Hans Bräuner

Hans Bräuner

Prodekan for forskning

ORCID: 0000-0001-9495-7388

Publication year:
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1 - 100 out of 252Page size: 100
  1. 2024
  2. Published

    Characterization of the real-time internalization of nine GPCRs reveals distinct dependence on arrestins and G proteins

    Møller, T. C., Moo, Ee Von, Inoue, A., Pedersen, M. F. & Bräuner, Hans, 2024, In: Biochimica et Biophysica Acta - Molecular Cell Research. 1871, 1, 12 p., 119584.

    Research output: Contribution to journal › Journal article › Research › peer-review

  3. Published

    Structure-Activity Relationship Studies and Optimization of 4-Hydroxypyridones as GPR84 Agonists

    Ieremias, L., Kaspersen, M. H., Manandhar, Asmita, Schultz-Knudsen, Katrine, Vrettou, C. I., Pokhrel, R., Heidtmann, C. V., Jenkins, L., Kanellou, C., Marsango, S., Li, Y., Bräuner, Hans, Ulven, Elisabeth Rexen, Milligan, G. & Ulven, Trond, 2024, In: Journal of Medicinal Chemistry. 67, 5, p. 3542-3570

    Research output: Contribution to journal › Journal article › Research › peer-review

  4. 2023
  5. Published

    The Concise Guide to PHARMACOLOGY 2023/24: G protein-coupled receptors

    Alexander, S. P. H., Christopoulos, A., Davenport, A. P., Kelly, E., Mathie, A. A., Peters, J. A., Veale, E. L., Armstrong, J. F., Faccenda, E., Harding, S. D., Davies, J. A., Abbracchio, M. P., Abraham, G., Agoulnik, A., Alexander, W., Al-Hosaini, K., Bäck, M., Baker, J. G., Barnes, N. M., Bathgate, R. & 146 others, Beaulieu, J., Beck-Sickinger, A. G., Behrens, M., Bernstein, K. E., Bettler, B., Birdsall, N. J. M., Blaho, V., Boulay, F., Bousquet, C., Bräuner, Hans, Burnstock, G., Caló, G., Castaño, J. P., Catt, K. J., Ceruti, S., Chazot, P., Chiang, N., Chini, B., Chun, J., Cianciulli, A., Civelli, O., Clapp, L. H., Couture, R., Cox, H. M., Csaba, Z., Dahlgren, C., Dent, G., Douglas, S. D., Dournaud, P., Eguchi, S., Escher, E., Filardo, E. J., Fong, T., Fumagalli, M., Gainetdinov, R. R., Garelja, M. L., de Gasparo, M., Gerard, C., Gershengorn, M., Gobeil, F., Goodfriend, T. L., Goudet, C., Grätz, L., Gregory, K. J., Gundlach, A. L., Hamann, J., Hanson, J., Hauger, R. L., Hay, D. L., Heinemann, A., Herr, D., Hollenberg, M. D., Holliday, N. D., Horiuchi, M., Hoyer, D., Hunyady, L., Husain, A., IJzerman, A. P., Inagami, T., Jacobson, K. A., Jensen, R. T., Jockers, R., Jonnalagadda, D., Karnik, S., Kaupmann, K., Kemp, J., Kennedy, C., Kihara, Y., Kitazawa, T., Kozielewicz, P., Kreienkamp, H., Kukkonen, J. P., Langenhan, T., Larhammar, D., Leach, K., Lecca, D., Lee, J. D., Leeman, S. E., Leprince, J., Li, X. X., Lolait, S. J., Lupp, A., Macrae, R., Maguire, J., Malfacini, D., Mazella, J., McArdle, C. A., Melmed, S., Michel, M. C., Miller, L. J., Mitolo, V., Mouillac, B., Müller, C. E., Murphy, P. M., Nahon, J., Ngo, T., Norel, X., Nyimanu, D., O'Carroll, A., Offermanns, S., Panaro, M. A., Parmentier, M., Pertwee, R. G., Pin, J., Prossnitz, E. R., Quinn, M., Ramachandran, R., Ray, M., Reinscheid, R. K., Rondard, P., Rovati, G. E., Ruzza, C., Sanger, G. J., Schöneberg, T., Schulte, G., Schulz, S., Segaloff, D. L., Serhan, C. N., Singh, K. D., Smith, C. M., Stoddart, L. A., Sugimoto, Y., Summers, R., Tan, V. P., Thal, D., Thomas, W. W., Timmermans, P. B. M. W. M., Tirupula, K., Toll, L., Tulipano, G., Unal, H., Unger, T., Valant, C., Vanderheyden, P., Vaudry, D., Vaudry, H., Vilardaga, J., Walker, C. S., Wang, J. M., Ward, D. T., Wester, H., Willars, G. B., Williams, T. L., Woodruff, T. M., Yao, C. & Ye, R. D., Oct 2023, In: British Journal of Pharmacology. 180 Suppl 2, p. S23-S144

    Research output: Contribution to journal › Journal article › Research › peer-review

  6. Published

    Endocytic proteins mediating GPR15 receptor internalization provide insight into the underlying mechanisms

    Deng, Y., Moo, Ee Von, Inoue, A. & Bräuner, Hans, 2023, In: FEBS Letters. 597, 11, p. 1528-1540

    Research output: Contribution to journal › Journal article › Research › peer-review

  7. Published

    Pharmacological characterization of novel small molecule agonists and antagonists for the orphan receptor GPR139

    Pallareti, L., Rath, T. F., Trapkov, Boris, Tsonkov, T., Nielsen, A. T., Harpsøe, Kasper, Gentry, P. R., Bräuner, Hans, Gloriam, David E. & Foster, S. R., 2023, In: European Journal of Pharmacology. 943, 175553.

    Research output: Contribution to journal › Journal article › Research › peer-review

  8. Published

    Structure–activity relationship of GPR15L peptide analogues and investigation of their interaction with the GPR15 receptor

    Deng, Y., Perez Almeria, C. V., van Gijzel, L., Schaller, Kay, Vedel, L., Gloriam, David E., Ulven, Trond & Bräuner, Hans, 2023, In: Basic and Clinical Pharmacology and Toxicology. 132, 6, p. 459-471

    Research output: Contribution to journal › Journal article › Research › peer-review

  9. 2022
  10. Published

    Delineation of the GPR15 receptor-mediated Gα protein signalling profile in recombinant mammalian cells

    Deng, Y., Moo, Ee Von, Almería, C. V. P., Gentry, P. R., Vedel, L., Mathiesen, Jesper M. & Bräuner, Hans, 2022, In: Basic and Clinical Pharmacology and Toxicology. 131, 2, p. 104-113

    Research output: Contribution to journal › Journal article › Research › peer-review

  11. Published

    Development of a medium throughput whole-cell microtiter plate Thr286 autophosphorylation assay for CaMKIIα using ELISA

    Palmelund, L. B., van Woerden, G. M., Bräuner, Hans & Wellendorph, Petrine, 2022, In: Journal of Pharmacological and Toxicological Methods. 118, 8 p., 107226.

