Frederik Diness

Frederik Diness

Guest researcher, Guest Researcher

Member of:

    ORCID: 0000-0001-5098-7198

    Publication year:
    All
    1 - 45 out of 45Page size: 50
    1. 2024
    2. Accepted/In press

      Self-Promoted Glycosylation of Carbamoylated Peptides on Solid Phase

      Fischer, Niklas Henrik, Vævest, B. N., Dam, Andreas Ketilsø, Diness, Frederik & Pedersen, Christian Marcus, 2024, (Accepted/In press) In: ChemPlusChem. e202400066.

      Research output: Contribution to journal › Journal article › Research › peer-review

    3. 2023
    4. Published

      Chemical modification of proteins - challenges and trends at the start of the 2020s

      Fischer, Niklas Henrik, Oliveira, M. T. & Diness, Frederik, 2023, In: Biomaterials Science. 11, 3, p. 719–748 30 p.

      Research output: Contribution to journal › Review › Research › peer-review

    5. 2022
    6. Published

      Carbon dioxide enhances sulphur-selective conjugate addition reactions

      Yang, Y., Fischer, Niklas Henrik, Oliveira, M. T., Hadaf, Gul Barg, Liu, J., Brock-Nannestad, Theis, Diness, Frederik & Lee, Ji-Woong, 2022, In: Organic & Biomolecular Chemistry. 20, 22, p. 4526–4533 8 p.

      Research output: Contribution to journal › Journal article › Research › peer-review

    7. Published

      Lignin-Inspired Polybenzylethersulfone Synthesis via SNAr Reaction

      Nikitin, S., Lie, Yann & Diness, Frederik, 2022, In: Macromolecular Chemistry and Physics. 223, 13, p. 2100484 8 p.

      Research output: Contribution to journal › Journal article › Research › peer-review

    8. Published

      Radiolabeled albumin through SNAr of cysteines as a potential pretargeting theranostic agent

      Fischer, Niklas Henrik, van den Broek, S. I. L. I., Herth, Matthias Manfred & Diness, Frederik, 2022, In: RSC Advances. 12, 54, p. 35032-35036

      Research output: Contribution to journal › Journal article › Research › peer-review

    9. Published

      Tuning Peptide Structure and Function through Fluorobenzene Stapling

      Fischer, Niklas Henrik, Fumi, E., Oliveira, M. T., Thulstrup, Peter Waaben & Diness, Frederik, 2022, In: Chemistry: A European Journal. 28, 8, 7 p., e202103788.

      Research output: Contribution to journal › Journal article › Research › peer-review

    10. 2021
    11. Published

      C-Terminal lactamization of peptides

      Fischer, Niklas Henrik, Nielsen, D. S., Palmer, D., Meldal, Morten Peter & Diness, Frederik, 2021, In: Chemical Communications. 57, 7, p. 895-898 4 p.

      Research output: Contribution to journal › Journal article › Research › peer-review

    12. 2020
    13. Published

      Recent Fascinating Aspects of the CuAAC Click Reaction

      Meldal, Morten Peter & Diness, Frederik, 1 Jun 2020, In: Trends in Chemistry. 2, 6, p. 569-584 16 p.

      Research output: Contribution to journal › Review › Research › peer-review

    14. Published

      Design and Combinatorial Development of Shield-1 Peptide Mimetics Binding to Destabilized FKBP12

      Madsen, D., Jørgensen, F. P., Palmer, D., Roux, M. E., Olsen, J. V., Bols, Mikael, Schoffelen, S., Diness, Frederik & Meldal, Morten Peter, 2020, In: ACS Combinatorial Science. 22, 3, p. 156-164

      Research output: Contribution to journal › Journal article › Research › peer-review

    15. Published

      Dihydroquinazolinones via A3‐Type Reactions of N‐Carbamoyliminium Ions

      Wang, Y., Oliveira, M. T., Madsen, D., Thompson, A., Meldal, Morten Peter & Diness, Frederik, 2020, In: Chemistry: A European Journal. 26, 68, p. 15825-15829 6 p.

      Research output: Contribution to journal › Letter › Research › peer-review

    16. 2019
    17. Published

      Azotides as Modular Peptide-Based Ligands for Asymmetric Lewis Acid Catalysis

      Jacobsen, C. B., Nielsen, D. S., Meldal, Morten Peter & Diness, Frederik, 7 Jun 2019, In: Journal of Organic Chemistry. 84, 11, p. 6940-6945 6 p.

