Hans Bräuner

Hans Bräuner

Prodekan for forskning


  1. 2005
  2. Published

    Rigid nonproteinogenic cyclic amino acids as ligands for glutamate receptors: trans-tris(homoglutamic) acids

    Meyer, U., Bisel, P., Bräuner, Hans, Madsen, Ulf, Höfner, G., Wanner, K. T. & Frahm, A. W., Feb 2005, In: Chirality. 17, 2, p. 99-107

    Research output: Contribution to journalJournal articleResearchpeer-review

  3. Published

    Deorphanization of GPRC6A: a promiscuous L-alpha-amino acid receptor with preference for basic amino acids

    Wellendorph, Petrine, Hansen, K. B., Balsgaard, A., Greenwood, J. R., Egebjerg, J. & Bräuner, Hans, Mar 2005, In: Molecular Pharmacology. 67, 3, p. 589-97

    Research output: Contribution to journalJournal articleResearchpeer-review

  4. Published

    Synthesis of novel N1-substituted bicyclic pyrazole amino acids and evaluation of their interaction with glutamate receptors

    Conti, P., Grazioso, G., di Ventimiglia, S. J., Pinto, A., Roda, G., Madsen, Ulf, Bräuner, Hans, Nielsen, Birgitte, Costagli, C. & Galli, A., Jun 2005, In: Chemistry & Biodiversity. 2, 6, p. 748-57

    Research output: Contribution to journalJournal articleResearchpeer-review

  5. Published

    Tetrazolyl isoxazole amino acids as ionotropic glutamate receptor antagonists: synthesis, modelling and molecular pharmacology

    Frølund, Bente, Greenwood, J. R., Holm, M. M., Egebjerg, J., Madsen, Ulf, Nielsen, Birgitte, Bräuner, Hans, Stensbøl, T. B. & Krogsgaard-Larsen, Povl, 15 Sep 2005, In: Bioorganic & Medicinal Chemistry. 13, 18, p. 5391-8

    Research output: Contribution to journalJournal articleResearchpeer-review

  6. Published

    Novel cyclic gamma-hydroxybutyrate (GHB) analogs with high affinity and stereoselectivity of binding to GHB sites in rat brain

    Wellendorph, Petrine, Høg, S., Greenwood, J. R., de Lichtenberg, A., Nielsen, Birgitte, Frølund, Bente, Brehm, L., Clausen, Rasmus Prætorius & Bräuner, Hans, Oct 2005, In: Journal of Pharmacology and Experimental Therapeutics. 315, 1, p. 346-51

    Research output: Contribution to journalJournal articleResearchpeer-review

  7. Published

    Synthesis, binding affinity at glutamic acid receptors, neuroprotective effects, and molecular modeling investigation of novel dihydroisoxazole amino acids

    Conti, P., De Amici, M., Grazioso, G., Roda, G., Pinto, A., Hansen, K. B., Nielsen, Birgitte, Madsen, Ulf, Bräuner, Hans, Egebjerg, J., Vestri, V., Pellegrini-Giampietro, D. E., Sibille, P., Acher, F. C. & De Micheli, C., 6 Oct 2005, In: Journal of Medicinal Chemistry. 48, 20, p. 6315-25

    Research output: Contribution to journalJournal articleResearchpeer-review

  8. Published

    Tweaking agonist efficacy at N-methyl-D-aspartate receptors by site-directed mutagenesis

    Hansen, K. B., Clausen, Rasmus Prætorius, Bjerrum, E. J., Bechmann, C., Greenwood, J. R., Christensen, C., Kristensen, Jesper Langgaard, Egebjerg, J. & Bräuner, Hans, Dec 2005, In: Molecular Pharmacology. 68, 6, p. 1510-23

    Research output: Contribution to journalJournal articleResearchpeer-review

  9. 2006
  10. Published

    Functional characterisation of homomeric ionotropic glutamate receptors GluR1-GluR6 in a fluorescence-based high throughput screening assay

    Strange, M., Bräuner, Hans & Jensen, Anders A., 2006, In: Combinatorial Chemistry & High Throughput Screening. 9, 2, p. 147-58 12 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  11. Published
  12. Published

    Known regulators of nitric oxide synthase and arginase are agonists at the human G-protein-coupled receptor GPRC6A

    Christiansen, B., Wellendorph, Petrine & Bräuner, Hans, Apr 2006, In: British Journal of Pharmacology. 147, 8, p. 855-63

    Research output: Contribution to journalJournal articleResearchpeer-review

  13. Published

    Activity of L-alpha-amino acids at the promiscuous goldfish odorant receptor 5.24

    Christiansen, B., Wellendorph, Petrine & Bräuner, Hans, 24 Apr 2006, In: European Journal of Pharmacology. 536, 1-2, p. 98-101

    Research output: Contribution to journalJournal articleResearchpeer-review

  14. Published

    Differential compartmentalization and distinct functions of GABAB receptor variants

    Vigot, R., Barbieri, S., Bräuner, Hans, Turecek, R., Shigemoto, R., Zhang, Y., Luján, R., Jacobson, L. H., Biermann, B., Fritschy, J., Vacher, C., Müller, M., Sansig, G., Guetg, N., Cryan, J. F., Kaupmann, K., Gassmann, M., Oertner, T. G. & Bettler, B., 18 May 2006, In: Neuron. 50, 4, p. 589-601

    Research output: Contribution to journalJournal articleResearchpeer-review

  15. 2007
  16. Published

    Allosteric modulation of the calcium-sensing receptor

    Jensen, Anders A. & Bräuner, Hans, 2007, In: Current Neuropharmacology. 5, 3, p. 180-186

    Research output: Contribution to journalJournal articleResearchpeer-review

  17. Published

    Cloning and characterization of a functional human ¿-aminobutyric acid (GABA) transporter, human GAT-2

    Christiansen, B., Meinild, A., Jensen, Anders A. & Bräuner, Hans, 2007, In: Journal of Biological Chemistry. 282, 27, p. 19331-19341 11 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  18. Published

    En genetisk variation i en serotonin-receptor: et muligt link til depression?