    Research output: Contribution to journal › Journal article › Research › peer-review

  12. Published

    Ligand-directed bias of G protein signaling at the dopamine D2 receptor

    Moo, Ee Von, Harpsøe, Kasper, Hauser, Alexander Sebastian, Masuho, I., Bräuner, Hans, Gloriam, David E. & Martemyanov, K. A., 2022, In: Cell Chemical Biology. 29, 2, p. 226-238

    Research output: Contribution to journal › Journal article › Research › peer-review

  13. Published

    Molecular insights into ligand recognition and G protein coupling of the neuromodulatory orphan receptor GPR139

    Zhou, Y., Daver, H., Trapkov, B., Wu, L., Wu, M., Harpsøe, Kasper, Gentry, P. R., Liu, K., Larionova, M., Liu, J., Chen, N., Bräuner, Hans, Gloriam, David E., Hua, T. & Liu, Z. J., 2022, In: Cell Research. 32, 2, p. 210-213

    Research output: Contribution to journal › Letter › Research › peer-review

  14. Published

    Somatostatin venom analogs evolved by fish-hunting cone snails: From prey capture behavior to identifying drug leads

    Ramiro, Iris Bea L. , Bjørn-Yoshimoto, Walden, Imperial, J. S., Gajewiak, J., Salcedo, P. F., Watkins, M., Taylor, D., Resager, W., Ueberheide, B., Bräuner, Hans, Whitby, F. G., Hill, C. P., Martin, L. F., Patwardhan, A., Concepcion, G. P., Olivera, B. M. & Safavi-Hemami, H., 2022, In: Science Advances. 8, 12, 16 p., eabk1410.

    Research output: Contribution to journal › Journal article › Research › peer-review

  15. Published

    Use of CRISPR/Cas9-edited HEK293 cells reveals that both conventional and novel protein kinase C isozymes are involved in mGlu5a receptor internalization

    van Senten, Jeffrey Roy, Møller, T. C., Moo, Ee Von, Seiersen, S. D. & Bräuner, Hans, 2022, In: Journal of Biological Chemistry. 298, 10, 16 p., 102466.

    Research output: Contribution to journal › Journal article › Research › peer-review

  16. 2021
  17. Published

    Positive allosteric modulators of metabotropic glutamate receptor 5 as tool compounds to study signaling bias

    Arsova, A., Møller, T. C., Hellyer, S. D., Vedel, L., Foster, S. R., Hansen, J. L., Bräuner, Hans & Gregory, K. J., 1 May 2021, In: Molecular Pharmacology. 99, 5, p. 328-241

    Research output: Contribution to journal › Journal article › Research › peer-review

  18. Published

    Arrestin-Dependent and -Independent Internalization of G Protein–Coupled Receptors: Methods, Mechanisms, and Implications on Cell Signaling

    Moo, Ee Von, van Senten, Jeffrey Roy, Bräuner, Hans & Møller, T. C., 2021, In: Molecular Pharmacology. 99, 4, p. 242-255

    Research output: Contribution to journal › Journal article › Research › peer-review

  19. Published

    Asymmetric activation of the calcium-sensing receptor homodimer

    Gao, Y., Robertson, M. J., Rahman, Sabrina Nalini, Seven, A. B., Zhang, C., Meyerowitz, J. G., Panova, O., Hannan, F. M., Thakker, R. V., Bräuner, Hans, Mathiesen, Jesper M. & Skiniotis, G., 2021, In: Nature. 595, p. 455-459

    Research output: Contribution to journal › Journal article › Research › peer-review

  20. Published

    GLP-1 Val8: A Biased GLP-1R Agonist with Altered Binding Kinetics and Impaired Release of Pancreatic Hormones in Rats

    van der Velden, W. J. C., Smit, F. X., Christiansen, Charlotte Bayer, Møller, T. C., Hjortø, Gertrud Malene, Larsen, Olav, Schiellerup, S. P., Bräuner, Hans, Holst, Jens Juul, Hartmann, Bolette, Frimurer, Thomas Michael & Rosenkilde, Mette, 2021, In: ACS Pharmacology & Translational Science. 4, 1, p. 296-313 18 p.

    Research output: Contribution to journal › Journal article › Research › peer-review

  21. Published

    Mutational Landscape of the Proglucagon-Derived Peptides

    Lindquist, Peter, Madsen, Jakob Sture, Bräuner, Hans, Rosenkilde, Mette & Hauser, Alexander Sebastian, 2021, In: Frontiers in Endocrinology. 12, 14 p., 698511.

    Research output: Contribution to journal › Journal article › Research › peer-review

