Birgitte Holst

Birgitte Holst

Guest Researcher


  1. Published

    Molecular basis for agonism in the BB3 receptor: an epitope located on the interface of transmembrane-III, -VI, and -VII

    Gbahou, F., Holst, Birgitte & Schwartz, Thue W., 2010, In: Journal of Pharmacology and Experimental Therapeutics. 333, 1, p. 51-9 8 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  2. Published

    Model-Based Discovery of Synthetic Agonists for the Zn2+-Sensing G-Protein-Coupled Receptor 39 (GPR39) Reveals Novel Biological Functions.

    Frimurer, Thomas Michael, Mende, F., Graae, A., Engelstoft, M. S., Egerod, Kristoffer Lihme, Nygaard, R., Gerlach, L., Hansen, J. B., Schwartz, Thue W. & Holst, Birgitte, 2017, In: Journal of Medicinal Chemistry. 60, 3, p. 886-898 13 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  3. Published

    A gut feeling for obesity: 7TM sensors on enteroendocrine cells

    Engelstoft, M. S., Egerod, Kristoffer Lihme, Holst, Birgitte & Schwartz, Thue W., 2008, In: Cell Metabolism. 8, 6, p. 447-9 2 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  4. Published

    An aromatic region to induce a switch between agonism and inverse agonism at the ghrelin receptor

    Els, S., Schild, E., Petersen, P. S., Kilian, T., Mokrosinski, J., Frimurer, Thomas Michael, Chollet, C., Schwartz, Thue W., Holst, Birgitte & Beck-Sickinger, A. G., 13 Sep 2012, In: Journal of Medicinal Chemistry. 55, 17, p. 7437-49 13 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  5. Published

    Conversion of agonist site to metal-ion chelator site in the ¿2-adrenergic receptor

    Elling, C. E., Thirstrup, K., Holst, Birgitte & Schwartz, Thue W., 1999, In: Proceedings of the National Academy of Science of the United States of America. 96, no. 22, p. 12322-12327

    Research output: Contribution to journalJournal articleResearchpeer-review

  6. Published

    Metal ion site engineering indicates a global toggle switch model for seven-transmembrane receptor activation

    Elling, C. E., Frimurer, T. M., Gerlach, L., Jorgensen, R., Holst, Birgitte & Schwartz, Thue W., 2006, In: Journal of Biological Chemistry. 281, 25, p. 17337-46 9 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  7. Published

    Conversion of agonist site to metal-ion chelator site in the beta(2)-adrenergic receptor

    Elling, C. E., Thirstrup, K., Holst, Birgitte & Schwartz, Thue W., 1999, In: Proceedings of the National Academy of Sciences of the United States of America. 96, 22, p. 12322-7 6 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  8. Published

    GPR119 - a major Enteroendocrine Sensor of Dietary Triglyceride Metabolites Co-acting in Synergy with FFA1 (GPR40)

    Ekberg, J. H., Pedersen, M. H., Kristensen, L. V., Madsen, A. N., Engelstoft, M. S., Husted, Anna Sofie, Sichlau, R., Egerod, Kristoffer Lihme, Timshel, P., Kowalski, T. J., Gribble, F. M., Reiman, F., Hansen, Harald S., Howard, A. D., Holst, Birgitte & Schwartz, Thue W., 25 Oct 2016, In: Endocrinology. 157, 12, p. 4561-4569 9 p., en20161334.

    Research output: Contribution to journalJournal articleResearchpeer-review

  9. Published

    ß-Cell Specific Overexpression of GPR39 Protects against Streptozotocin-Induced Hyperglycemia

    Egerod, Kristoffer Lihme, Jin, C., Petersen, P. S., Wierup, N., Sundler, F., Holst, Birgitte & Schwartz, Thue W., 2011, In: International Journal of Endocrinology. 2011, p. 401258

    Research output: Contribution to journalJournal articleResearchpeer-review

  10. Published

    GPR39 splice variants versus antisense gene LYPD1: expression and regulation in gastrointestinal tract, endocrine pancreas, liver, and white adipose tissue.

