrik, Nielsen, J., Kongstad, Kenneth Thermann, Zabicka, D., Tomczak, M., Urbas, M., Nielsen, Peter E. & Franzyk, Henrik, 2019, In: European Journal of Medicinal Chemistry. 168, p. 134-145 12 p.

    Research output: Contribution to journal › Journal article › Research › peer-review

  24. Published

    Jagten på kongens efterfølger

    Franzyk, Henrik, Björkling, Fredrik, Nielsen, J. & Nielsen, Peter E., 2015, In: Lægemiddelforskning. 2015, p. 24-27 4 p.

    Research output: Contribution to journal › Journal article › Communication

  25. Published

    Inhibitors of human histone deacetylase with potent activity against the African trypanosome Trypanosoma brucei

    Kelly, J., Taylor, M. C., Horn, D., Loza, E., Kalvinsh, I. & Björkling, Fredrik, 2012, In: Bioorganic & Medicinal Chemistry Letters. 22, 5, p. 1886–1890 5 p.

    Research output: Contribution to journal › Journal article › Research › peer-review

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ID: 8863737