      Research output: Contribution to journal › Journal article › Research › peer-review

    18. Published

      Computational Evolution of Threonine-Rich β-Hairpin Peptides Mimicking Specificity and Affinity of Antibodies

      Hu, H., Kofoed, Christian, Li, M., Gonçalves, J. P. L., Hansen, J., Wolfram, M., Hansen, Axel Kornerup, Hansen, Camilla Hartmann Friis, Diness, Frederik, Schoffelen, S. & Meldal, Morten Peter, 27 Feb 2019, In: ACS Central Science. 5, 2, p. 259-269 11 p.

      Research output: Contribution to journal › Journal article › Research › peer-review

    19. Published

      Twists or turns: stabilising alpha vs. beta turns in tetrapeptides

      Hoang, H. N., Hill, T. A., Ruiz-Gómez, G., Diness, Frederik, Mason, J. M., Wu, C., Abbenante, G., Shepherd, N. E. & Fairlie, D. P., 2019, In: Chemical Science. 10, 45, p. 10595-10600

      Research output: Contribution to journal › Journal article › Research › peer-review

    20. Published

      X-ray diffraction data as a source of the vibrational free-energy contribution in polymorphic systems

      Kofoed, P. M., Hoser, A. A., Diness, Frederik, Capelli, S. C. & Madsen, Anders Østergaard, 2019, In: IUCrJ. 6, 4, p. 558-571 14 p.

      Research output: Contribution to journal › Journal article › Research › peer-review

    21. 2018
    22. Published

      Sustainable Flow Synthesis of Encoded Beads for Combinatorial Chemistry and Chemical Biology

      Hu, H., Nikitin, S., Berthelsen, A. B., Diness, Frederik, Schoffelen, S. & Meldal, Morten Peter, 13 Aug 2018, In: ACS Combinatorial Science. 20, 8, p. 492-498 7 p.

      Research output: Contribution to journal › Journal article › Research › peer-review

    23. Published

      Rational Tuning of Fluorobenzene Probes for Cysteine-Selective Protein Modification

      Embaby, A. M., Schoffelen, S., Kofoed, Christian, Meldal, Morten Peter & Diness, Frederik, 2 Jul 2018, In: Angewandte Chemie International Edition. 57, 27, p. 8022-8026 5 p.

      Research output: Contribution to journal › Journal article › Research › peer-review

    24. Published

      Metallo-Organozymes with Specific Proteolytic Activity

      Embaby, A. M., Lelieveldt, L. P. W. M., Diness, Frederik & Meldal, Morten Peter, 2018, In: Chemistry - A European Journal. 24, 66, p. 17424-17428 5 p.

      Research output: Contribution to journal › Journal article › Research › peer-review

    25. Published

      Synthesis and stability of strongly acidic benzamide derivatives

      Diness, Frederik, Bjerrum, N. J. & Begtrup, M., 2018, In: Beilstein Journal of Organic Chemistry. 14, p. 523-530 8 p.

      Research output: Contribution to journal › Journal article › Research › peer-review

    26. 2017
    27. Published

      Advances in merging triazoles with peptides and proteins

      Diness, Frederik, Schoffelen, S. & Meldal, Morten Peter, 2017, [Awaiting title]. Springer, p. 1-38 38 p. (Topics in Heterocyclic Chemistry).

      Research output: Chapter in Book/Report/Conference proceeding › Book chapter › Research › peer-review

    28. Published

      Click-Chemistry-Mediated Synthesis of Selective Melanocortin Receptor 4 Agonists

      Palmer, D., Gonçalves, J. P. L., Hansen, L. V., Wu, B., Hald, H., Schoffelen, S., Diness, Frederik, Le Quement, S. T., Nielsen, Thomas Eiland & Meldal, Morten Peter, 2017, In: Journal of Medicinal Chemistry. 60, 21, p. 8716-8730 15 p.

      Research output: Contribution to journal › Journal article › Research › peer-review

    29. Published

      Diversity-Oriented Syntheses by Combining CuAAC and Stereoselective INCIC Reactions with Peptides

      Wang, Y., Madsen, Anders Østergaard, Diness, Frederik & Meldal, Morten Peter, 2017, In: Chemistry - A European Journal. 23, 56, p. 13869–13874 6 p.

      Research output: Contribution to journal › Journal article › Research › peer-review

    30. Published

      Mechanism and Scope of Base-Controlled Catalyst-Free N-Arylation of Amines with Unactivated Fluorobenzenes

      Jacobsen, C. B., Meldal, Morten Peter & Diness, Frederik, 2017, In: Chemistry: A European Journal. 23, 4, p. 846-851 6 p.

