Christian Adam Olsen

Christian Adam Olsen

Professor


  1. Published

    Hydroxamic acid-modified peptide microarrays for profiling isozyme-selective interactions and inhibition of histone deacetylases

    Moreno Yruela, Carlos, Bæk, M., Vrsanova, A., Schulte, C., Maric, H. M. & Olsen, Christian Adam, 4 Jan 2021, In: Nature Communications. 12, 1

    Research output: Contribution to journalJournal articleResearchpeer-review

  2. Published

    Kinetic Characterization of Inhibitors of Histone Deacetylases (HDACs) and Sirtuins

    Moreno Yruela, Carlos, Madsen, A. S. & Olsen, Christian Adam, 2019, 14 p.

    Research output: Working paperPreprintResearch

  3. Published

    Synthesis of Trifluoromethyl Ketone Containing Amino Acid Building Blocks for the Preparation of Peptide-Based Histone Deacetylase (HDAC) Inhibitors

    Moreno Yruela, Carlos & Olsen, Christian Adam, 2018, In: Synthesis. 50, 20, p. 4037-4046

    Research output: Contribution to journalJournal articleResearchpeer-review

  4. Published

    Selective inhibitors of SIRT2 regulate perinuclear α-tubulin acetylation, migration, and invasion of breast cancer cells

    Nielsen, A. L., Rajabi, N., Kudo, N., Jørgensen, Kathrine Lundø, Fontenas, M., Lucidi, A., Madsen, A. S., Yoshida, M. & Olsen, Christian Adam, 2020, In: bioRxiv. 26 p.

    Research output: Contribution to journalJournal articleResearch

  5. Published

    Mechanism-based inhibitors of SIRT2: structure–activity relationship, X-ray structures, target engagement, regulation of α-tubulin acetylation and inhibition of breast cancer cell migration

    Nielsen, A. L., Rajabi, N., Kudo, N., Jørgensen, Kathrine Lundø, Moreno Yruela, Carlos, Bæk, M., Fontenas, M., Lucidi, A., Madsen, A. S., Yoshida, M. & Olsen, Christian Adam, 2021, In: RSC Chemical Biology. 2, p. 612-626

    Research output: Contribution to journalJournal articleResearchpeer-review

  6. Published

    Finding the gas pedal on a slow sirtuin

    Nielsen, A. L. & Olsen, Christian Adam, 31 Jan 2020, In: Journal of Biological Chemistry. 295, p. 400-401

    Research output: Contribution to journalLiterature reviewResearchpeer-review

  7. Published

    Potent and selective inhibition of sirtuin 2 deacylation

    Nielsen, A. L., Rajabi, N., Madsen, A. & Olsen, Christian Adam, 19 Aug 2018.

    Research output: Contribution to conferenceConference abstract for conferenceResearchpeer-review

  8. Published

    An NAD+-Dependent Sirtuin Depropionylase and Deacetylase (Sir2La) from the Probiotic Bacterium Lactobacillus acidophilus NCFM

    Olesen, S., Rajabi, N., Svensson, B., Olsen, Christian Adam & Madsen, A. S., 4 Jun 2018, In: Biochemistry. 57, 26, p. 3903-3915

    Research output: Contribution to journalJournal articleResearchpeer-review

  9. Published

    Antimicrobial, hemolytic, and cytotoxic activities of β-peptoid- peptide hybrid oligomers: Improved properties compared to natural AMPs (ChemBioChem (2010) 11, (152-160))

    Olsen, Christian Adam, Ziegler, H. L., Nielsen, Hanne Mørck, Frimodt-Møller, N., Jaroszewski, J. W. & Franzyk, Henrik, 16 Aug 2010, In: ChemBioChem. 11, 12, 1 p.

    Research output: Contribution to journalComment/debateResearchpeer-review

  10. Published

    Side-chain-anchored N(alpha)-Fmoc-Tyr-OPfp for bidirectional solid-phase synthesis

    Olsen, Christian Adam, Jørgensen, M., Hansen, S. H., Witt, M., Jaroszewski, J. W. & Franzyk, Henrik, 2005, In: Organic Letters. 7, 9, p. 1703-6 4 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

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