Kristian Strømgaard

Kristian Strømgaard

Professor


  1. 2003
  2. Published

    Modification of the philanthotoxin-343 polyamine moiety results in different structure-activity profiles at muscle nicotinic ACh, NMDA and AMPA receptors

    Mellor, I. R., Brier, T. J., Pluteanu, F., Strømgaard, Kristian, Saghyan, A., Eldursi, N., Brierley, M. J., Andersen, K., Jaroszewski, J. W., Krogsgaard-Larsen, Povl & Usherwood, P. N. R., Jan 2003, In: Neuropharmacology. 44, 1, p. 70-80 11 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  3. Published

    Preparation of 7-substituted ginkgolide derivatives: potent platelet activating factor (PAF) receptor antagonists

    Vogensen, S. B., Strømgaard, Kristian, Shindou, H., Jaracz, S., Suehiro, M., Ishii, S., Shimizu, T. & Nakanishi, K., 13 Feb 2003, In: Journal of Medicinal Chemistry. 46, 4, p. 601-608 8 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  4. Published

    Contrasting actions of philanthotoxin-343 and philanthotoxin-(12) on human muscle nicotinic acetylcholine receptors

    Brier, T. J., Mellor, I. R., Tikhonov, D. B., Neagoe, I., Shao, Z., Brierley, M. J., Strømgaard, Kristian, Jaroszewski, J. W., Krogsgaard-Larsen, Povl & Usherwood, P. N. R., Oct 2003, In: Molecular Pharmacology. 64, 4, p. 954-964 11 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  5. Terpene trilactones from Ginkgo biloba are antagonists of cortical glycine and GABA(A) receptors

    Ivic, L., Sands, T. T. J., Fishkin, N., Nakanishi, K., Kriegstein, A. R. & Strømgaard, Kristian, 5 Dec 2003, In: Journal of Biological Chemistry. 278, 49, p. 49279-49285 7 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  6. 2004
  7. Published

    Ginkgolides and glycine receptors: a structure-activity relationship study

    Jaracz, S., Nakanishi, K., Jensen, Anders A. & Strømgaard, Kristian, 2004, In: Chemistry: A European Journal. 10, 6, p. 1507-18 12 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  8. Published

    Site-specific incorporation of unnatural amino acids into proteins

    Strømgaard, A., Jensen, Anders A. & Strømgaard, Kristian, 2004, In: ChemBioChem. 5, 7, p. 909-16 8 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  9. Published

    Synthesis of polyamines and polyamine toxins. An improved alkylation procedure

    Strømgaard, Kristian & Andersen, T., 2004, In: Tetrahedron Letters. 45, p. 7929-7933

    Research output: Contribution to journalJournal articleResearchpeer-review

  10. Published

    Chemistry and biology of terpene trilactones from Ginkgo biloba

    Strømgaard, Kristian & Nakanishi, K., 19 Mar 2004, In: Angewandte Chemie International Edition. 43, 13, p. 1640-1658 19 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  11. Published

    AMPA receptor ligands: synthetic and pharmacological studies of polyamines and polyamine toxins

    Strømgaard, Kristian & Mellor, I., Sep 2004, In: Medicinal Research Reviews. 24, 5, p. 589-620 32 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  12. Published

    Preparation of a tritiated ginkgolide

    Strømgaard, Kristian, Suehiro, M. & Nakanishi, K., 15 Nov 2004, In: Bioorganic & Medicinal Chemistry Letters. 14, 22, p. 5673-5675 3 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  13. 2005
  14. Published

    Natural products as tools for studies of ligand-gated ion channels

    Strømgaard, Kristian, 2005, In: Chemical Record. 5, 4, p. 229-239 11 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  15. Published

    Polyamine toxins: development of selective ligands for ionotropic receptors

    Strømgaard, Kristian, Jensen, L. S. & Vogensen, S. B., 1 Mar 2005, In: Toxicon. 45, 3, p. 249-254 6 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  16. Published

    Design and synthesis of labeled analogs of PhTX-56, a potent and selective AMPA receptor antagonist

    Andersen, T. F., Vogensen, S. B., Jensen, L. S., Knapp, K. M. & Strømgaard, Kristian, 1 Sep 2005, In: Bioorganic & Medicinal Chemistry. 13, 17, p. 5104-5112 9 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  17. 2006
  18. Published

    Protolytic properties of polyamine wasp toxin analogues studied by 13C NMR spectroscopy

