Fredrik Björkling
Emeritus
Medicinal Chemistry
Jagtvej 162
2100 København Ø
- 2021
- Published
Structural Basis of Metallo-β-lactamase Inhibition by N-Sulfamoylpyrrole-2-carboxylates
Farley, A. J. M., Ermolovich, Y., Calvopiña, K., Rabe, P., Panduwawala, T., Brem, J., Björkling, Fredrik & Schofield, C. J., 2021, In: ACS Infectious Diseases. 7, 6, p. 1809–1817Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Synthesis of thiazole linked chalcones and their pyrimidine analogues as anticancer agents
Kesari, C., Rama, K. R., Sedighi, K., Stenvang, Jan, Björkling, Fredrik, Kankala, S. & Thota, N., 2021, In: Synthetic Communications. 51, 9, p. 1406-1416 11 p.Research output: Contribution to journal › Journal article › Research › peer-review
- 2020
- Published
Alternating Cationic-Hydrophobic Peptide/Peptoid Hybrids: Influence of Hydrophobicity on Antibacterial Activity and Cell Selectivity
Frederiksen, N., Hansen, Paul Robert, Zabicka, D., Tomczak, M., Urbas, M., Domraceva, I., Björkling, Fredrik & Franzyk, Henrik, 2020, In: ChemMedChem. 15, 24, p. 2544-2561Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Discovery of Novel Non-Steroidal Cytochrome P450 17A1 Inhibitors as Potential Prostate Cancer Agents
Wróbel, T. M., Rogova, O., Andersen, Kasper Langebjerg, Yadav, R., Brixius-Anderko, S., Scott, E. E., Olsen, L., Jørgensen, Flemming Steen & Björkling, Fredrik, 2020, In: International Journal of Molecular Sciences . 21, 14, p. 1-11 4868.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Synthesis of novel fluorophenylpyrazole-picolinamide derivatives and determination of their anticancer activity
Kankala, S., Rama, K. R., Kesari, C., Björkling, Fredrik, Nerella, S., Gundepaka, P., Guguloth, H. & Thota, N., 2020, In: Synthetic Communications. 50, 19, p. 2997-3006 10 p.Research output: Contribution to journal › Journal article › Research › peer-review
- 2019
- Published
Peptide/Peptoid Hybrid Oligomers: The Influence of Hydrophobicity and Relative Side-Chain Length on Antibacterial Activity and Cell Selectivity
Frederiksen, N., Hansen, Paul Robert, Björkling, Fredrik & Franzyk, Henrik, 4 Dec 2019, In: Molecules (Print Archive Edition). 24, 18 p., 4429.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Silver carbene complexes: An emerging class of anticancer agents
Kankala, S., Thota, N., Björkling, Fredrik, Taylor, M. K., Vadde, R. & Balusu, R., Mar 2019, In: Drug Development Research. 80, 2, p. 188-199Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Microwave-assisted solid-phase synthesis of antisense acpP peptide nucleic acid-peptide conjugates active against colistin- and tigecycline-resistant E. coli and K. pneumoniae
Hansen, A. M., Bonke, G., Hogendorf, W. F. J., Björkling, Fredrik, Nielsen, J., Kongstad, Kenneth Thermann, Zabicka, D., Tomczak, M., Urbas, M., Nielsen, Peter E. & Franzyk, Henrik, 2019, In: European Journal of Medicinal Chemistry. 168, p. 134-145 12 p.Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Triphenylcarbenium Tetrafluoroborate as an Efficient Catalyst in the Regioselective Reductive Ring Opening of Benzylidene Acetals of Carbohydrates
Thota, N., Björkling, Fredrik & Kankala, S., 2019, In: ChemistrySelect. 4, 27, p. 7976-7980Research output: Contribution to journal › Journal article › Research › peer-review
- 2018
- Published
Non-natural Amino Acid and Peptoid Building Blocks for Optimization of the Cell-Penetrating (R-X-R)n Motif
Wester, A., Björkling, Fredrik, Nieslen, P. & Franzyk, Henrik, Sep 2018, In: Journal of Peptide Science. 24, p. S94-S94Research output: Contribution to journal › Conference abstract in journal › Research › peer-review
ID: 8863737
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Imaging of treatment response to the combination of carboplatin and paclitaxel in human ovarian cancer xenograft tumors in mice using FDG and FLT PET
Research output: Contribution to journal › Journal article › Research › peer-review
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1262
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Non-natural Amino Acid and Peptoid Building Blocks for Optimization of the Cell-Penetrating (R-X-R)n Motif
Research output: Contribution to journal › Conference abstract in journal › Research › peer-review
Published -
262
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Novel Agonist Bioisosteres and Common Structure-Activity Relationships for The Orphan G Protein-Coupled Receptor GPR139
Research output: Contribution to journal › Journal article › Research › peer-review
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