Frederik Diness
Guest researcher, Guest Researcher
- 2003
- Published
The Pictet-Spengler reaction in solid-phase combinatorial chemistry
Nielsen, T. E., Diness, Frederik & Meldal, Morten Peter, Nov 2003, In: Current Opinion in Drug Discovery & Development. 6, 6, p. 801-14 14 p.Research output: Contribution to journal › Journal article › Research › peer-review
- 2004
- Published
INTRAMOLECULAR CARBAMOYLIMINIUM ACTIVATED SOLID PHASE PICTET-SPENGLER REACTIONS. TOWARDS MCR AGONISTS
Diness, Frederik, Beyer, J. & Meldal, Morten Peter, 2004, In: Journal of Peptide Science. 10, p. 126-126Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Synthesis of 3-Boc-(1,3)-oxazinane-protected amino aldehydes from amino acids and their conversion into urea precursors. Novel building blocks for combinatorial synthesis
Diness, Frederik, Beyer, J. & Meldal, Morten Peter, Apr 2004, In: Molecular Informatics. 23, 2-3, p. 130-144Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Probing the aglycon binding site of a beta-glucosidase: a collection of C-1-modified 2,5-dideoxy-2,5-imino-D-mannitol derivatives and their structure-activity relationships as competitive inhibitors
Wrodnigg, T. M., Diness, Frederik, Gruber, C., Häusler, H., Lundt, I., Rupitz, K., Steiner, A. J., Stütz, A. E., Tarling, C. A., Withers, S. G. & Wölfler, H., 1 Jul 2004, In: Bioorganic & Medicinal Chemistry. 12, 13, p. 3485-95 11 p.Research output: Contribution to journal › Journal article › Research › peer-review
- 2005
- Published
Dual approach to intramolecular carbamoyliminium activated solid phase Pictet-Spengler reactions
Diness, Frederik & Meldal, Morten Peter, 2005, Peptides 2004, Proceedings. p. 208-209Research output: Chapter in Book/Report/Conference proceeding › Book chapter › Research › peer-review
- 2006
- Published
Solid-phase reactions of N-carbamyliminium ions: from amino aldehydes to on-bead GPCR-screening : PH.D. thesis
Diness, Frederik, 2006, Copenhagen: Department of Medical Chemistry, Danish University of Pharmaceutical Sciences. 179 p.Research output: Book/Report › Book › Research
- Published
Solid-phase synthesis of tetrahydro-beta-carbolines and tetrahydroisoquinolines by stereoselective intramolecular N-carbamyliminium Pictet-Spengler reactions
Diness, Frederik & Meldal, Morten Peter, 25 Oct 2006, In: Chemistry: A European Journal. 12, 31, p. 8056-66 11 p.Research output: Contribution to journal › Journal article › Research › peer-review
- 2009
- Published
Imidazolones in diastereoselective cyclization reactions and Cu(II)-catalysed cross-coupling reactions
Diness, Frederik & Meldal, Morten Peter, 20 Jul 2009, In: Chemistry: A European Journal. 15, 29, p. 7044-7 4 p.Research output: Contribution to journal › Journal article › Research › peer-review
- 2010
Ralph F. Hirschmann award address 2009: merger of organic chemistry with peptide diversity
Meldal, Morten Peter, Tornøe, C. W., Nielsen, T. E., Diness, Frederik, Le Quement, S. T., Christensen, C. A., Jensen, J. F., Worm-Leonhard, K., Groth, T., Bouakaz, L., Wu, B., Hagel, G. & Keinicke, L., 2010, In: Biopolymers. 94, 2, p. 161-182 22 p.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Amino acid derived 1,4-dialkyl substituted imidazolones
Diness, Frederik & Meldal, Morten Peter, 11 Mar 2010, In: Biopolymers. 94, 2, p. 236-241Research output: Contribution to journal › Journal article › Research › peer-review
ID: 33654400
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263
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C-Terminally modified peptides via cleavage of the HMBA linker by O-, N- or S-nucleophiles
Research output: Contribution to journal › Journal article › Research › peer-review
Published -
250
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X-ray diffraction data as a source of the vibrational free-energy contribution in polymorphic systems
Research output: Contribution to journal › Journal article › Research › peer-review
Published -
153
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Design and Combinatorial Development of Shield-1 Peptide Mimetics Binding to Destabilized FKBP12
Research output: Contribution to journal › Journal article › Research › peer-review
Published