Hans Bräuner

Hans Bräuner

Prodekan for forskning


  1. Published

    Metabolic and skeletal homeostasis are maintained in full locus GPRC6A knockout mice

    Jørgensen, C. V., Gasparini, S. J., Tu, J., Zhou, H., Seibel, M. J. & Bräuner, Hans, 12 Apr 2019, In: Scientific Reports. 9, 1, 8 p., 5995.

    Research output: Contribution to journalJournal articleResearchpeer-review

  2. Published

    Label-free dynamic mass redistribution analysis of endogenous adrenergic receptor signaling in primary preadipocytes and differentiated adipocytes

    Jørgensen, C. V., Zhou, H., Seibel, M. J. & Bräuner, Hans, 1 Apr 2019, In: Journal of Pharmacological and Toxicological Methods. 97, p. 59-66 8 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  3. Published

    Structure-Activity Relationship, Pharmacological Characterization, and Molecular Modeling of Noncompetitive Inhibitors of the Betaine/γ-Aminobutyric Acid Transporter 1 (BGT1)

    Jørgensen, L., Al-Khawaja, A., Kickinger, S., Vogensen, S. B., Skovgaard-Petersen, J., Rosenthal, E., Borkar, N., Löffler, R., Madsen, K. K., Bräuner, Hans, Schousboe, Arne, Ecker, G. F., Wellendorph, Petrine & Clausen, Rasmus Prætorius, 9 Oct 2017, In: Journal of Medicinal Chemistry. 60, 21, p. 8834-8846

    Research output: Contribution to journalJournal articleResearchpeer-review

  4. Published

    Structure-activity relationships for negative allosteric mGluR5 modulators

    Kaae, B. H., Harpsøe, Kasper, Kvist, T., Mathiesen, Jesper M., Mølck, C., Gloriam, David E., Jimenez, H. N., Uberti, M. A., Nielsen, S. M., Nielsen, Birgitte, Bräuner, Hans, Sauerberg, P., Clausen, Rasmus Prætorius & Madsen, Ulf, 2012, In: ChemMedChem. 7, 3, p. 440-451

    Research output: Contribution to journalJournal articleResearchpeer-review

  5. Published

    Specific gamma-hydroxybutyrate-binding sites but loss of pharmacological effects of gamma-hydroxybutyrate in GABA-B1-deficient mice

    Kaupmann, K., Cryan, J. F., Wellendorph, Petrine, Mombereau, C., Sansig, G., Klebs, K., Schmutz, M., Froestl, W., van der Putten, H., Mosbacher, J., Bräuner, Hans, Waldmeier, P. & Bettler, B., Nov 2003, In: European Journal of Neuroscience. 18, 10, p. 2722-30

    Research output: Contribution to journalJournal articleResearchpeer-review

  6. Published

    Discovery of a subtype-selective of the human betaine/GABA transporter 1 (BGT-1) with a non-competitive pharmacological profile

    Kragholm, B., Kvist, T., Madsen, K. K., Jørgensen, L., Vogensen, S. B., Schousboe, Arne, Clausen, Rasmus Prætorius, Jensen, Anders A. & Bräuner, Hans, 2013, In: Biochemical Pharmacology. 86, p. 521-528

    Research output: Contribution to journalJournal articleResearchpeer-review

  7. Published

    Design of excitatory amino acid receptor agonists, partial agonists and antagonists: Ibotenic acid as a key lead structure

    Krogsgaard-Larsen, Povl, Ebert, B., Lund, Trine Meldgaard, Bräuner, Hans, Sloøk, F. A., Johansen, Tommy Nørskov, Brehm, L. & Madsen, Ulf, 10 Sep 1996, In: European Journal of Medicinal Chemistry. 31, 7-8, p. 515-537 23 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  8. Published

    Selective antagonists at group I metabotropic glutamate receptors: synthesis and molecular pharmacology of 4-aryl-3-isoxazolol amino acids

    Kromann, H., Sløk, F. A., Stensbøl, T. B., Bräuner, Hans, Madsen, Ulf & Krogsgaard-Larsen, Povl, 14 Feb 2002, In: Journal of Medicinal Chemistry. 45, 4, p. 988-91

    Research output: Contribution to journalJournal articleResearchpeer-review

  9. Published

    High-frequency HTR3B variant associated with major depression dramatically augments the signaling of the human 5-HT3AB receptor

    Krzywkowski, K. M., Davies, P. A., Feinberg-Zadek, P. L., Bräuner, Hans & Jensen, Anders A., 2008, In: Proceedings of the National Academy of Science of the United States of America. 105, 2, p. 722-727

    Research output: Contribution to journalJournal articleResearchpeer-review

  10. Published

    En genetisk variation i en serotonin-receptor: et muligt link til depression?

    Krzywkowski, K. M., Davies, P. A., Feinberg-Zadek, P. L., Jensen, Anders A. & Bräuner, Hans, 2007, In: Lægemiddelforskning. p. 30-31

    Research output: Contribution to journalJournal articleCommunication

  11. Published

    Characterization of the effects of four HTR3B polymorphisms on human 5-HT3AB receptor expression and signalling

    Krzywkowski, K. M., Davies, P. A., Irving, A. J., Bräuner, Hans & Jensen, Anders A., 2008, In: Pharmacogenetics and Genomics (Print Edition). 18, 12, p. 1027-1040

    Research output: Contribution to journalJournal articleResearchpeer-review

  12. Published

    En genetisk variation i en serotonin–receptor – et muligt link til depression?