    Egerod, Kristoffer Lihme, Holst, Birgitte, Petersen, P. S., Hansen, Jacob B., Mulder, J., Hökfelt, T. & Schwartz, Thue W., 2007, In: Molecular Endocrinology. 21, 7, p. 1685-98 13 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  11. Published

    Dietary fat decreases intestinal levels of the anorectic lipids through a fat sensor

    Diep, T. A., Madsen, A. N., Holst, Birgitte, Kristiansen, M. M., Andersen, N. W., Hansen, S. H. & Hansen, Harald S., 2011, In: The FASEB Journal. 25, 2, p. 765-774

    Research output: Contribution to journalJournal articleResearchpeer-review

  12. Published

    Dietary non-esterified oleic Acid decreases the jejunal levels of anorectic N-acylethanolamines

    Diep, T. A., Madsen, A. N., Krogh-Hansen, S., Al-Shahwani, M., Al-Sabagh, L., Holst, Birgitte & Hansen, Harald S., 2014, In: PloS one. 9, 6, p. 1-7 7 p., e100365.

    Research output: Contribution to journalJournal articleResearchpeer-review

  13. Published

    Proteomics-Based Comparative Mapping of the Secretomes of Human Brown and White Adipocytes Reveals EPDR1 as a Novel Batokine

    Deshmukh, A. S., Peijs, L., Beaudry, J. L., Jespersen, N. Z., Nielsen, C. H., Ma, T., Brunner, A. D., Larsen, T. J., Bayarri-Olmos, R., Prabhakar, B. S., Helgstrand, C., Severinsen, M. C. K., Holst, B., Kjaer, A., Tang-Christensen, M., Sanfridson, A., Garred, P., Privé, G. G., Pedersen, B. K., Gerhart-Hines, Z. & 4 others, Nielsen, S., Drucker, D. J., Mann, Matthias & Schéele, Camilla Charlotte Nielsen, 2019, In: Cell Metabolism. 30, 5, p. 963-975.e7 21 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  14. Published

    Initial Pharmacological Characterization of a Major Hydroxy Metabolite of PF-5190457: Inverse Agonist Activity of PF-6870961 at the Ghrelin Receptor

    Deschaine, S. L., Hedegaard, M. A., Pince, C. L., Farokhnia, M., Moose, J. E., Stock, I. A., Adusumalli, S., Akhlaghi, F., Hougland, J. L., Sulima, A., Rice, K. C., Koob, G. F., Vendruscolo, L. F., Holst, Birgitte & Leggio, L., 2023, In: Journal of Pharmacology and Experimental Therapeutics. 386, 2, p. 117-128 12 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  15. Published

    PHARMACOLOGICAL CHARACTERIZATION OF A GHRELIN RECEPTOR ANTAGONIST/ INVERSE AGONIST, PF-5190457, AND ITS MAJOR ACTIVE HYDROXY METABOLITE

    Deschaine, S. L., Hedegaard, M. A., Sulima, A., Moose, J., Stock, I. A., Hougland, J. L., Akhlaghi, F., Rice, K. C., Holst, Birgitte & Leggio, L., 2021, In: Alcoholism: Clinical and Experimental Research. 45, Supl. 1/SI, p. 146A-146A 1 p., 674.

    Research output: Contribution to journalConference abstract in journalResearchpeer-review

  16. Published

    Synthesis and in Vitro Evaluation of Stabilized and Selective Neuromedin U-1 Receptor Agonists

    De Prins, A., Martin, C., Van Wanseele, Y., Tömböly, C., Tourwé, D., Caveliers, V., Holst, Birgitte, Van Eeckhaut, A., Rosenkilde, M. M., Smolders, I. & Ballet, S., 10 May 2018, In: ACS Medicinal Chemistry Letters. 9, 5, p. 496-501 6 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  17. Published

    Development of potent and proteolytically stable human neuromedin U receptor agonists

