David E. Gloriam

David E. Gloriam

Professor


  1. Published

    Identification and characterization of small molecular NPR-B receptor antagonists. / Andresen, Henriette; Moltzau, Lise; Fagerheim, Steffen; Gloriam, David; Bach, Trond; Levy, Finn.

    In: BMC Pharmacology and Toxicology, Vol. 16, No. Suppl 1, 01.01.2015, p. A70.

    Research output: Contribution to journalJournal articleCommunication

  2. Published

    Creating a specialist protein resource network: a meeting report for the protein bioinformatics and community resources retreat. / Babbitt, Patricia C.; Bagos, Pantelis G.; Bairoch, Amos; Bateman, Alex; Chatonnet, Arnaud; Chen, Mark Jinan; Craik, David J.; Finn, Robert D.; Gloriam, David; Haft, Daniel H.; Henrissat, Bernard; Holliday, Gemma L.; Isberg, Vignir; Kaas, Quentin; Landsman, David; Lenfant, Nicolas; Manning, Gerard; Nagano, Nozomi; Srinivasan, Narayanaswamy; O’Donovan, Claire; Pruitt, Kim D.; Sowdhamini, Ramanathan; Rawlings, Neil D.; Saier, Milton H.; Sharman, Joanna L.; Spedding, Michael; Tsirigos, Konstantinos D.; Vastermark, Ake; Vriend, Gerrit.

    In: Database, Vol. 2015, 18.05.2015, p. 1-5.

    Research output: Contribution to journalJournal articleResearchpeer-review

  3. Comprehensive repertoire and phylogenetic analysis of the G protein-coupled receptors in human and mouse. / Bjarnadóttir, Thóra K; Gloriam, David E.; Hellstrand, Sofia H; Kristiansson, Helena; Fredriksson, Robert; Schiöth, Helgi B.

    In: Genomics, Vol. 88, No. 3, 09.2006, p. 263-73.

    Research output: Contribution to journalJournal articleResearchpeer-review

  4. The human and mouse repertoire of the adhesion family of G-protein-coupled receptors. / Bjarnadóttir, Thóra K; Fredriksson, Robert; Höglund, Pär J; Gloriam, David E.; Lagerström, Malin C; Schiöth, Helgi B.

    In: Genomics, Vol. 84, No. 1, 07.2004, p. 23-33.

    Research output: Contribution to journalJournal articleResearchpeer-review

  5. Published

    Minimum information about a protein affinity reagent (MIAPAR). / Bourbeillon, Julie; Orchard, Sandra; Benhar, Itai; Borrebaeck, Carl; de Daruvar, Antoine; Dübel, Stefan; Frank, Ronald; Gibson, Frank; Gloriam, David Erik Immanuel; Haslam, Niall; Hiltker, Tara; Humphrey-Smith, Ian; Hust, Michael; Juncker, David; Koegl, Manfred; Konthur, Zoltàn; Korn, Bernhard; Krobitsch, Sylvia; Muyldermans, Serge; Nygren, Per-Åke; Palcy, Sandrine; Polic, Bojan; Rodriguez, Henry; Sawyer, Alan; Schlapshy, Martin; Snyder, Michael; Stoevesandt, Oda; Taussig, Michael J; Templin, Markus; Uhlen, Matthias; van der Maarel, Silvere; Wingren, Christer; Hermjakob, Henning; Sherman, David.

    In: Nature Biotechnology, Vol. 28, No. 7, 2010, p. 650-653.

    Research output: Contribution to journalJournal articleResearch

  6. E-pub ahead of print

    G protein-coupled receptor pharmacology-The next generation. / Bräuner-Osborne, Hans; Rosenkilde, Mette M; Gether, Ulrik; Gloriam, David E.

    In: Basic & Clinical Pharmacology & Toxicology, 13.07.2019.

    Research output: Contribution to journalJournal articleResearchpeer-review

  7. Published

    Structure-Activity Relationships and Identification of Optmized CC-Chemokine Receptor CCR1, 5, and 8 Metal-Ion Chelators. / Chalikiopoulos, Alexander; Thiele, Stefanie; Malmgaard-Clausen, Mikkel; Rydberg, Patrik; Isberg, Vignir; Ulven, Trond; Frimurer, Thomas M; Rosenkilde, Mette M; Gloriam, David E.

