Michael Lückmann

Michael Lückmann

senior adviser


Publication year:
  1. 2019
  2. Published

    Molecular dynamics-guided discovery of an ago-allosteric modulator for GPR40/FFAR1. / Lückmann, Michael; Trauelsen, Mette; Bentsen, Marie A; Nissen, Tinne A D; Martins, Joao; Fallah, Zohreh; Nygaard, Mads M; Papaleo, Elena; Lindorff-Larsen, Kresten; Schwartz, Thue W; Frimurer, Thomas M.

    In: Proceedings of the National Academy of Sciences of the United States of America, Vol. 116, No. 14, 02.04.2019, p. 7123-7128.

    Research output: Contribution to journalJournal articleResearchpeer-review

  3. 2018
  4. Published

    Ligand-selective small molecule modulators of the constitutively active vGPCR US28. / Amarandi, Roxana-Maria; Luckmann, Michael; Melynis, Motiejus; Jakobsen, Mette H.; Fallah, Zohreh; Spiess, Katja; Hjorto, Gertrud M.; Pui, Aurel; Frimurer, Thomas M.; Rosenkilde, Mette M.

    In: European Journal of Medicinal Chemistry, Vol. 155, 2018, p. 244-254.

    Research output: Contribution to journalJournal articleResearchpeer-review

  5. Published

    Structure-Activity Investigations and Optimisations of Non-metabolite Agonists for the Succinate Receptor 1. / Rexen Ulven, Elisabeth; Trauelsen, Mette; Brvar, Matjaz; Lückmann, Michael; Bielefeldt, Line Ø; Jensen, Lisa K I; Schwartz, Thue W; Frimurer, Thomas M.

    In: Scientific Reports, Vol. 8, No. 1, 10010, 2018, p. 1-18.

    Research output: Contribution to journalJournal articleResearchpeer-review

  6. Published

    The HETE Is on FFAR1 and Pancreatic Islet Cells. / Trauelsen, Mette; Lückmann, Michael; Frimurer, Thomas M; Schwartz, Thue W.

    In: Cell Metabolism, Vol. 27, No. 2, 2018, p. 273-275.

    Research output: Contribution to journalJournal articleResearchpeer-review

  7. Published

    Translating biased signaling in the ghrelin receptor system into differential in vivo functions. / Mende, Franziska; Hundahl, Cecilie; Plouffe, Bianca; Skov, Louise Julie; Sivertsen, Bjørn; Madsen, Andreas Nygaard; Lückmann, Michael; Diep, Thi Ai; Offermanns, Stefan; Frimurer, Thomas Michael; Bouvier, Michel; Holst, Birgitte.

    In: Proceedings of the National Academy of Sciences of the United States of America, Vol. 115, No. 43, 2018, p. E10255-E10264.

    Research output: Contribution to journalJournal articleResearchpeer-review

  8. 2017
  9. Published

    Biased agonism and allosteric modulation of GPR183- a 7TM receptor also known as EBV-induced EBI2. / Daugvilaite, Viktorija; Madsen, Christian Medom; Lückmann, Michael; Castello Echeverria, Clara; Sailer, Andreas Walter; Frimurer, Thomas Michael; Rosenkilde, Mette Marie; Benned-Jensen, Tau.

    In: British Journal of Pharmacology, Vol. 174, No. 13, 2017, p. 2031–2042.

    Research output: Contribution to journalJournal articleResearchpeer-review

  10. Published

    Structure-based discovery of novel US28 small molecule ligands with different modes of action. / Lückmann, Michael; Amarandi, Roxana-Maria; Papargyri, Natalia; Jakobsen, Mette H; Christiansen, Elisabeth; Jensen, Lars Juhl; Pui, Aurel; Schwartz, Thue W.; Rosenkilde, Mette Marie; Frimurer, Thomas Michael.

    In: Chemical Biology & Drug Design, Vol. 89, No. 3, 2017, p. 289–296.

    Research output: Contribution to journalJournal articleResearchpeer-review

  11. 2016
  12. Published

    Role of Conserved Disulfide Bridges and Aromatic Residues in Extracellular Loop 2 of Chemokine Receptor CCR8 for Chemokine and Small Molecule Binding. / Barington, Line; Rummel, Pia C; Lückmann, Michael; Pihl, Heidi; Larsen, Olav; Daugvilaite, Viktorija; Johnsen, Anders H.; Frimurer, Thomas M; Karlshøj, Stefanie; Rosenkilde, Mette M.

    In: The Journal of Biological Chemistry, Vol. 291, No. 31, 19.05.2016, p. 16208-16220.

    Research output: Contribution to journalJournal articleResearchpeer-review

  13. Published
  14. 2015
  15. Published

    Optimisation of in silico derived 2-aminobenzimidazole hits as unprecedented selective kappa opioid receptor agonists. / Sasmal, Pradip K; Krishna, C Vamsee; Sudheerkumar Adabala, S; Rawoof, khaji Abdul; Thadi, Amima; Sukumar, K Pawan; Cheera, Srisailam; Abbineni, Chandrasekhar; Rao, K V L Narasimha; Prasanthi, A; Nijhawan, Kamal; Jaleel, Mahaboobi; Ramachandran Iyer, Lakshmi; Chaitanya, T Krishna; Tiwari, Nirbhay Kumar; Krishna, N Lavanya; Potluri, Vijay; Khanna, Ish; Frimurer, Thomas M; Lückmann, Michael; Rist, Øystein; Elster, Lisbeth; Högberg, Thomas.

    In: Bioorganic & Medicinal Chemistry Letters, Vol. 25, No. 4, 15.02.2015, p. 887-92.

    Research output: Contribution to journalJournal articleResearchpeer-review

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