Probing the Bioactive Conformation of an Archetypal Natural Product HDAC Inhibitor with Conformationally Homogeneous Triazole-Modified Cyclic Tetrapeptides

Research output: Contribution to journalJournal articleResearchpeer-review

Original languageEnglish
JournalAngewandte Chemie International Edition
Volume48
Issue number26
Pages (from-to)4718-4724
ISSN1433-7851
DOIs
Publication statusPublished - 2009

    Research areas

  • cyclic peptides, drug design, enzyme inhibitors, structure-activity relationships, triazoles

ID: 112999511