    In: Journal of Chemical Information and Modeling, Vol. 53, No. 11, 25.11.2013, p. 2863-73.

    Research output: Contribution to journalJournal articleResearchpeer-review

  8. Published

    Applying label-free dynamic mass redistribution assay for studying endogenous FPR1 receptor signalling in human neutrophils. / Christensen, Hanna B; Gloriam, David E; Pedersen, Daniel Sejer; Cowland, Jack B; Borregaard, Niels; Bräuner-Osborne, Hans.

    In: Journal of Pharmacological and Toxicological Methods, Vol. 88, No. Pt 1, 15.07.2017, p. 72-78.

    Research output: Contribution to journalJournal articleResearchpeer-review

  9. Published

    Present perspectives on the automated classification of the G-protein coupled receptors (GPCRs) at the protein sequence level. / Davies, Matthew N; Gloriam, David E; Secker, Andrew; Freitas, Alex A.; Timmis, Jon; Flower, Darren R.

    In: Current Topics in Medicinal Chemistry, Vol. 11, No. 15, 2011, p. 1994-2009.

    Research output: Contribution to journalJournal articleResearchpeer-review

  10. Published

    In silico identification of novel G protein-coupled receptors. / Davies, Matthew N; Gloriam, David E; Flower, Darren R.

    Methods for the discovery and characterization of G protein-coupled receptors. ed. / Craig W Stevens. Vol. 60 New York : Humana Press, 2011. p. 3-18 (Neuromethods, Vol. 60).

    Research output: Chapter in Book/Report/Conference proceedingBook chapterResearch

  11. Proteomic applications of automated GPCR classification. / Davies, Matthew N; Gloriam, David E.; Secker, Andrew; Freitas, Alex A; Mendao, Miguel; Timmis, Jon; Flower, Darren R.

    In: Proteomics, Vol. 7, No. 16, 08.2007, p. 2800-14.

    Research output: Contribution to journalJournal articleResearchpeer-review

  12. Published

    Development of a human vasopressin V1a-receptor antagonist from an evolutionary-related insect neuropeptide. / Di Giglio, Maria Giulia; Muttenthaler, Markus; Harpsøe, Kasper; Liutkeviciute, Zita; Keov, Peter; Eder, Thomas; Rattei, Thomas; Arrowsmith, Sarah; Wray, Susan; Marek, Ales; Elbert, Tomas; Alewood, Paul F; Gloriam, David E; Gruber, Christian W.

    In: Scientific Reports, Vol. 7, 41002, 01.02.2017.

    Research output: Contribution to journalJournal articleResearchpeer-review

  13. Published

    A new crystal structure fragment-based pharmacophore method for G protein-coupled receptors. / Fidom, Kimberley; Isberg, Vignir; Hauser, Alexander Sebastian; Mordalski, Stefan; Lehto, Thomas; Bojarski, Andrzej J; Gloriam, David E.

    In: Methods, Vol. 71, 01.2015, p. 104-112.

    Research output: Contribution to journalJournal articleResearchpeer-review

  14. Published

    Selectivity determinants of GPCR-G-protein binding. / Flock, Tilman; Hauser, Alexander S; Lund, Nadia; Gloriam, David E; Balaji, Santhanam; Babu, M Madan.

    In: Nature, Vol. 545, No. 7654, 18.05.2017, p. 317-322.

    Research output: Contribution to journalJournal articleResearchpeer-review

  15. Published

    Identification of Histamine H3 Receptor Ligands Using a New Crystal Structure Fragment-based Method. / Frandsen, Ida Osborn; Boesgaard, Michael W; Fidom, Kimberley; Hauser, Alexander S; Isberg, Vignir; Bräuner-Osborne, Hans; Wellendorph, Petrine; Gloriam, David E.

    In: Scientific Reports, Vol. 7, No. 1, 4829, 06.07.2017.

    Research output: Contribution to journalJournal articleResearchpeer-review

  16. Seven evolutionarily conserved human rhodopsin G protein-coupled receptors lacking close relatives. / Fredriksson, Robert; Höglund, Pär J; Gloriam, David E.; Lagerström, Malin C; Schiöth, Helgi B.

    In: F E B S Letters, Vol. 554, No. 3, 20.11.2003, p. 381-8.