      Research output: Contribution to journal › Journal article › Research › peer-review

    31. 2016
    32. Published

      C-Terminally modified peptides via cleavage of the HMBA linker by O-, N- or S-nucleophiles

      Hansen, J., Diness, Frederik & Meldal, Morten Peter, 2016, In: Organic & Biomolecular Chemistry. 14, 12, p. 3238-3245 8 p.

      Research output: Contribution to journal › Journal article › Research › peer-review

    33. Published

      Comparative studies of adhesion peptides based on L- or D-amino acids

      Nikitin, S., Palmer, D., Meldal, Morten Peter & Diness, Frederik, 2016, In: Journal of Peptide Science. 22, 10, p. 642-646 5 p.

      Research output: Contribution to journal › Journal article › Research › peer-review

    34. 2015
    35. Published

      Fmox: a base-labile aldehyde protecting group

      Diness, Frederik & Meldal, Morten Peter, 2015, In: European Journal of Organic Chemistry. 2015, 7, p. 1433-1436 4 p.

      Research output: Contribution to journal › Journal article › Research › peer-review

    36. 2014

    37. Comparative α-helicity of cyclic pentapeptides in water

      de Araujo, A. D., Hoang, H. N., Kok, W. M., Diness, Frederik, Gupta, P., Driver, R. W., Price, D. A., Liras, S. & Fairlie, D. P., 2014, In: Angewandte Chemie International Edition. 53, 27, p. 6965-6969 5 p.

      Research output: Contribution to journal › Journal article › Research › peer-review

    38. Published

      Constraining cyclic peptides to mimic protein structure motifs

      Hill, T. A., Shepherd, N. E., Diness, Frederik & Fairlie, D. P., 2014, In: Angewandte Chemie - International Edition. 53, 48, p. 13020-13041 22 p.

      Research output: Contribution to journal › Journal article › Research › peer-review

    39. Published

      Sequential direct SNAr reactions of pentafluorobenzenes with azole or indole derivatives

      Diness, Frederik & Begtrup, M., 2014, In: Organic Letters. 16, 11, p. 3130-3133 4 p.

      Research output: Contribution to journal › Journal article › Research › peer-review

    40. 2012
    41. Published

      Total synthesis, structure, and oral absorption of a thiazole cyclic peptide, sanguinamide A

      Nielsen, D. S., Hoang, H. N., Lohman, R., Diness, Frederik & Fairlie, D. P., 16 Nov 2012, In: Organic Letters. 14, 22, p. 5720-3 4 p.

      Research output: Contribution to journal › Journal article › Research › peer-review

    42. Published

      Biophysical characterization of the proton-coupled oligopeptide transporter YjdL

      Jensen, J. M., Simonsen, F. C., Mastali, A., Hald, H., Lillebro, I., Diness, Frederik, Olsen, L. & Mirza, Osman Asghar, Nov 2012, In: Peptides. 38, 1, p. 89-93 5 p.

      Research output: Contribution to journal › Journal article › Research › peer-review

    43. Published

      Fluorobenzene derivatives as multifunctional tools

      Diness, Frederik, Begtrup, M. B. & Fairlie, D. P., 25 Mar 2012, In: American Chemical Society. Abstracts of Papers (at the National Meeting). 243

      Research output: Contribution to journal › Journal article › Research › peer-review

    44. Published

      Catalyst-Free N-Arylation Using Unactivated Fluorobenzenes

      Diness, Frederik & Fairlie, D. P., 2012, In: Angewandte Chemie International Edition. 51, 32, p. 8012-8016

      Research output: Contribution to journal › Journal article › Research › peer-review

    45. Published

      D-amino acid adhesion peptides by combinatorial selection: control of cellular growth on inert surfaces

      Meldal, Morten Peter, Wu, B., Diness, Frederik, Michael, R., Hagel, G., Nygaard, J. & Martinez, K., 2012, In: Journal of Peptide Science. 18, S1, p. S21-S22 2 p., IL1.