    De Prins, A., Martin, C., Van Wanseele, Y., Skov, Louise Julie, Tömböly, C., Tourwé, D., Caveliers, V., Van Eeckhaut, A., Holst, Birgitte, Rosenkilde, Mette, Smolders, I. & Ballet, S., 20 Jan 2018, In: European Journal of Medicinal Chemistry. 144, p. 887-897 11 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  18. Published

    Hepatic NAD+ levels and NAMPT abundance are unaffected during prolonged high-fat diet consumption in C57BL/6JBomTac mice

    Dall, M., Penke, M., Sulek, K., Matz-Soja, M., Holst, Birgitte, Garten, A., Kiess, W. & Treebak, Jonas Thue, 2018, In: Molecular and Cellular Endocrinology. 473, p. 245-256 12 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  19. Published

    Neuromedin U inhibits food intake partly by inhibiting gastric emptying

    Dalbøge, L. S., Pedersen, S. L., Secher, T., Holst, Birgitte, Vrang, N. & Jelsing, J., Jul 2015, In: Peptides. 69, p. 56-65 10 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  20. Published

    L-Arginine improves multiple physiological parameters in mice exposed to diet-induced metabolic disturbances

    Clemmensen, Christoffer, Madsen, A. N., Smajilovic, S., Holst, Birgitte & Bräuner, Hans, 2012, In: Amino Acids. 43, 3, p. 1265-1275

    Research output: Contribution to journalJournal articleResearchpeer-review

  21. Published

    Increased susceptibility to diet-induced obesity in GPRC6A receptor knockout mice

    Clemmensen, Christoffer, Smajilovic, S., Madsen, A. N., Klein, A. B., Holst, Birgitte & Bräuner, Hans, 2013, In: Journal of Endocrinology. 217, 2, p. 151-60 10 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  22. Published

    The Apolipoprotein M/S1P Axis Controls Triglyceride Metabolism and Brown Fat Activity

    Christoffersen, Christina, Federspiel, C. K., Borup, A., Christensen, P. M., Madsen, A. N., Heine, M., Nielsen, C. H., Kjaer, A., Holst, Birgitte, Heeren, J. & Nielsen, L. B., 2 Jan 2018, In: Cell Reports. 22, 1, p. 175-188

    Research output: Contribution to journalJournal articleResearchpeer-review

  23. Published

    LEAP2 is associated with cardiometabolic markers but is unchanged by antidiabetic treatment in people with prediabetes

    Byberg, Sarah, Blond, Martin Bæk, Holm, Stephanie Kjærulff, Amadid, H., Nielsen, L. B., Clemmensen, K. K. B., Færch, K. & Holst, Birgitte, 2023, In: American journal of physiology. Endocrinology and metabolism. 325, 3, p. E244-E251

    Research output: Contribution to journalJournal articleResearchpeer-review

  24. Published

    Increased meal-induced neurotensin response predicts successful maintenance of weight loss: Data from a randomized controlled trial

    Brethvad, Annemette Overgaard, Zakariassen, Hannah Louise, Holt, Joachim, Lundgren, J. R., Jakobsen, A., Hartmann, Bolette, Lehmann, E. W., Kissow, Hannelouise, Holst, Jens Juul, Madsbad, Sten, Torekov, Signe Sørensen & Holst, Birgitte, 2023, In: Metabolism: Clinical and Experimental. 143, 8 p., 155534.

    Research output: Contribution to journalJournal articleResearchpeer-review

  25. Published

    Pannexin-2-deficiency sensitizes pancreatic beta-cells to cytokine-induced apoptosis in vitro and impairs glucose tolerance in vivo

    Berchtold, L. A., Miani, M., Diep, T. A., Madsen, A. N., Cigliola, V., Colli, M., Miskovic Krivokapic, Jelena, Pociot, Flemming, Eizirik, D. L., Meda, P., Holst, Birgitte, Billestrup, Nils & Storling, J., 2017, In: Molecular and Cellular Endocrinology. 448, p. 108-121 4 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

ID: 9886