Hans Bräuner
Prodekan for forskning
Faculty Service
Blegdamsvej 3
2200 København N.
- 2005
- Published
Synthesis of novel N1-substituted bicyclic pyrazole amino acids and evaluation of their interaction with glutamate receptors
Conti, P., Grazioso, G., di Ventimiglia, S. J., Pinto, A., Roda, G., Madsen, Ulf, Bräuner, Hans, Nielsen, Birgitte, Costagli, C. & Galli, A., Jun 2005, In: Chemistry & Biodiversity. 2, 6, p. 748-57Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Deorphanization of GPRC6A: a promiscuous L-alpha-amino acid receptor with preference for basic amino acids
Wellendorph, Petrine, Hansen, K. B., Balsgaard, A., Greenwood, J. R., Egebjerg, J. & Bräuner, Hans, Mar 2005, In: Molecular Pharmacology. 67, 3, p. 589-97Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Rigid nonproteinogenic cyclic amino acids as ligands for glutamate receptors: trans-tris(homoglutamic) acids
Meyer, U., Bisel, P., Bräuner, Hans, Madsen, Ulf, Höfner, G., Wanner, K. T. & Frahm, A. W., Feb 2005, In: Chirality. 17, 2, p. 99-107Research output: Contribution to journal › Journal article › Research › peer-review
- Published
GABA and Glutamate Receptor Ligands and Their Therapeutic Potential in CNS Disorders
Madsen, Ulf, Bräuner, Hans, Greenwood, J. R., Johansen, Tommy Nørskov, Krogsgaard-Larsen, Povl, Liljefors, T., Nielsen, M. & Frølund, Bente, 27 Jan 2005, Drug Discovery Handbook. John Wiley & Sons, Inc., p. 797-907 111 p.Research output: Chapter in Book/Report/Conference proceeding › Book chapter › Research › peer-review
- Published
4-Alkylated homoibotenic acid (HIBO) analogues: versatile pharmacological agents with diverse selectivity profiles towards metabotropic and ionotropic glutamate receptor subtypes
Madsen, Ulf, Pickering, Darryl S, Nielsen, Birgitte & Bräuner, Hans, 2005, In: Neuropharmacology. 49 Suppl 1, p. 114-9 5 p.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Azetidinic amino acids: stereocontrolled synthesis and pharmacological characterization as ligands for glutamate receptors and transporters
Bräuner, Hans, Bunch, Lennart, Chopin, N., Couty, F., Evano, G., Jensen, Anders A., Kusk, M. L., Nielsen, Birgitte & Rabasso, N., 2005, In: Organic & Biomolecular Chemistry. 3, 21, p. 3926-36 11 p.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Chemoenzymatic synthesis of a series of 4-substituted glutamate analogues and pharmacological characterization at human glutamate transporters subtypes 1-3
Alaux, S., Kusk, M., Sagot, E., Bolte, J., Jensen, Anders A., Bräuner, Hans, Gefflaut, T. & Bunch, Lennart, 2005, In: Journal of Medicinal Chemistry. 48, 25, p. 7980-92 13 p.Research output: Contribution to journal › Journal article › Research › peer-review
- 2004
- Published
Design, synthesis, and pharmacological characterization of novel, potent NMDA receptor antagonists
Conti, P., De Amici, M., Grazioso, G., Roda, G., Barberis Negra, F. F., Nielsen, Birgitte, Stensbøl, T. B., Madsen, Ulf, Bräuner, Hans, Frydenvang, Karla Andrea, De Sarro, G., Toma, L. & De Micheli, C., 30 Dec 2004, In: Journal of Medicinal Chemistry. 47, 27, p. 6740-8 9 p.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
The respective N-hydroxypyrazole analogues of the classical glutamate receptor ligands ibotenic acid and (RS)-2-amino-2-(3-hydroxy-5-methyl-4-isoxazolyl)acetic acid
Clausen, Rasmus Prætorius, Hansen, K. B., Calí, P., Nielsen, Birgitte, Greenwood, J. R., Begtrup, M., Egebjerg, J. & Bräuner, Hans, 19 Sep 2004, In: European Journal of Pharmacology. 499, 1-2, p. 35-44 10 p.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Mutation-induced quisqualic acid and ibotenic acid affinity at the metabotropic glutamate receptor subtype 4: ligand selectivity results from a synergy of several amino acid residues
Hermit, M. B., Greenwood, J. R. & Bräuner, Hans, 13 Aug 2004, In: Journal of Biological Chemistry. 279, 33, p. 34811-7Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Synthesis, theoretical and structural analyses, and enantiopharmacology of 3-carboxy homologs of AMPA
Brehm, L., Greenwood, J. R., Sløk, F. A., Holm, M. M., Nielsen, Birgitte, Geneser, U., Stensbøl, T. B., Bräuner, Hans, Begtrup, M., Egebjerg, J. & Krogsgaard-Larsen, Povl, Aug 2004, In: Chirality. 16, 7, p. 452-66Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Molecular cloning, expression, and sequence analysis of GPRC6A, a novel family C G-protein-coupled receptor
Wellendorph, Petrine & Bräuner, Hans, 23 Jun 2004, In: Gene. 335, p. 37-46Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Ibotenic acid and thioibotenic acid: a remarkable difference in activity at group III metabotropic glutamate receptors