      Research output: Contribution to journal › Conference abstract in journal › Research › peer-review

    46. 2011
    47. Published

      Identifying a compound modifying a cellular response, comprises attaching cells having a reporter system onto solid supports, releasing a library member, screening and identifying target cells

      Hagel, G., Thastrup, Ole, Meldal, Morten Peter, Norrild, J. C., Hentzer, M., Norrild, J. & Diness, Frederik, 29 Dec 2011, IPC No. G01N 35/ 00 A N, Patent No. US2011319274, Priority date 25 May 2005, Priority No. WO2005DK00348

      Research output: Patent

    48. Published

      Synthesis of the thiazole-thiazoline fragment of largazole analogues

      Diness, Frederik, Nielsen, D. S. & Fairlie, D. P., 2 Dec 2011, In: Journal of Organic Chemistry. 76, 23, p. 9845-9851

      Research output: Contribution to journal › Journal article › Research › peer-review

    49. 2010
    50. Published

      Amino acid derived 1,4-dialkyl substituted imidazolones

      Diness, Frederik & Meldal, Morten Peter, 11 Mar 2010, In: Biopolymers. 94, 2, p. 236-241

      Research output: Contribution to journal › Journal article › Research › peer-review

    51. Ralph F. Hirschmann award address 2009: merger of organic chemistry with peptide diversity

      Meldal, Morten Peter, Tornøe, C. W., Nielsen, T. E., Diness, Frederik, Le Quement, S. T., Christensen, C. A., Jensen, J. F., Worm-Leonhard, K., Groth, T., Bouakaz, L., Wu, B., Hagel, G. & Keinicke, L., 2010, In: Biopolymers. 94, 2, p. 161-182 22 p.

      Research output: Contribution to journal › Journal article › Research › peer-review

    52. 2009
    53. Published

      Imidazolones in diastereoselective cyclization reactions and Cu(II)-catalysed cross-coupling reactions

      Diness, Frederik & Meldal, Morten Peter, 20 Jul 2009, In: Chemistry: A European Journal. 15, 29, p. 7044-7 4 p.

      Research output: Contribution to journal › Journal article › Research › peer-review

    54. 2006
    55. Published

      Solid-phase synthesis of tetrahydro-beta-carbolines and tetrahydroisoquinolines by stereoselective intramolecular N-carbamyliminium Pictet-Spengler reactions

      Diness, Frederik & Meldal, Morten Peter, 25 Oct 2006, In: Chemistry: A European Journal. 12, 31, p. 8056-66 11 p.

      Research output: Contribution to journal › Journal article › Research › peer-review

    56. Published

      Solid-phase reactions of N-carbamyliminium ions: from amino aldehydes to on-bead GPCR-screening : PH.D. thesis

      Diness, Frederik, 2006, Copenhagen: Department of Medical Chemistry, Danish University of Pharmaceutical Sciences. 179 p.

      Research output: Book/Report › Book › Research

    57. 2005
    58. Published

      Dual approach to intramolecular carbamoyliminium activated solid phase Pictet-Spengler reactions

      Diness, Frederik & Meldal, Morten Peter, 2005, Peptides 2004, Proceedings. p. 208-209

      Research output: Chapter in Book/Report/Conference proceeding › Book chapter › Research › peer-review

    59. 2004
    60. Published

      Probing the aglycon binding site of a beta-glucosidase: a collection of C-1-modified 2,5-dideoxy-2,5-imino-D-mannitol derivatives and their structure-activity relationships as competitive inhibitors

      Wrodnigg, T. M., Diness, Frederik, Gruber, C., Häusler, H., Lundt, I., Rupitz, K., Steiner, A. J., Stütz, A. E., Tarling, C. A., Withers, S. G. & Wölfler, H., 1 Jul 2004, In: Bioorganic & Medicinal Chemistry. 12, 13, p. 3485-95 11 p.

      Research output: Contribution to journal › Journal article › Research › peer-review

    61. Published

      Synthesis of 3-Boc-(1,3)-oxazinane-protected amino aldehydes from amino acids and their conversion into urea precursors. Novel building blocks for combinatorial synthesis

      Diness, Frederik, Beyer, J. & Meldal, Morten Peter, Apr 2004, In: Molecular Informatics. 23, 2-3, p. 130-144

      Research output: Contribution to journal › Journal article › Research › peer-review

    62. Published

      INTRAMOLECULAR CARBAMOYLIMINIUM ACTIVATED SOLID PHASE PICTET-SPENGLER REACTIONS. TOWARDS MCR AGONISTS

      Diness, Frederik, Beyer, J. & Meldal, Morten Peter, 2004, In: Journal of Peptide Science. 10, p. 126-126

      Research output: Contribution to journal › Journal article › Research › peer-review

    63. 2003
    64. Published

      The Pictet-Spengler reaction in solid-phase combinatorial chemistry

      Nielsen, T. E., Diness, Frederik & Meldal, Morten Peter, Nov 2003, In: Current Opinion in Drug Discovery & Development. 6, 6, p. 801-14 14 p.

      Research output: Contribution to journal › Journal article › Research › peer-review

    ID: 33654400