  22. Published

    THE CONCISE GUIDE TO PHARMACOLOGY 2021/22: G protein-coupled receptors

    Alexander, S. P., Christopoulos, A., Davenport, A. P., Kelly, E., Mathie, A., Peters, J. A., Veale, E. L., Armstrong, J. F., Faccenda, E., Harding, S. D., Pawson, A. J., Southan, C., Davies, J. A., Abbracchio, M. P., Alexander, W., Al-Hosaini, K., Bäck, M., Barnes, N. M., Bathgate, R., Beaulieu, J-M. & 135 others, Bernstein, K. E., Bettler, B., Birdsall, N. J. M., Blaho, V., Boulay, F., Bousquet, C., Bräuner, Hans, Burnstock, G., Caló, G., Castaño, J. P., Catt, K. J., Ceruti, S., Chazot, P., Chiang, N., Chini, B., Chun, J., Cianciulli, A., Civelli, O., Clapp, L. H., Couture, R., Csaba, Z., Dahlgren, C., Dent, G., Singh, K. D., Douglas, S. D., Dournaud, P., Eguchi, S., Escher, E., Filardo, E. J., Fong, T., Fumagalli, M., Gainetdinov, R. R., Gasparo, M. D., Gerard, C., Gershengorn, M., Gobeil, F., Goodfriend, T. L., Goudet, C., Gregory, K. J., Gundlach, A. L., Hamann, J., Hanson, J., Hauger, R. L., Hay, D. L., Heinemann, A., Hollenberg, M. D., Holliday, N. D., Horiuchi, M., Hoyer, D., Hunyady, L., Husain, A., IJzerman, A. P., Inagami, T., Jacobson, K. A., Jensen, R. T., Jockers, R., Jonnalagadda, D., Karnik, S., Kaupmann, K., Kemp, J., Kennedy, C., Kihara, Y., Kitazawa, T., Kozielewicz, P., Kreienkamp, H., Kukkonen, J. P., Langenhan, T., Leach, K., Lecca, D., Lee, J. D., Leeman, S. E., Leprince, J., Li, X. X., Williams, T. L., Lolait, S. J., Lupp, A., Macrae, R., Maguire, J., Mazella, J., McArdle, C. A., Melmed, S., Michel, M. C., Miller, L. J., Mitolo, V., Mouillac, B., Müller, C. E., Murphy, P., Nahon, J., Ngo, T., Norel, X., Nyimanu, D., O'Carroll, A., Offermanns, S., Panaro, M. A., Parmentier, M., Pertwee, R. G., Pin, J., Prossnitz, E. R., Quinn, M., Ramachandran, R., Ray, M., Reinscheid, R. K., Rondard, P., Rovati, G. E., Ruzza, C., Sanger, G. J., Schöneberg, T., Schulte, G., Schulz, S., Segaloff, D. L., Serhan, C. N., Stoddart, L. A., Sugimoto, Y., Summers, R., Tan, V. P., Thal, D., Thomas, W. W., Timmermans, P. B. M. W. M., Tirupula, K., Tulipano, G., Unal, H., Unger, T., Valant, C., Vanderheyden, P., Vaudry, D., Vaudry, H., Vilardaga, J., Walker, C. S., Wang, J. M., Ward, D. T., Wester, H., Willars, G. B., Woodruff, T. M., Yao, C. & Ye, R. D., 2021, In: British Journal of Pharmacology. 178 , S1, p. S27-S156

    Research output: Contribution to journal › Journal article › Research › peer-review

  23. Published

    The Calcium-Sensing Receptor Is Essential for Calcium and Bicarbonate Sensitivity in Human Spermatozoa

    Boisen, I. M., Rehfeld, Anders Aagaard, Mos, I., Poulsen, N. N., Nielsen, J. E., Schwarz, Peter, Rejnmark, L., Dissing, Steen, Bach-Mortensen, P., Juul, Anders, Bräuner, Hans, Lanske, B. & Blomberg Jensen, M., 2021, In: The Journal of clinical endocrinology and metabolism. 106, 4, p. e1775-e1792

    Research output: Contribution to journal › Journal article › Research › peer-review

  24. 2020
  25. Published

    International Union of Basic and Clinical Pharmacology. CVIII. Calcium-Sensing Receptor Nomenclature, Pharmacology, and Function

    Leach, K., Hannan, F. M., Josephs, T. M., Keller, A. N., Møller, T. C., Ward, D. T., Kallay, E., Mason, R. S., Thakker, R. V., Riccardi, D., Conigrave, A. D. & Bräuner, Hans, Jul 2020, In: Pharmacological Reviews. 72, 3, p. 558-604 47 p.

    Research output: Contribution to journal › Review › Research › peer-review

  26. Published

    Heterozygous Mutation (Q459R) in the Calcium-Sensing Receptor Gene Causes Familial Hypocalciuric Hypercalcemia 1 (FHH1)

    Boisen, I. M., Mos, I., Lerche-Black, E. M., Juul, Anders, Bräuner, Hans & Blomberg Jensen, M., 1 Apr 2020, In: The Journal of clinical endocrinology and metabolism. 105, 4, p. e1322-e1330

    Research output: Contribution to journal › Journal article › Research › peer-review

  27. Published

    Novel approaches leading towards peptide GPCR de-orphanisation

    Hauser, Alexander Sebastian, Gloriam, David E., Bräuner, Hans & Foster, S. R., 1 Mar 2020, In: British Journal of Pharmacology. 177, 5, p. 961-968 8 p.

    Research output: Contribution to journal › Review › Research › peer-review

  28. Published

    Biased agonism of clinically approved μ-opioid receptor agonists and TRV130 is not controlled by binding and signaling kinetics

    Pedersen, M. F., Wrobel, T. M., Marcher, Emil, Pedersen, D. S., Møller, T. C., Gabriele, F., Pedersen, H., Matosiuk, D., Foster, S. R., Bouvier, M. & Bräuner, Hans, 2020, In: Neuropharmacology. 166, 13 p., 107718.

    Research output: Contribution to journal › Journal article › Research › peer-review

  29. Published

    Delineation of molecular determinants for FR900359 inhibition of Gq/11 unlocks inhibition of Gαs

    Boesgaard, M. W., Harpsøe, Kasper, Malmberg, M., Underwood, C. R., Inoue, A., Mathiesen, Jesper M., König, G. M., Kostenis, E., Gloriam, David E. & Bräuner, Hans, 2020, In: Journal of Biological Chemistry. 295, 40, p. 13850-13861

    Research output: Contribution to journal › Journal article › Research › peer-review

  30. Published

    Detailed in vitro pharmacological characterization of clinically tested negative allosteric modulators of the metabotropic glutamate receptor 5 (mGlu5)

    Arsova, A., Møller, T. C., Vedel, L., Hansen, J. L., Foster, S. R., Gregory, K. J. & Bräuner, Hans, 2020, In: Molecular Pharmacology. 98, 1, p. 49-60

    Research output: Contribution to journal › Journal article › Research › peer-review

  31. Published

    Dissecting the roles of GRK2 and GRK3 in μ-opioid receptor internalization and β-arrestin2 recruitment using CRISPR/Cas9-edited HEK293 cells

    Møller, T. C., Pedersen, M. F., van Senten, Jeffrey Roy, Seiersen, S. D., Mathiesen, Jesper M., Bouvier, M. & Bräuner, Hans, 2020, In: Scientific Reports. 10, 1, 13 p., 17395.

    Research output: Contribution to journal › Journal article › Research › peer-review

  32. Published

    Enhanced agonist residence time, internalization rate and signalling of the GIP receptor variant [E354Q] facilitate receptor desensitization and long-term impairment of the GIP system

    Gabe, M. B. N., van der Velden, W. J. C., Gadgaard, S., Smit, F. X., Hartmann, Bolette, Bräuner, Hans & Rosenkilde, Mette, 2020, In: Basic & Clinical Pharmacology & Toxicology. 126, p. 122-132

    Research output: Contribution to journal › Journal article › Research › peer-review

  33. Published

    G protein-coupled receptor pharmacology-The next generation

    Bräuner, Hans, Rosenkilde, Mette, Gether, Ulrik & Gloriam, David E., 2020, In: Basic & Clinical Pharmacology & Toxicology. 126, Supplement 6, p. 3-4 2 p.