    Krzywkowski, K. M., Feinberg-Zadek, P., Davies, P. A., Jensen, Anders A. & Bräuner, Hans, 2008, In: Dansk Kemi 83. 89, 6/7

    Research output: Contribution to journalJournal articleCommunication

  13. Published

    Naturally occurring variations in the human 5-HT3A gene profoundly impact 5-HT3 receptor function and expression

    Krzywkowski, K. M., Jensen, Anders A., Connolly, C. N. & Bräuner, Hans, 2007, In: Pharmacogenetics and Genomics (Print Edition). 17, 4, p. 255-266

    Research output: Contribution to journalJournal articleResearchpeer-review

  14. Published

    Radiosynthesis and characterisation of a potent and selective GPR139 agonist radioligand

    Kuhne, S., Nøhr, A. C., Marek, A., Elbert, T., Klein, A. B., Bräuner, Hans, Wellendorph, Petrine & Pedersen, D. S., 2016, In: RSC Advances. 6, 2, p. 947-952 6 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  15. Published

    The use of Xenopus oocytes in drug screening

    Kvist, T., Hansen, K. B. & Bräuner, Hans, 2011, In: Expert Opinion on Drug Discovery. 6, 2, p. 141-153

    Research output: Contribution to journalReviewResearchpeer-review

  16. Published

    Structure-based discovery of antagonists for GluN3-containing N-methyl-D-aspartate receptors

    Kvist, T., Greenwood, J. R., Hansen, K. B., Traynelis, S. F. & Bräuner, Hans, 22 Aug 2013, In: Neuropharmacology. 75, p. 324-336 13 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  17. Published

    Crystal structure and pharmacological characterization of a novel N-methyl-D-aspartate (NMDA) receptor antagonist at the GluN1 glycine binding site

    Kvist, T., Steffensen, T. B., Greenwood, J. R., Mehrzad Tabrizi, F., Hansen, K. B., Gajhede, Michael, Pickering, Darryl S, Traynelis, S. F., Kastrup, Jette Sandholm Jensen & Bräuner, Hans, 2013, In: The Journal of Biological Chemistry. 288, p. 33124-35 12 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  18. Published

    The four human ¿-aminobutyric acid (GABA) transporters: pharmacological characterization and validation of a highly efficient screening assay

    Kvist, T., Christiansen, B., Jensen, Anders A. & Bräuner, Hans, 2009, In: Combinatorial Chemistry & High Throughput Screening. 12, 3, p. 241-249

    Research output: Contribution to journalJournal articleResearchpeer-review

  19. Published

    International Union of Basic and Clinical Pharmacology. CVIII. Calcium-Sensing Receptor Nomenclature, Pharmacology, and Function

    Leach, K., Hannan, F. M., Josephs, T. M., Keller, A. N., Møller, T. C., Ward, D. T., Kallay, E., Mason, R. S., Thakker, R. V., Riccardi, D., Conigrave, A. D. & Bräuner, Hans, Jul 2020, In: Pharmacological Reviews. 72, 3, p. 558-604 47 p.

    Research output: Contribution to journalReviewResearchpeer-review

  20. Published

    (R)-(3-amino-2-fluoropropyl) phosphinic acid (AZD3355), a novel GABAB receptor agonist, inhibits transient lower esophageal sphincter relaxation through a peripheral mode of action

    Lehmann, A., Antonsson, M., Holmberg, A. A., Blackshaw, L. A., Brändén, L., Bräuner, Hans, Christiansen, B., Dent, J., Elebring, T., Jacobson, B., Jensen, J., Mattsson, J. P., Nilsson, K., Oja, S. S., Page, A. J., Saransaari, P. & von Unge, S., 2009, In: Journal of Pharmacology and Experimental Therapeutics. 331, 2, p. 504-512

    Research output: Contribution to journalJournal articleResearchpeer-review

  21. Published

    Mutational Landscape of the Proglucagon-Derived Peptides

    Lindquist, Peter, Madsen, Jakob Sture, Bräuner, Hans, Rosenkilde, Mette & Hauser, Alexander Sebastian, 2021, In: Frontiers in Endocrinology. 12, 14 p., 698511.

    Research output: Contribution to journalJournal articleResearchpeer-review

  22. Published

    Synthesis and pharmacology of 3-isoxazolol amino acids as selective antagonists at group I metabotropic glutamic acid receptors

    Madsen, Ulf, Bräuner, Hans, Frydenvang, Karla Andrea, Hvene, L., Johansen, Tommy Nørskov, Nielsen, Birgitte, Sánchez, C., Stensbøl, T. B., Bischoff, F. & Krogsgaard-Larsen, Povl, 2001, In: Journal of Medicinal Chemistry. 44, 7, p. 1051-9 9 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  23. Published

    Ionotropic excitatory amino acid receptor ligands. Synthesis and pharmacology of a new amino acid AMPA antagonist

    Madsen, Ulf, Sløk, F. A., Stensbøl, T. B., Bräuner, Hans, Lützhøft, H. H., Poulsen, M. V., Eriksen, L. & Krogsgaard-Larsen, Povl, Jan 2000, In: European Journal of Medicinal Chemistry. 35, 1, p. 69-76

    Research output: Contribution to journalJournal articleResearchpeer-review

  24. Published

    Synthesis and pharmacology of N-alkylated derivatives of the excitotoxin ibotenic acid

    Madsen, Ulf, Dumpis, M. A., Bräuner, Hans & Piotrovsky, L. B., 16 Jun 1998, In: Bioorganic & Medicinal Chemistry Letters. 8, 12, p. 1563-8

    Research output: Contribution to journalJournal articleResearchpeer-review

  25. Published

ID: 1302910