Hermit, M. B., Greenwood, J. R., Nielsen, Birgitte, Bunch, Lennart, Jørgensen, Charlotte Grube, Vestergaard, H. T., Stensbøl, T. B., Sanchez, C., Krogsgaard-Larsen, Povl, Madsen, Ulf & Bräuner, Hans, 23 Feb 2004, In: European Journal of Pharmacology. 486, 3, p. 241-50Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Carbamoylcholine homologs: synthesis and pharmacology at nicotinic acetylcholine receptors
Jensen, Anders A., Mikkelsen, I. B., Frølund, Bente, Frydenvang, Karla Andrea, Brehm, L., Jaroszewski, J. W., Bräuner, Hans, Falch, E. & Krogsgaard-Larsen, Povl, 2004, In: European Journal of Pharmacology. 497, 2, p. 125-37 13 p.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Fluorescensbaseret farmakologi
Jensen, Anders A., Strange, M. & Bräuner, Hans, 2004, In: Dansk Kemi 83. p. 29 31 p.Research output: Contribution to journal › Journal article › Communication
- Published
Pharmacological characterization of human excitatory amino acid transporters EAAT1, EAAT2 and EAAT3 in a fluorescence-based membrane potential assay
Jensen, Anders A. & Bräuner, Hans, 2004, In: Biochemical Pharmacology. 67, 11, p. 2115-27 13 p.Research output: Contribution to journal › Journal article › Research › peer-review
- 2003
- Published
Design of Cyclopentaisoxazoline Amino Acids as Conformationally Constrained Agonists at Glutamate Receptors
Conti, P., De Amici, M., Grazioso, G., Roda, G., Stensbøl, T. B., Bräuner, Hans, Madsen, Ulf, Toma, L. & De Micheli, C., 14 Nov 2003, In: European Journal of Organic Chemistry. 22, p. 4455-4461 7 p.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Specific gamma-hydroxybutyrate-binding sites but loss of pharmacological effects of gamma-hydroxybutyrate in GABA-B1-deficient mice
Kaupmann, K., Cryan, J. F., Wellendorph, Petrine, Mombereau, C., Sansig, G., Klebs, K., Schmutz, M., Froestl, W., van der Putten, H., Mosbacher, J., Bräuner, Hans, Waldmeier, P. & Bettler, B., Nov 2003, In: European Journal of Neuroscience. 18, 10, p. 2722-30Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Three distinct epitopes on the extracellular face of the glucagon receptor determine specificity for the glucagon amino terminus
Runge, S., Gram, C., Bräuner, Hans, Madsen, K., Knudsen, L. B. & Wulff, B. S., 25 Jul 2003, In: Journal of Biological Chemistry. 278, 30, p. 28005-10Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Synthesis and anticonvulsant activity of novel bicyclic acidic amino acids
Conti, P., De Amici, M., Joppolo Di Ventimiglia, S., Stensbøl, T. B., Madsen, Ulf, Bräuner, Hans, Russo, E., De Sarro, G., Bruno, G. & De Micheli, C., 3 Jul 2003, In: Journal of Medicinal Chemistry. 46, 14, p. 3102-8Research output: Contribution to journal › Journal article › Research › peer-review
- Published
(S)-2-Amino-3-(3-hydroxy-7,8-dihydro-6H-cyclohepta[d]isoxazol-4-yl)propionic acid, a potent and selective agonist at the GluR5 subtype of ionotropic glutamate receptors. Synthesis, modeling, and molecular pharmacology
Brehm, L., Greenwood, J. R., Hansen, K. B., Nielsen, Birgitte, Egebjerg, J., Stensbøl, T. B., Bräuner, Hans, Sløk, F. A., Kronborg, T. T. A. & Krogsgaard-Larsen, Povl, 10 Apr 2003, In: Journal of Medicinal Chemistry. 46, 8, p. 1350-8Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Different domains of the glucagon and glucagon-like peptide-1 receptors provide the critical determinants of ligand selectivity
Runge, S., Wulff, B. S., Madsen, K., Bräuner, Hans & Knudsen, L. B., Mar 2003, In: British Journal of Pharmacology. 138, 5, p. 787-94Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Positive allosteric modulation of the human metabotropic glutamate receptor 4 (hmGluR4) by SIB-1893 and MPEP
Mathiesen, Jesper M., Svendsen, N., Bräuner, Hans, Thomsen, C. & Ramirez, M. T., Mar 2003, In: British Journal of Pharmacology. 138, 6, p. 1026-30Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Design of novel conformationally restricted analogues of glutamic acid
Conti, P., De Amici, M., Roda, G., Vistoli, G., Stensbøl, T. B., Bräuner, Hans, Madsen, Ulf, Toma, L. & De Micheli, C., 24 Feb 2003, In: Tetrahedron. 59, 9, p. 1443-1452 10 p.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Carbamoylcholine homologs: novel and potent agonists at neuronal nicotinic acetylcholine receptors
Jensen, Anders A., Frølund, Bente, Bräuner, Hans, Falch, E. & Krogsgaard-Larsen, Povl, 2003, In: Molecular Pharmacology. 64, 4, p. 865-75 11 p.Research output: Contribution to journal › Journal article › Research › peer-review
ID: 1302910
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