    Research output: Contribution to journal › Editorial › Research

  34. Published

    Pharmacology and physiological function of the orphan GPRC6A receptor

    Jorgensen, C. V. & Bräuner, Hans, 2020, In: Basic & Clinical Pharmacology & Toxicology. 126, p. 77-87 11 p.

    Research output: Contribution to journal › Review › Research › peer-review

  35. Published

    The selective 5-HT2A receptor agonist 25CN-NBOH: structure-activity relationship, in vivo pharmacology, and in vitro and ex vivo binding characteristics of [3H]25CN-NBOH

    Jensen, Anders A., Halberstadt, A. L., Marcher, Emil, Odland, Anna Ulstein, Chatha, M., Speth, N., Liebscher, G., Hansen, M., Bräuner, Hans, Palner, M., Andreasen T., Jesper & Kristensen, Jesper Langgaard, 2020, In: Biochemical Pharmacology. 177, 16 p., 113979.

    Research output: Contribution to journal › Journal article › Research › peer-review

  36. 2019
  37. Published

    Calcium sensing receptor in male germ cells is essential for processes leading to fertilization

    Boisen, I. M., Jensen, Martin Blomberg, Rehfeld, Anders Aagaard, Nielsen, J. E., Juul, Anders, Mos, I., Bräuner, Hans & Lanske, B., Dec 2019, p. 216-216.

    Research output: Contribution to conference › Conference abstract for conference › Research › peer-review

  38. Published

    Discovery of Human Signaling Systems: Pairing Peptides to G Protein-Coupled Receptors

    Foster, S. R., Hauser, Alexander Sebastian, Vedel, L., Strachan, R. T., Huang, X., Gavin, A. C., Shah, S. D., Nayak, A. P., Haugaard-Kedström, L. M., Penn, R. B., Roth, B. L., Bräuner, Hans & Gloriam, David E., 31 Oct 2019, In: Cell. 179, 4, p. 895-908

    Research output: Contribution to journal › Journal article › Research › peer-review

  39. Published

    Calcium-Sensing Receptor Internalization Is β-Arrestin-Dependent and Modulated by Allosteric Ligands

    Mos, I., Jacobsen, S. E., Foster, S. R. & Bräuner, Hans, Oct 2019, In: Molecular Pharmacology. 96, 4, p. 463-474 12 p.

    Research output: Contribution to journal › Journal article › Research › peer-review

  40. Published

    Probing the Existence of a Metastable Binding Site at the β2-Adrenergic Receptor with Homobivalent Bitopic Ligands

    Gaiser, B. I., Danielsen, M., Marcher, Emil, Røpke Jørgensen, K., Wróbel, T. M., Frykman, M., Johansson, H., Bräuner, Hans, Gloriam, David E., Mathiesen, Jesper M. & Sejer Pedersen, D., 12 Sep 2019, In: Journal of Medicinal Chemistry. 62, 17, p. 7806-7839 34 p.

    Research output: Contribution to journal › Journal article › Research › peer-review

  41. Published

    Pharmacology and function of the orphan GPR139 G protein-coupled receptor

    Vedel, L., Nøhr, A. C., Gloriam, David E. & Bräuner, Hans, 27 May 2019, In: Basic & Clinical Pharmacology & Toxicology. 126, p. 35-46

    Research output: Contribution to journal › Review › Research › peer-review

  42. Published

    Metabolic and skeletal homeostasis are maintained in full locus GPRC6A knockout mice

    Jørgensen, C. V., Gasparini, S. J., Tu, J., Zhou, H., Seibel, M. J. & Bräuner, Hans, 12 Apr 2019, In: Scientific Reports. 9, 1, 8 p., 5995.

    Research output: Contribution to journal › Journal article › Research › peer-review

  43. Published

    Rational design of a heterotrimeric G protein α subunit with artificial inhibitor sensitivity

    Malfacini, D., Patt, J., Annala, S., Harpsøe, Kasper, Eryilmaz, F., Reher, R., Crüsemann, M., Hanke, W., Zhang, H., Tietze, D., Gloriam, David E., Bräuner, Hans, Strømgaard, Kristian, König, G. M., Inoue, A., Gomeza, J. & Kostenis, E., 12 Apr 2019, In: The Journal of Biological Chemistry. 294, 15, p. 5747-5758

    Research output: Contribution to journal › Journal article › Research › peer-review

  44. Published

    Label-free dynamic mass redistribution analysis of endogenous adrenergic receptor signaling in primary preadipocytes and differentiated adipocytes

    Jørgensen, C. V., Zhou, H., Seibel, M. J. & Bräuner, Hans, 1 Apr 2019, In: Journal of Pharmacological and Toxicological Methods. 97, p. 59-66 8 p.

    Research output: Contribution to journal › Journal article › Research › peer-review

  45. Published

    Structure–Activity Relationship Studies of the Natural Product G q/11 Protein Inhibitor YM-254890

    Xiong, X. F., Zhang, H., Boesgaard, M. W., Underwood, C. R., Bräuner, Hans & Strømgaard, Kristian, Apr 2019, In: ChemMedChem. 14, 8, p. 865-870

    Research output: Contribution to journal › Journal article › Research › peer-review

  46. Published

    Identification of a novel scaffold for a small molecule GPR139 receptor agonist

    Nøhr, A. C., Shehata, M. A., Palmer, D., Pokhrel, R., Vallianou, M., Foster, S. R., Gentry, P. R., Gloriam, David E. & Bräuner, Hans, 7 Mar 2019, In: Scientific Reports. 9, 1, 10 p., 3802.

    Research output: Contribution to journal › Journal article › Research › peer-review

  47. 2018
  48. Published

    Human GIP(3-30)NH inhibits G protein-dependent as well as G protein-independent signaling and is selective for the GIP receptor with high-affinity binding to primate but not rodent GIP receptors

    Gabe, M. B. N., Sparre-Ulrich, A. H., Pedersen, M. F., Gasbjerg, Lærke Smidt, Inoue, A., Bräuner, Hans, Hartmann, Bolette & Rosenkilde, M. M., 31 Jan 2018, In: Biochemical Pharmacology. 150, p. 97-107 11 p.