    Research output: Contribution to journalJournal articleResearchpeer-review

  17. There exist at least 30 human G-protein-coupled receptors with long Ser/Thr-rich N-termini. / Fredriksson, Robert; Gloriam, David E.; Höglund, Pär J; Lagerström, Malin C; Schiöth, Helgi B.

    In: Biochemical and Biophysical Research Communications, Vol. 301, No. 3, 14.02.2003, p. 725-34.

    Research output: Contribution to journalJournal articleResearchpeer-review

  18. Published

    Probing the Existence of a Metastable Binding Site at the β2-Adrenergic Receptor with Homobivalent Bitopic Ligands. / Gaiser, Birgit I; Danielsen, Mia; Marcher-Rørsted, Emil; Røpke Jørgensen, Kira; Wróbel, Tomasz M; Frykman, Mikael; Johansson, Henrik; Bräuner-Osborne, Hans; Gloriam, David E; Mathiesen, Jesper Mosolff; Sejer Pedersen, Daniel.

    In: Journal of Medicinal Chemistry, Vol. 62, No. 17, 12.09.2019, p. 7806-7839.

    Research output: Contribution to journalJournal articleResearchpeer-review

  19. Published

    A ligand's view of target similarity : chemogenomic binding site-directed techniques for drug discovery. / Garland, Stephen L; Gloriam, David E.

    In: Current Topics in Medicinal Chemistry, Vol. 11, No. 15, 2011, p. 1872-1881.

    Research output: Contribution to journalJournal articleResearchpeer-review

  20. Published

    Methods for the successful application of chemogenomics to GPCR drug design. / Garland, Stephen L (Editor); Gloriam, David E (Editor).

    In: Current Topics in Medicinal Chemistry, Vol. 11, No. 15, 2011, p. 1870-1871.

    Research output: Contribution to journalEditorialResearch

  21. Published

    Five-membered N-heterocyclic Scaffolds as Novel Amino Bioisosteres at -Aminobutyric Acid (GABA) Type A Receptors and GABA Transporters. / Giraudo, Alessandro; Krall, Jacob; Bavo, Francesco; Nielsen, Birgitte; Kongstad, Kenneth Thermann; Rolando, Barbara; De Blasio, Rosella; Gloriam, David E; Löffler, Rebekka; Thiesen, Louise; Harpsøe, Kasper; Frydenvang, Karla; Boschi, Donatella; Wellendorph, Petrine; Lolli, Marco L; Jensen, Anders A.; Frølund, Bente.

    In: Journal of Medicinal Chemistry, Vol. 62, No. 12, 27.06.2019, p. 5797-5809.

    Research output: Contribution to journalJournal articleResearchpeer-review

  22. Published

    Bigger is better in virtual drug screens. / Gloriam, David E.

    In: Nature, Vol. 566, No. 7743, 02.2019, p. 193-194.

    Research output: Contribution to journalJournal articleResearchpeer-review

  23. Published

    How can I teach to maximize the learning of “Roberts” (slow/nonambitious) and “Susans” (fast/ambitious)? Improving University Science Teaching and Learning - Pedagogical Projects 2008. / Gloriam, David E.

    Improving University Science Teaching and Learning - Pedagogical Projects 2008. ed. / Frederik V. Christiansen; Camilla Rump; Lise Degn. Vol. 1 København : Department of Science Education, University of Copenhagen, Denmark, 2008. p. 227-244.

    Research output: Chapter in Book/Report/Conference proceedingBook chapterEducation

  24. The G protein-coupled receptor subset of the rat genome. / Gloriam, David E.; Fredriksson, Robert; Schiöth, Helgi B.

    In: B M C Genomics, Vol. 8, 2007, p. 338.

    Research output: Contribution to journalJournal articleResearchpeer-review

  25. Published

    Chemogenomic discovery of allosteric antagonists at the GPRC6A receptor. / Gloriam, David E.; Wellendorph, Petrine; Johansen, Lars Dan; Thomsen, Alex Rojas Bie; Phonekeo, Karina; Pedersen, Daniel Sejer; Bräuner-Osborne, Hans.

    In: Chemistry & Biology, Vol. 18, No. 11, 23.11.2011, p. 1489-1498.

    Research output: Contribution to journalJournal articleResearchpeer-review

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