    Strømgaard, Kristian, Piazzi, L., Olsen, Christian Adam, Franzyk, Henrik & Jaroszewski, J. W., 2006, In: Magnetic Resonance in Chemistry. 44, 11, p. 1013-22 10 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  19. Published

    Stoffer fra Tempeltæet (Ginkgo biloba) som redskaber for studier af hjernens funktion

    Jensen, Anders A. & Strømgaard, Kristian, 2006, In: Dansk Kemi 83. 87, 1, p. 16-18

    Research output: Contribution to journalJournal articleCommunication

  20. Published

    Unaturlige aminosyrer skaber ny viden om proteiner

    Rannes, J., Andersen, J., Jensen, Anders A., Christensen, L. & Strømgaard, Kristian, 2006, In: Lægemiddelforskning. p. 28-29

    Research output: Contribution to journalJournal articleCommunication

  21. Published

    Design, synthesis, and pharmacological characterization of polyamine toxin derivatives: potent ligands for the pore-forming region of AMPA receptors

    Jensen, L. S., Bølcho, U., Egebjerg, J. & Strømgaard, Kristian, Apr 2006, In: ChemMedChem. 1, 4, p. 419-428 10 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  22. Published

    Uncompetitive antagonism of AMPA receptors: Mechanistic insights from studies of polyamine toxin derivatives

    Andersen, T. F., Tikhonov, D. B., Bølcho, U., Bolshakov, K., Nelson, J. K., Pluteanu, F., Mellor, I. R., Egebjerg, J. & Strømgaard, Kristian, 7 Sep 2006, In: Journal of Medicinal Chemistry. 49, 18, p. 5414-5423 10 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  23. 2007
  24. Published

    Expressed protein ligation of ionotropic glutamate receptors

    Jensen, M. S., Kristensen, Anders Skov & Strømgaard, Kristian, 2007, In: Biopolymers. 88, 4, p. 602

    Research output: Contribution to journalConference abstract in journalResearch

  25. Published

    Probing the pharmacophore of ginkgolides as glycine receptor antagonists

    Jensen, Anders A., Begum, N., Vogensen, S. B., Knapp, K. M., Gundertofte, K., Dzyuba, S. V., Ishii, H., Nakanishi, K., Kristiansen, Uffe & Strømgaard, Kristian, 2007, In: Journal of Medicinal Chemistry. 50, 7, p. 1610-1617

    Research output: Contribution to journalJournal articleResearchpeer-review

  26. 2008
  27. Published

    Electrophysiological characterization of analogues of philanthotoxin-343 on ionotropic glutamate receptors

    Frølund, S. U., Ziegler, H. L., Franzyk, Henrik, Strømgaard, Kristian, Kristensen, Anders Skov & Jaroszewski, J. W., 2008.

    Research output: Contribution to conferencePosterResearch

  28. Published

    From the selective serotonin transporter inhibitor citalopram to the selective norepinephrine transporter inhibitor talopram: Synthesis and structure-activity relationship studies

    Eildal, J. N. N., Andersen, J., Kristensen, Anders Skov, Jørgensen, A. M., Bang-Andersen, B., Jørgensen, M. & Strømgaard, Kristian, 2008, In: Journal of Medicinal Chemistry. 51, 10, p. 3045-3048

    Research output: Contribution to journalJournal articleResearchpeer-review

  29. Published

    Giftstoffer fra hvepse og edderkopper i forskning og lægemiddeludvikling

    Strømgaard, Kristian, 2008, In: Carlsbergfondet. Aarsskrift. p. 42-47

    Research output: Contribution to journalJournal articleCommunication

  30. Published

    Modified peptides as potent inhibitors of the postsynaptic density-95/N-methyl-D-aspartate receptor interaction

    Bach, Anders, Chi, C. N., Olsen, T. B., Pedersen, S. W., Røder, M. U., Pang, G. F., Clausen, Rasmus Prætorius, Jemth, P. & Strømgaard, Kristian, 2008, In: Journal of Medicinal Chemistry. 51, 20, p. 6450-6459

    Research output: Contribution to journalJournal articleResearchpeer-review

  31. Published

    Protein-protein interaktion: et nyt mål for udvikling af lægemidler

    Bach, Anders, Gottschalk, M., Kristensen, Anders Skov & Strømgaard, Kristian, 2008, In: Lægemiddelforskning. p. 10-12

    Research output: Contribution to journalJournal articleCommunication

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