    Research output: Contribution to journal › Journal article › Research › peer-review

  49. Published

    Structure–activity relationship and conformational studies of the natural product cyclic depsipeptides YM-254890 and FR900359

    Zhang, H., Nielsen, A. L., Boesgaard, M. W., Harpsøe, Kasper, Daly, N. L., Xiong, X., Underwood, C. R., Haugaard-kedström, L. M., Bräuner, Hans, Gloriam, David E. & Strømgaard, Kristian, 2018, In: European Journal of Medicinal Chemistry. 156, p. 847-860

    Research output: Contribution to journal › Journal article › Research › peer-review

  50. 2017
  51. Published

    THE CONCISE GUIDE TO PHARMACOLOGY 2017/18: Overview

    CGTP Collaborators, C. C., Dec 2017, In: British Journal of Pharmacology. 174, p. S1-S16

    Research output: Contribution to journal › Journal article › Research › peer-review

  52. Published

    Investigating Internalization and Intracellular Trafficking of GPCRs: New Techniques and Real-Time Experimental Approaches

    Foster, S. R. & Bräuner, Hans, 11 Oct 2017, Handbook of Experimental Pharmacology. Springer, Vol. 245. p. 41-61 (Handbook of Experimental Pharmacology).

    Research output: Chapter in Book/Report/Conference proceeding › Book chapter › Research › peer-review

  53. Published

    Structure-Activity Relationship, Pharmacological Characterization, and Molecular Modeling of Noncompetitive Inhibitors of the Betaine/γ-Aminobutyric Acid Transporter 1 (BGT1)

    Jørgensen, L., Al-Khawaja, A., Kickinger, S., Vogensen, S. B., Skovgaard-Petersen, J., Rosenthal, E., Borkar, N., Löffler, R., Madsen, K. K., Bräuner, Hans, Schousboe, Arne, Ecker, G. F., Wellendorph, Petrine & Clausen, Rasmus Prætorius, 9 Oct 2017, In: Journal of Medicinal Chemistry. 60, 21, p. 8834-8846

    Research output: Contribution to journal › Journal article › Research › peer-review

  54. Published

    Identification of AICP as a GluN2C-Selective N-Methyl-d-Aspartate Receptor Superagonist at the GluN1 Glycine Site

    Jessen, M., Frederiksen, K., Yi, F., Clausen, Rasmus Prætorius, Hansen, K. B., Bräuner, Hans, Kilburn, J. P. & Damholt, A., Aug 2017, In: Molecular Pharmacology. 92, 2, p. 151-161 11 p.

    Research output: Contribution to journal › Journal article › Research › peer-review

  55. Published

    Applying label-free dynamic mass redistribution assay for studying endogenous FPR1 receptor signalling in human neutrophils

    Christensen, H. B., Gloriam, David E., Pedersen, D. S., Cowland, J. B., Borregaard, N. & Bräuner, Hans, 15 Jul 2017, In: Journal of Pharmacological and Toxicological Methods. 88, Pt 1, p. 72-78 7 p.

    Research output: Contribution to journal › Journal article › Research › peer-review

  56. Published

    Identification of Histamine H3 Receptor Ligands Using a New Crystal Structure Fragment-based Method

    Frandsen, I. O., Boesgaard, M. W., Fidom, K., Hauser, Alexander Sebastian, Isberg, V., Bräuner, Hans, Wellendorph, Petrine & Gloriam, David E., 6 Jul 2017, In: Scientific Reports. 7, 1, 10 p., 4829.

    Research output: Contribution to journal › Journal article › Research › peer-review

  57. Published

    Structure-Activity Relationship Studies of the Cyclic Depsipeptide Natural Product YM-254890, Targeting the Gq Protein

    Zhang, H., Xiong, X., Boesgaard, M. W., Underwood, C. R., Bräuner, Hans & Strømgaard, Kristian, 7 Jun 2017, In: ChemMedChem. 12, 11, p. 830-834 5 p.

    Research output: Contribution to journal › Journal article › Research › peer-review

  58. Published

    The GPR139 reference agonists 1a and 7c, and tryptophan and phenylalanine share a common binding site

    Shehata, M. A., Jensen, A. C. N., Jespers, W., Floryan, L., Isberg, V., Andersen, K. B., Åqvist, J., Gutiérrez-de-Terán, H., Bräuner, Hans & Gloriam, David E., 25 Apr 2017, In: Scientific Reports. 7, 9 p., 1128.

    Research output: Contribution to journal › Journal article › Research › peer-review

  59. Published

    Knockin mouse with mutant Gα11 mimics human inherited hypocalcemia and is rescued by pharmacologic inhibitors

    Roszko, K. L., Bi, R., Gorvin, C. M., Bräuner, Hans, Xiong, X., Inoue, A., Thakker, R. V., Strømgaard, Kristian, Gardella, T. & Mannstadt, M., 9 Feb 2017, In: JCI insight. 2, 3, 15 p., e91079.

    Research output: Contribution to journal › Journal article › Research › peer-review

  60. Published

    The orphan G protein-coupled receptor GPR139 is activated by the peptides: Adrenocorticotropic hormone (ACTH), α-, and β-melanocyte stimulating hormone (α-MSH, and β-MSH), and the conserved core motif HFRW

    Jensen, A. C. N., Shehata, M. A., Hauser, Alexander Sebastian, Isberg, V., Mokrosinski, J., Farooqi, I. S., Pedersen, D. S., Gloriam, David E. & Bräuner, Hans, 1 Jan 2017, In: Neurochemistry International. 102, p. 105-113

    Research output: Contribution to journal › Journal article › Research › peer-review

  61. Published

    Detailed characterization of the in vitro pharmacological and pharmacokinetic properties of N-(2-hydroxybenzyl)-2,5-dimethoxy-4-cyanophenylethylamine (25CN-NBOH), a highly selective and brain-penetrant 5-HT2A receptor agonist

    Jensen, Anders A., McCorvy, J. D., Petersen, S. L., Bundgaard, C., Liebscher, G., Kenakin, T. P., Bräuner, Hans, Kehler, J. & Kristensen, Jesper Langgaard, 2017, In: Journal of Pharmacology and Experimental Therapeutics. 361, 3, p. 441-453

    Research output: Contribution to journal › Journal article › Research › peer-review

  62. Published

    Genetic Variations in the Human G Protein-coupled Receptor Class C, Group 6, Member A (GPRC6A) Control Cell Surface Expression and Function

    Jorgensen, S., Have, C. T., Underwood, C. R., Johansen, L. D., Wellendorph, Petrine, Gjesing, A. P., Jorgensen, C. V., Quan, S., Rui, G., Inoue, A., Linneberg, Allan René, Grarup, Niels, Jun, W., Pedersen, Oluf Borbye, Hansen, Torben & Bräuner, Hans, 2017, In: The Journal of Biological Chemistry. 292, 4, p. 1524-1534 11 p.