    Krzywkowski, K. M., Davies, P. A., Feinberg-Zadek, P. L., Jensen, Anders A. & Bräuner, Hans, 2007, In: Lægemiddelforskning. p. 30-31

    Research output: Contribution to journalJournal articleCommunication

  19. Published

    Erratum: Synthesis and pharmacology of glutamate receptor ligands: New isothiazole analogues of ibotenic acid (Organic and Biomolecular Chemistry (2007) 5 DOI:10.1039/b615162k)

    Jørgensen, Charlotte Grube, Clausen, Rasmus Prætorius, Hansen, K. B., Bräuner, Hans, Nielsen, Birgitte, Metzler, B., Kehler, J., Krogsgaard-Larsen, Povl & Madsen, Ulf, 2007, In: Organic and Biomolecular Chemistry. 5, 5, p. 848 1 p.

    Research output: Contribution to journalComment/debateResearchpeer-review

  20. Published

    Functional characterization of Tet-AMPA [tetrazolyl-2-amino-3-(3-hydroxy-5-methyl- 4-isoxazolyl)propionic acid] analogues at ionotropic glutamate receptors GluR1-GluR4. The molecular basis for the functional selectivity profile of 2-Bn-Tet-AMPA

    Jensen, Anders A., Christesen, T., Bølcho, U., Greenwood, J. R., Postorino, G., Vogensen, S. B., Johansen, Tommy Nørskov, Egebjerg, J., Bräuner, Hans & Clausen, Rasmus Prætorius, 2007, In: Journal of Medicinal Chemistry. 50, 17, p. 4177-4185 9 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  21. Published

    GABA/benzodiazepinreceptorer

    Bräuner, Hans, 2007, Basal og klinisk farmakologi. Kampmann, J. P., Brøsen, K. & Simonsen, U. (eds.). 3 ed. København: FADL's Forlag, p. 209-212

    Research output: Chapter in Book/Report/Conference proceedingBook chapterEducation

  22. Published

    Molekylær farmakologiske subtyper

    Bräuner, Hans, 2007, In: Lundbeckfondens årsskrift 2006-2007. 2006-2007, p. 30-32

    Research output: Contribution to journalJournal articleCommunication

  23. Published

    Naturally occurring variations in the human 5-HT3A gene profoundly impact 5-HT3 receptor function and expression

    Krzywkowski, K. M., Jensen, Anders A., Connolly, C. N. & Bräuner, Hans, 2007, In: Pharmacogenetics and Genomics (Print Edition). 17, 4, p. 255-266

    Research output: Contribution to journalJournal articleResearchpeer-review

  24. Published

    Novel 5-substituted 1-pyrazolol analogues of ibotenic acid: synthesis and pharmacology at glutamate receptors

    Jørgensen, Charlotte Grube, Bräuner, Hans, Nielsen, Birgitte, Kehler, J., Clausen, Rasmus Prætorius, Krogsgaard-Larsen, Povl & Madsen, Ulf, 2007, In: Bioorganic & Medicinal Chemistry. 15, 10, p. 3524-3538

    Research output: Contribution to journalJournal articleResearchpeer-review

  25. Published

    Pharmacological characterization of mouse GPRC6A, an L-alpha-amino-acid receptor modulated by divalent cations

    Christiansen, B., Hansen, K. B., Wellendorph, Petrine & Bräuner, Hans, 2007, In: British Journal of Pharmacology. 150, 6, p. 798-807

    Research output: Contribution to journalJournal articleResearchpeer-review

  26. Published

    Structure, pharmacology and therapeutic prospects of family C G-protein coupled receptors

    Bräuner, Hans, Wellendorph, Petrine & Jensen, Anders A., 2007, In: Current Drug Targets. 8, 1, p. 169-184

    Research output: Contribution to journalJournal articleResearchpeer-review

  27. Published

    Synthesis and pharmacological characterization at glutamate receptors of erythro- and threo-tricholomic acid and homologues thereof

    Conti, P., De Amici, M., Roda, G., Pinto, A., Tamborini, L., Madsen, Ulf, Nielsen, Birgitte, Bräuner, Hans & De Micheli, C., 2007, In: Tetrahedron. 63, 10, p. 2249-2256

    Research output: Contribution to journalJournal articleResearchpeer-review

  28. Published

    Synthesis and pharmacology of glutamate receptor ligands: new isothiazole analogues of ibotenic acid

    Jørgensen, Charlotte Grube, Clausen, Rasmus Prætorius, Hansen, K. B., Bräuner, Hans, Nielsen, Birgitte, Metzler, B., Kehler, J., Krogsgaard-Larsen, Povl & Madsen, Ulf, 2007, In: Organic & Biomolecular Chemistry. 5, 3, p. 463-471

    Research output: Contribution to journalJournal articleResearchpeer-review

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