Karla Andrea Frydenvang
Associate Professor
Structural Biology
Universitetsparken 2
2100 København Ø
ORCID: 0000-0002-5823-3478
Introductory remarks on publicationslist
See Homepage for complete list of publications (incl. all publications from before 2007)1 - 6 out of 6Page size: 50
- 2024
- Accepted/In press
AI Based Discovery of a New AKR1C3 Inhibitor for Anticancer Applications
Pippione, A. C., Vigato, C., Tucciarello, C., Hussain, Samrina, Salladini, Edoardo, Truong, H. H., Henriksen, N. M., Vanzetti, G., Giordano, G., Zonari, D., Mirza, Osman Asghar, Frydenvang, Karla Andrea, Pignochino, Y., Oliaro-Bosso, S., Boschi, D. & Lolli, M. L., 2024, (Accepted/In press) In: ACS Medicinal Chemistry Letters.Research output: Contribution to journal › Letter › Research › peer-review
- Published
Discovery and Structure-Activity Relationships of 2,5-Dimethoxyphenylpiperidines as Selective Serotonin 5-HT2A Receptor Agonists
Marcher, Emil, Jensen, Anders A., Smits, G., Frydenvang, Karla Andrea & Kristensen, Jesper Langgaard, 2024, In: Journal of Medicinal Chemistry. 69, 9, p. 7224–7244Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Exploring thienothiadiazine dioxides as isosteric analogues of benzo- and pyridothiadiazine dioxides in the search of new AMPA and kainate receptor positive allosteric modulators
Francotte, P., Bay, Y., Goffin, E., Colson, T., Lesenfants, C., Dorosz, J., Laulumaa, S., Fraikin, P., de Tullio, P., Beaufour, C., Botez, I., Pickering, Darryl S, Frydenvang, Karla Andrea, Danober, L., Kristensen, A. S., Kastrup, Jette Sandholm Jensen & Pirotte, B., 2024, In: European Journal of Medicinal Chemistry. 264, 15 p., 116036.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Small-molecule positive allosteric modulation of homomeric kainate receptors GluK1-3: development of screening assays and insight into GluK3 structure
Bay, Y., Venskutonytė, R., Frantsen, S. M., Thorsen, T. S., Musgaard, M., Frydenvang, Karla Andrea, Francotte, P., Pirotte, B., Biggin, P. C., Kristensen, Anders Skov, Boesen, T., Pickering, Darryl S, Gajhede, Michael & Kastrup, Jette Sandholm Jensen, 2024, In: FEBS Journal. 291, 7, p. 1506-1529Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Structure-guided optimization of 3-hydroxybenzoisoxazole derivatives as inhibitors of Aldo-keto reductase 1C3 (AKR1C3) to target prostate cancer
Pippione, A. C., Kovachka, S., Vigato, C., Bertarini, L., Mannella, I., Sainas, S., Rolando, B., Denasio, E., Piercy-Mycock, H., Romalho, L., Salladini, E., Adinolfi, S., Zonari, D., Peraldo-Neia, C., Chiorino, G., Passoni, A., Mirza, O. A., Frydenvang, K., Pors, K., Lolli, M. L. & 3 others, , 2024, In: European Journal of Medicinal Chemistry. 268, 20 p., 116193.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
The positive allosteric modulator BPAM344 and L-glutamate introduce an active-like structure of the ligand-binding domain of GluK2
Bay, Y., Egeberg Jeppesen, M., Frydenvang, Karla Andrea, Francotte, P., Pirotte, B., Pickering, Darryl S, Kristensen, Anders Skov & Kastrup, Jette Sandholm Jensen, 2024, In: FEBS Letters. 598, 7, p. 743-757Research output: Contribution to journal › Journal article › Research › peer-review
ID: 1305625
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290
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Structural analysis of Cytochrome P450 BM3 mutant M11 in complex with dithiothreitol
Research output: Contribution to journal › Journal article › Research › peer-review
Published -
153
downloads
Structure elucidation of prenyl- and geranyl substituted coumarins in Gerbera piloselloides by NMR spectroscopy, electronic circular dichroism calculations, and single crystal X-ray crystallography
Research output: Contribution to journal › Journal article › Research › peer-review
Published