    Research output: Contribution to journal › Journal article › Research › peer-review

  63. Published

    Investigating the molecular mechanism of positive and negative allosteric modulators in the calcium-sensing receptor dimer

    Jacobsen, S. E., Gether, Ulrik & Bräuner, Hans, 2017, In: Scientific Reports. 7, 14 p., 46355.

    Research output: Contribution to journal › Journal article › Research › peer-review

  64. Published

    Robust GLP-1 secretion by basic L-amino acids does not require the GPRC6A receptor

    Clemmensen, Christoffer, Jørgensen, C. V., Smajilovic, S. & Bräuner, Hans, 2017, In: Diabetes, Obesity and Metabolism. 19, 4, p. 599-603

    Research output: Contribution to journal › Journal article › Research › peer-review

  65. Published

    Structural insight to mutation effects uncover a common allosteric site in class C GPCRs

    Harpsøe, Kasper, Boesgaard, M. W., Munk, C., Bräuner, Hans & Gloriam, David E., 2017, In: Bioinformatics (Oxford, England). 33, 8, p. 1116-1120 5 p., btw784.

    Research output: Contribution to journal › Journal article › Research › peer-review

  66. Published

    The GPRC6A Receptor displays Constitutive Internalization and Sorting to the Slow Recycling Pathway

    Jacobsen, S. E., Ammendrup-Johnsen, I., Jansen, A. M., Gether, Ulrik, Madsen, Kenneth Lindegaard & Bräuner, Hans, 2017, In: The Journal of Biological Chemistry. 292, 17, p. 6910-6926

    Research output: Contribution to journal › Journal article › Research › peer-review

  67. 2016
  68. Published

    Novel Agonist Bioisosteres and Common Structure-Activity Relationships for The Orphan G Protein-Coupled Receptor GPR139

    Shehata, M. A., Jensen, A. C. N., Lissa, D., Bisig, C., Isberg, V., Andersen, K. B., Harpsøe, Kasper, Björkling, Fredrik, Bräuner, Hans & Gloriam, David E., 10 Nov 2016, In: Scientific Reports. 6, p. 1-13 13 p., 36681.

    Research output: Contribution to journal › Journal article › Research › peer-review

  69. Published

    Receptors structure, function, and pharmacology

    Bräuner, Hans, 19 Aug 2016, Textbook of Drug Design and Discovery, Fifth Edition. CRC Press, p. 193-212 20 p.

    Research output: Chapter in Book/Report/Conference proceeding › Book chapter › Research › peer-review

  70. Published

    Radiosynthesis and characterisation of a potent and selective GPR139 agonist radioligand

    Kuhne, S., Nøhr, A. C., Marek, A., Elbert, T., Klein, A. B., Bräuner, Hans, Wellendorph, Petrine & Pedersen, D. S., 2016, In: RSC Advances. 6, 2, p. 947-952 6 p.

    Research output: Contribution to journal › Journal article › Research › peer-review

  71. Published

    Receptors: Structure, Function, and Pharmacology

    Bräuner, Hans, 2016, Textbook of Drug Design and Discovery. Strømgaard, K., Krogsgaard-Larsen, P. & Madsen, U. (eds.). 5th ed. CRC Press, p. 193-212

    Research output: Chapter in Book/Report/Conference proceeding › Book chapter › Education › peer-review

  72. Published

    Total synthesis and structure–activity relationship studies of a series of selective G protein inhibitors

    Xiong, X., Zhang, H., Underwood, C. R., Harpsøe, Kasper, Gardella, T. J., Wöldike, M. F., Mannstadt, M., Gloriam, David E., Bräuner, Hans & Strømgaard, Kristian, 2016, In: Nature Chemistry. 8, 11, p. 1035-1041 7 p.

    Research output: Contribution to journal › Journal article › Research › peer-review

  73. 2015
  74. Published

    The Concise Guide to PHARMACOLOGY 2015/16: Overview

    CGTP Collaborators, C. C., 1 Dec 2015, In: British Journal of Pharmacology. 172, 24, p. 5729-5743 15 p.

    Research output: Contribution to journal › Review › Research › peer-review

  75. Published

    Selective Allosteric Antagonists for the G Protein-Coupled Receptor GPRC6A Based on the 2-Phenylindole Privileged Structure Scaffold

    Johansson, H., Boesgaard, M. W., Nørskov-Lauritsen, L., Larsen, I., Kuhne, S., Gloriam, David E., Bräuner, Hans & Sejer Pedersen, D., 25 Nov 2015, In: Journal of Medicinal Chemistry. 58, 22, p. 8938-51 14 p.

    Research output: Contribution to journal › Journal article › Research › peer-review

  76. Published

    Selective Negative Allosteric Modulation Of Metabotropic Glutamate Receptors - A Structural Perspective of Ligands and Mutants

    Harpsøe, Kasper, Isberg, V., Tehan, B. G., Weiss, D., Arsova, A., Marshall, F. H., Bräuner, Hans & Gloriam, David E., 11 Sep 2015, In: Scientific Reports. 5, p. 1-11 11 p., 13869.

    Research output: Contribution to journal › Journal article › Research › peer-review

  77. Published

    L-amino acid sensing G protein-coupled receptors and their role in food intake sensing

    Bräuner, Hans, Mar 2015, In: Chemical Senses. 40, 3, p. 231-231 1 p.

    Research output: Contribution to journal › Conference abstract in journal › Research › peer-review

  78. Published

    N-glycosylation and disulfide bonding affects GPRC6A receptor expression, function, and dimerization

    Nørskov-Lauritsen, L., Jørgensen, S. & Bräuner, Hans, 21 Jan 2015, In: FEBS Letters. 589, p. 588–597 10 p.

    Research output: Contribution to journal › Journal article › Research › peer-review

  79. Published

    Functional Consequences of Glucagon-like Peptide-1 Receptor Cross-talk and Trafficking

    Roed, S. N., Nøhr, A. C., Wismann, P., Iversen, H., Bräuner, Hans, Knudsen, S. M. & Waldhoer, M., 9 Jan 2015, In: The Journal of Biological Chemistry. 290, 2, p. 1233-1243 11 p.

    Research output: Contribution to journal › Journal article › Research › peer-review

  80. Published

    A cAMP Biosensor-Based High-Throughput Screening Assay for Identification of Gs-Coupled GPCR Ligands and Phosphodiesterase Inhibitors

    Vedel, L., Bräuner, Hans & Mathiesen, Jesper M., 2015, In: Journal of Biomolecular Screening. 20, p. 849-857 9 p.

