Birgitte Nielsen
Academic Coordinator, !!Faglig koordinator
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A new metabotropic glutamate receptor agonist with in vivo anti-allodynic activity
Stanley, N. J., Hutchinson, M. R., Kvist, T., Nielsen, Birgitte, Mathiesen, Jesper M., Bräuner, Hans, Avery, T. D., Tiekink, E. R. T., Pedersen, D. S., Irvine, R. J., Abell, A. D. & Taylor, D. K., 2010, In: Bioorganic & Medicinal Chemistry. 18, 16, p. 6089-6098Research output: Contribution to journal › Journal article › Research › peer-review
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A new phenylalanine derivative acts as an antagonist at the AMPA receptor GluA2 and introduces partial domain closure: Synthesis, resolution, pharmacology, and crystal structure
Szymanska, E., Frydenvang, Karla Andrea, Contreras-Sanz, A., Pickering, Darryl S, Frola, E., Serafimoska, Z., Nielsen, Birgitte, Kastrup, Jette Sandholm Jensen & Johansen, Tommy Nørskov, 4 Oct 2011, In: Journal of Medicinal Chemistry. 54, 20, p. 7289-7298Research output: Contribution to journal › Journal article › Research › peer-review
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A new structural class of subtype-selective inhibitor of cloned excitatory amino acid transporter, EAAT2
Bräuner, Hans, Hermit, M. B., Nielsen, Birgitte, Krogsgaard-Larsen, Povl & Johansen, Tommy Nørskov, 6 Oct 2000, In: European Journal of Pharmacology. 406, 1, p. 41-4Research output: Contribution to journal › Journal article › Research › peer-review
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A stereochemical anomaly: the cyclised (R)-AMPA analogue (R)-3-hydroxy-4,5,6,7-tetrahydroisoxazolo[5,4-c]pyridine-5-carboxylic acid [(R)-5-HPCA] resembles (S)-AMPA at glutamate receptors
Vogensen, S., Greenwood, J., Varming, A. R., Brehm, L., Pickering, Darryl S, Nielsen, Birgitte, Liljefors, T., Clausen, Rasmus Prætorius, Johansen, Tommy Nørskov & Krogsgaard-Larsen, Povl, 2004, In: Organic & Biomolecular Chemistry. 2, 2, p. 206-213Research output: Contribution to journal › Journal article › Research › peer-review
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A tetrazolyl-substituted subtype-selective AMPA receptor agonist
Vogensen, S. B., Frydenvang, Karla Andrea, Greenwood, J. R., Postorino, G., Nielsen, Birgitte, Pickering, Darryl S, Ebert, B., Bølcho, U., Egebjerg, J., Gajhede, Michael, Kastrup, Jette Sandholm Jensen, Johansen, Tommy Nørskov, Clausen, Rasmus Prætorius & Krogsgaard-Larsen, Povl, 2007, In: Journal of Medicinal Chemistry. 50, 10, p. 2408-2414Research output: Contribution to journal › Journal article › Research › peer-review
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AMPA receptor agonists: structural, conformational and stereochemical aspects
Hansen, J., Jørgensen, Flemming Steen, Lund, Trine Meldgaard, Nielsen, Birgitte, Reinhardt, A., Breum, I., Brehm, L. & Krogsgaard-Larsen, Povl, 1992, Excitatory Amino Acid Receptors. Krogsgaard-Larsen, P. & Hansen, J. J. (eds.). Ellis Horwood: Chichester, 30 p.Research output: Chapter in Book/Report/Conference proceeding › Book chapter › Research › peer-review
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Adskillelse af lægemidlers spejlbilledformer
Nielsen, Birgitte, Breum, I. & Hansen, J. J., 1991, In: Lægemiddelforskning. p. 40-41 2 p.Research output: Contribution to journal › Journal article › Research
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Aminolysis of resin-bound N-nosylaziridine-2-carboxylic acids
Olsen, Christian Adam, Christensen, C., Nielsen, Birgitte, Farah, M. M., Mohamed, F. M., Witt, M., Clausen, Rasmus Prætorius, Kristensen, Jesper Langgaard, Franzyk, Henrik & Jaroszewski, J. W., 2006, In: Organic Letters. 8, 15, p. 3371-4 4 p.Research output: Contribution to journal › Journal article › Research › peer-review
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Analogues of 3-Hydroxyisoxazole-Containing Glutamate Receptor Ligands Based on the 3-Hydroxypyrazole-Moiety: Design, Synthesis and Pharmacological Characterization
Jørgensen, L., Nielsen, Birgitte, Pickering, Darryl S, Kristensen, Anders Skov, Frydenvang, Karla Andrea, Madsen, Ulf & Clausen, Rasmus Prætorius, 2014, In: Neurochemical Research. 39, 10, p. 1895-1905 11 p.Research output: Contribution to journal › Journal article › Research › peer-review
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Aryl and cycloalkyl analogues of AMPA: synthetic, pharmacological and stereochemical aspects
Skjærbæk, N., Brehm, L., Johansen, Tommy Nørskov, Hansen, L. M., Nielsen, Birgitte, Ebert, B., Søby, K., Stensbøl, T. B., Falch, E. & Krogsgaard-Larsen, Povl, 1998, In: Bioorganic & Medicinal Chemistry. 6, 1, p. 119-131 13 p.Research output: Contribution to journal › Journal article › Research › peer-review
ID: 88868846
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5-(Piperidine-4-yl)-3-hydroxypyrazole: a novel scaffold forprobing the orthosteric GABAA receptor binding site
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Exploring pharmacological mechanisms of lavender (Lavandula angustifolia) essential oil on central nervous system targets
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Discovery of the First Highly Selective Antagonist of the GluK3 Kainate Receptor Subtype
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