Biased agonism of clinically approved μ-opioid receptor agonists and TRV130 is not controlled by binding and signaling kinetics

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  • Mie Fabricius Pedersen
  • Tomasz Marcin Wrobel
  • Märcher-Rørsted, Emil
  • Daniel Sejer Pedersen
  • Thor Christian Møller
  • Federica Gabriele
  • Henrik Pedersen
  • Dariusz Matosiuk
  • Simon Richard Foster
  • Michel Bouvier
  • Bräuner, Hans
Original languageEnglish
Article number107718
JournalNeuropharmacology
Volume166
Number of pages13
ISSN0028-3908
DOIs
Publication statusPublished - 2020

    Research areas

  • Biased agonism, Binding kinetics, mu-opioid receptor, Oliceridine ((R)-TRV130)

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