    Research output: Contribution to journal › Journal article › Research › peer-review

  81. Published

    Identification of the first surrogate agonists for the G protein-coupled receptor GPR132

    Shehata, M. A., Christensen, H. B., Isberg, V., Pedersen, D. S., Bender, A., Bräuner, Hans & Gloriam, David E., 2015, In: RSC Advances. 5, p. 48551-48557 7 p.

    Research output: Contribution to journal › Journal article › Research › peer-review

  82. Published

    Role of post-translational modifications on structure, function and pharmacology of class C G protein-coupled receptors

    Nørskov-Lauritsen, L. & Bräuner, Hans, 2015, In: European Journal of Pharmacology. 763, p. 233-240 8 p.

    Research output: Contribution to journal › Journal article › Research › peer-review

  83. Published

    Synthesis and pharmacological evaluation of N-benzyl substituted 4-bromo-2,5-dimethoxyphenethylamines as 5-HT2A/2C partial agonists

    Hansen, M., Jacobsen, S. E., Plunkett, S., Liebscher, G. E., McCorvy, J. D., Bräuner, Hans & Kristensen, Jesper Langgaard, 2015, In: Bioorganic & Medicinal Chemistry. 23, 14, p. 3933-3937 5 p.

    Research output: Contribution to journal › Journal article › Research › peer-review

  84. 2014
  85. Published

    Introduction to special issue in honor of Professor Povl Krogsgaard-Larsen

    Bräuner, Hans & Schousboe, Arne, Oct 2014, In: Neurochemical Research. 39, 10, p. 1845-6 2 p.

    Research output: Contribution to journal › Journal article › Research

  86. Published

    mGluR5: Exploration of Orthosteric and Allosteric Ligand Binding Pockets and Their Applications to Drug Discovery

    Mølck, C., Harpsøe, Kasper, Gloriam, David E., Mathiesen, Jesper M., Nielsen, S. M. & Bräuner, Hans, Oct 2014, In: Neurochemical Research. 39, 10, p. 1862-1875 14 p.

    Research output: Contribution to journal › Journal article › Research › peer-review

  87. Published

    Pharmacological Identification of a Guanidine-Containing β-Alanine Analogue with Low Micromolar Potency and Selectivity for the Betaine/GABA Transporter 1 (BGT1)

    Al-Khawaja, A. M. A., Petersen, J. G., Damgaard, M., Jensen, M. H., Vogensen, S. B., Lie, M. E. K., Kragholm, B., Bräuner, Hans, Clausen, Rasmus Prætorius, Frølund, Bente & Wellendorph, Petrine, 23 May 2014, In: Neurochemical Research. 39, 10, p. 1988-1996 9 p.

    Research output: Contribution to journal › Journal article › Research › peer-review

  88. Published

    Computer-aided discovery of aromatic L-α-amino acids as agonists of the orphan G protein-coupled receptor GPR139

    Ísberg, V., Andersen, K. B., Bisig, C., Dietz, G. P., Bräuner, Hans & Gloriam, David E., 14 May 2014, In: Journal of Chemical Information and Modeling. 54, 6, p. 1553-1557 5 p.

    Research output: Contribution to journal › Journal article › Research › peer-review

  89. Published

    Real-time trafficking and signaling of the glucagon-like peptide-1 receptor

    Roed, S. N., Wismann, P., Underwood, C. R., Kulahin, N., Iversen, H., Cappelen, K. A., Schäffer, L., Lehtonen, J., Hecksher-Soerensen, J., Secher, A., Mathiesen, Jesper M., Bräuner, Hans, Whistler, J. L., Knudsen, S. M. & Waldhoer, M., Feb 2014, In: Molecular and Cellular Endocrinology. 382, 2, p. 938-949 12 p.

    Research output: Contribution to journal › Journal article › Research › peer-review

  90. Published

    Synthesis and structure-activity relationships of N-benzyl phenethylamines as 5-HT2A/2C agonists

    Hansen, M., Phonekeo, K., Paine, J. S., Leth-Petersen, S., Begtrup, M., Bräuner, Hans & Kristensen, Jesper Langgaard, 7 Jan 2014, In: A C S Chemical Neuroscience. 5, 3, p. 243-249 8 p.

    Research output: Contribution to journal › Journal article › Research › peer-review

  91. Published

    G protein-coupled receptor signaling analysis using homogenous time-resolved Förster resonance energy transfer (HTRF®) technology.

    Nørskov-Lauritsen, L., Thomsen, A. R. B. & Bräuner, Hans, 2014, In: International Journal of Molecular Sciences (Online). 15, 2, p. 2554-2572

    Research output: Contribution to journal › Journal article › Research › peer-review

  92. Published

    Promiscuous Seven Transmembrane Receptors Sensing L-α-amino Acids

    Smajilovic, S., Wellendorph, Petrine & Bräuner, Hans, 2014, In: Current Pharmaceutical Design. 20, p. 2693-702 10 p.

    Research output: Contribution to journal › Journal article › Research › peer-review

  93. Published

    The G protein-coupled receptor, class C, group 6, subtype A (GPRC6A) receptor: from cloning to physiological function

    Clemmensen, Christoffer, Smajilovic, S., Wellendorph, Petrine & Bräuner, Hans, 2014, In: British Journal of Pharmacology. 171, 5, p. 1129-1141

    Research output: Contribution to journal › Journal article › Research › peer-review

  94. 2013
  95. Published

    Delineation of the GPRC6A Receptor Signaling Pathways Using a Mammalian Cell Line Stably Expressing the Receptor

    Jacobsen, S. E., Nørskov-Lauritsen, L., Thomsen, A. R. B., Smajilovic, S., Wellendorph, Petrine, Larsson, N. H. P., Lehmann, A., Bhatia, V. K. & Bräuner, Hans, Nov 2013, In: Journal of Pharmacology and Experimental Therapeutics. 347, 2, p. 298-309 12 p.

    Research output: Contribution to journal › Journal article › Research › peer-review

  96. Published

    Oral L-Arginine Stimulates GLP-1 Secretion to Improve Glucose Tolerance in Male Mice

    Clemmensen, C., Smajilovic, S., Smith, E. P., Woods, S. C., Bräuner, Hans, Seeley, R. J., D'Alessio, D. A. & Ryan, K. K., Nov 2013, In: Endocrinology. 154, 11, p. 3978-83 6 p.

