Fredrik Björkling

Fredrik Björkling

Emeritus

ORCID: 0000-0001-7018-8334

Publication year:
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  1. 2024
  2. Published

    Studies of antibacterial activity (in vitro and in vivo) and mode of action for des-acyl tridecaptins (DATs)

    Couturier, C., Ronzon, Q., Lattanzi, G., Lingard, I., Coyne, S., Cazals, V., Dubarry, N., Yvon, S., Leroi-Geissler, C., Gracia, O. R., Teague, J., Sordello, S., Corbett, D., Bauch, C., Monlong, C., Payne, L., Taillier, T., Fuchs, H., Broenstrup, M., Harrison, P. H. & 10 others, Moynié, L., Lakshminarayanan, A., Gianga, T. M., Hussain, R., Naismith, J. H., Mourez, M., Bacqué, E., Björkling, Fredrik, Sabuco, J. F. & Franzyk, Henrik, 2024, In: European Journal of Medicinal Chemistry. 265, 20 p., 116097.

    Research output: Contribution to journal › Journal article › Research › peer-review

  3. Published

    Polymyxins with Potent Antibacterial Activity against Colistin-Resistant Pathogens: Fine-Tuning Hydrophobicity with Unnatural Amino Acids

    Jørgensen, Johan Storm, Harifi Mood, Elnaz, Knap, A. S. H., Nielsen, S. E., Nielsen, Peter E., Żabicka, D., Matias, C., Domraceva, I., Björkling, Fredrik & Franzyk, Henrik, 2024, In: Journal of Medicinal Chemistry. 67, 2, p. 1370–1383

    Research output: Contribution to journal › Journal article › Research › peer-review

  4. 2023
  5. Published

    Antimicrobial Peptides Incorporating Halogenated Marine-Derived Amino Acid Substituents

    Craig, A. J., Ermolovich, Y., Cameron, A., Rodler, A., Wang, H., Hawkes, J. A., Hubert, M., Björkling, Fredrik, Molchanova, N., Brimble, M. A., Moodie, L. W. K. & Svenson, J., 2023, In: ACS Medicinal Chemistry Letters. 14, 6, p. 802–809 8 p.

    Research output: Contribution to journal › Letter › Research › peer-review

  6. Published

    Selected strategies to fight pathogenic bacteria

    Plotniece, A., Sobolev, A., Supuran, C. T., Carta, F., Björkling, Fredrik, Franzyk, Henrik, Yli-Kauhaluoma, J., Augustyns, K., Cos, P., De Vooght, L., Govaerts, M., Aizawa, J., Tammela, P. & Žalubovskis, R., 2023, In: Journal of Enzyme Inhibition and Medicinal Chemistry. 38, 1, 27 p., 2155816.

    Research output: Contribution to journal › Review › Research › peer-review

  7. Published

    Structure-activity study of oncocin: On-resin guanidinylation and incorporation of homoarginine, 4-hydroxyproline or 4,4-difluoroproline residues

    Shaikh, Ashif Yasin, Björkling, Fredrik, Zabicka, D., Tomczak, M., Urbas, M., Domraceva, I., Kreicberga, A. & Franzyk, Henrik, 2023, In: Bioorganic Chemistry. 141, 11 p., 106876.

    Research output: Contribution to journal › Journal article › Research › peer-review

  8. Published

    Exploring the Potential of Sulfur Moieties in Compounds Inhibiting Steroidogenesis

    Wróbel, T. M., Sharma, K., Mannella, I., Oliaro-Bosso, S., Nieckarz, P., Du Toit, T., Voegel, C. D., Rojas Velazquez, M. N., Yakubu, J., Matveeva, A., Therkelsen, S., Jørgensen, Flemming Steen, Pandey, A. V., Pippione, A. C., Lolli, M. L., Boschi, D. & Björkling, Fredrik, 2023, In: Biomolecules. 13, 9, 18 p., 1349.

    Research output: Contribution to journal › Journal article › Research › peer-review

  9. Published

    Non-steroidal CYP17A1 Inhibitors: Discovery and Assessment

    Wróbel, T. M., Jørgensen, Flemming Steen, Pandey, A. V., Grudzińska, A., Sharma, K., Yakubu, J. & Björkling, Fredrik, 2023, In: Journal of Medicinal Chemistry. 66, 10, p. 6542–6566

    Research output: Contribution to journal › Review › Research › peer-review

  10. 2022
  11. Published

    Imitation of β-lactam binding enables broad-spectrum metallo-β-lactamase inhibitors

    Brem, J., Panduwawala, T., Hansen, J. U., Hewitt, J., Liepins, E., Donets, P., Espina, L., Farley, A. J. M., Shubin, K., Campillos, G. G., Kiuru, P., Shishodia, S., Krahn, D., Leśniak, R. K., Schmidt (Adrian), J., Calvopiña, K., Turrientes, M. C., Kavanagh, M. E., Lubriks, D., Hinchliffe, P. & 41 others, Langley, G. W., Aboklaish, A. F., Eneroth, A., Backlund, M., Baran, A. G., Nielsen, E. I., Speake, M., Kuka, J., Robinson, J., Grinberga, S., Robinson, L., McDonough, M. A., Rydzik, A. M., Leissing, T. M., Jimenez-Castellanos, J. C., Avison, M. B., Da Silva Pinto, S., Pannifer, A. D., Martjuga, M., Widlake, E., Priede, M., Hopkins Navratilova, I., Gniadkowski, M., Belfrage, A. K., Brandt, P., Yli-Kauhaluoma, J., Bacque, E., Page, M. G. P., Björkling, Fredrik, Tyrrell, J. M., Spencer, J., Lang, P. A., Baranczewski, P., Cantón, R., McElroy, S. P., Jones, P. S., Baquero, F., Suna, E., Morrison, A., Walsh, T. R. & Schofield, C. J., 2022, In: Nature Chemistry. 14, p. 15–24

    Research output: Contribution to journal › Journal article › Research › peer-review

  12. Published

    Synthesis and Structure–Activity Relationships of Novel Non-Steroidal CYP17A1 Inhibitors as Potential Prostate Cancer Agents

    Wróbel, T. M., Rogova, O., Sharma, K., Velazquez, M. N. R., Pandey, A. V., Jørgensen, Flemming Steen, Arendrup, Frederic Schrøder, Andersen, Kasper Langebjerg & Björkling, Fredrik, 2022, In: Biomolecules. 12, 2, 165.

    Research output: Contribution to journal › Journal article › Research › peer-review

  13. 2021
  14. Published

    Structural Basis of Metallo-β-lactamase Inhibition by N-Sulfamoylpyrrole-2-carboxylates

    Farley, A. J. M., Ermolovich, Y., Calvopiña, K., Rabe, P., Panduwawala, T., Brem, J., Björkling, Fredrik & Schofield, C. J., 2021, In: ACS Infectious Diseases. 7, 6, p. 1809–1817

    Research output: Contribution to journal › Journal article › Research › peer-review

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ID: 8863737