    Research output: Contribution to journal › Journal article › Research

  97. Published

    The orthosteric GABAA receptor ligand Thio-4-PIOL displays distinctly different functional properties at synaptic and extrasynaptic receptors

    Hoestgaard-Jensen, K., O'Connor, R. M., Dalby, N. O., Simonsen, C., Finger, B. C., Golubeva, A., Hammer, H., Bergmann, M. L., Kristiansen, Uffe, Krogsgaard-Larsen, Povl, Bräuner, Hans, Ebert, B., Frølund, Bente, Cryan, J. F. & Jensen, Anders A., Oct 2013, In: British Journal of Pharmacology. 170, 4, p. 919-32 14 p.

    Research output: Contribution to journal › Journal article › Research › peer-review

  98. Published

    GABA-B-agonistic activity of certain baclofen homologues

    Attia, M., Herdeis, C. & Bräuner, Hans, 22 Aug 2013, In: Molecules. 18, 9, p. 10266-10284

    Research output: Contribution to journal › Journal article › Research › peer-review

  99. Published

    Structure-based discovery of antagonists for GluN3-containing N-methyl-D-aspartate receptors

    Kvist, T., Greenwood, J. R., Hansen, K. B., Traynelis, S. F. & Bräuner, Hans, 22 Aug 2013, In: Neuropharmacology. 75, p. 324-336 13 p.

    Research output: Contribution to journal › Journal article › Research › peer-review

  100. Published

    Interactions between calcium and phosphorus in the regulation of the production of fibroblast growth factor 23 in vivo

    Quinn, S. J., Thomsen, A. R. B., Pang, J. L., Kantham, L., Brown, E. M., Bräuner, Hans, Pollak, M. & Goltzman, D., 1 Feb 2013, In: American Journal of Physiology: Endocrinology and Metabolism. 304, 3, p. E310-320

    Research output: Contribution to journal › Journal article › Research › peer-review

  101. Published

    3-Substituted 2-phenyl-indoles: Privileged structures for medicinal chemistry

    Johansson, K. H., Jørgensen, T. B., Gloriam, David E., Bräuner, Hans & Pedersen, D. S., 21 Jan 2013, In: R S C Advances. 3, 3, p. 945-960

    Research output: Contribution to journal › Journal article › Research › peer-review

  102. Published

    Synthesis and pharmacological characterization of certain baclofen analogues

    Attia, M. I., Herdeis, C. & Bräuner, Hans, 1 Jan 2013, In: Digest Journal of Nanomaterials and Biostructures. 8, 1, p. 139-149

    Research output: Contribution to journal › Journal article › Research › peer-review

  103. Published

    Crystal structure and pharmacological characterization of a novel N-methyl-D-aspartate (NMDA) receptor antagonist at the GluN1 glycine binding site

    Kvist, T., Steffensen, T. B., Greenwood, J. R., Mehrzad Tabrizi, F., Hansen, K. B., Gajhede, Michael, Pickering, Darryl S, Traynelis, S. F., Kastrup, Jette Sandholm Jensen & Bräuner, Hans, 2013, In: The Journal of Biological Chemistry. 288, p. 33124-35 12 p.

    Research output: Contribution to journal › Journal article › Research › peer-review

  104. Published

    Discovery of a subtype-selective of the human betaine/GABA transporter 1 (BGT-1) with a non-competitive pharmacological profile

    Kragholm, B., Kvist, T., Madsen, K. K., Jørgensen, L., Vogensen, S. B., Schousboe, Arne, Clausen, Rasmus Prætorius, Jensen, Anders A. & Bräuner, Hans, 2013, In: Biochemical Pharmacology. 86, p. 521-528

    Research output: Contribution to journal › Journal article › Research › peer-review

  105. Published

    Enhanced voluntary wheel running in GPRC6A receptor knockout mice

    Clemmensen, Christoffer, Pehmøller, C., Klein, A. B., Ratner, C., Wojtaszewski, Jørgen F P & Bräuner, Hans, 2013, In: Physiology & Behavior. 118, p. 144-151 7 p.

    Research output: Contribution to journal › Journal article › Research › peer-review

  106. Published

    Increased susceptibility to diet-induced obesity in GPRC6A receptor knockout mice

    Clemmensen, Christoffer, Smajilovic, S., Madsen, A. N., Klein, A. B., Holst, Birgitte & Bräuner, Hans, 2013, In: Journal of Endocrinology. 217, 2, p. 151-60 10 p.

    Research output: Contribution to journal › Journal article › Research › peer-review

  107. Published

    Synthesis of the calcilytic ligand NPS2143

    Johansson, K. H., Cailly, T. B. G., Thomsen, A. R. B., Bräuner, Hans & Pedersen, D. S., 2013, In: Beilstein Journal of Organic Chemistry. 9, p. 1383-1387

    Research output: Contribution to journal › Journal article › Research › peer-review

  108. Published

    The L-alpha-amino acid receptor GPRC6A is expressed in the islets of Langerhans but is not involved in L-arginine-induced insulin release

    Smajilovic, S., Clemmensen, Christoffer, Johansen, L. D., Wellendorph, Petrine, Holst, Jens Juul, Thams, P. G., Ogo, E. & Bräuner, Hans, 2013, In: Amino Acids. 44, 2, p. 383-390 8 p.

    Research output: Contribution to journal › Journal article › Research › peer-review

  109. Published

    cAMP biosensors applied in molecular pharmacological studies of G protein-coupled receptors

    Mathiesen, Jesper M., Vedel, L. & Bräuner, Hans, 2013, In: Methods in Enzymology. 522, p. 191-207 17 p.

    Research output: Contribution to journal › Journal article › Research

  110. 2012
  111. Published

    Strontium is a biased agonist of the calcium-sensing receptor in rat medullary thyroid carcinoma 6-23 cells

    Thomsen, A. R. B., Worm, J., Jacobsen, S. E., Stahlhut, M., Latta, M. & Bräuner, Hans, Dec 2012, In: Journal of Pharmacology and Experimental Therapeutics. 343, 3, p. 638-49 12 p.

    Research output: Contribution to journal › Journal article › Research › peer-review

  112. Published

    Novel strategies in drug discovery of the calcium-sensing receptor based on biased signaling

    Thomsen, A. R. B., Smajilovic, S. & Bräuner, Hans, 1 Sep 2012, In: Current Drug Targets. 13, 10, p. 1324-35 12 p.

    Research output: Contribution to journal › Journal article › Research › peer-review

  113. Published

    Molecular pharmacology of human NMDA receptors

    Hedegaard, M., Hansen, K. B., Andersen, K. T., Bräuner, Hans & Traynelis, S. F., Sep 2012, In: Neurochemistry International. 61, 4, p. 601-609

    Research output: Contribution to journal › Journal article › Research › peer-review

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