Flemming Steen Jørgensen
Professor
Structural Biology
Universitetsparken 2
2100 København Ø
- Published
In silico predictions of hERG channel blockers in drug discovery: from ligand-based and target-based approaches to systems chemical biology
Taboureau, O. & Jørgensen, Flemming Steen, Jun 2011, In: Combinatorial Chemistry & High Throughput Screening. 14, 5, p. 375-387Research output: Contribution to journal › Journal article › Research › peer-review
- Published
A diversity optimized combinatorial library for the identification of Fc-fragment binding ligands
Nielsen, A. L., Jørgensen, Flemming Steen, Olsen, L., Christensen, S. F., Benie, A. J., Bjørnholm, T. & St. Hilaire, P. M., 2010, In: Biopolymers. 94, 2, p. 192-205Research output: Contribution to journal › Journal article › Research › peer-review
- Published
A quantitative structure-activity relationship for translocation of tripeptides via the human proton-coupled peptide transporter, hPEPT1 (SLC15A1)
Omkvist, D. H., Larsen, S. B., Nielsen, C. U., Steffansen, B., Olsen, L., Jørgensen, Flemming Steen & Larsen, Birger Brodin, 2010, In: The AAPS Journal. 12, 3, p. 385-396Research output: Contribution to journal › Journal article › Research › peer-review
- Published
A robust force field based method for calculating conformational energies of charged drug-like molecules
Pøhlsgaard, J., Harpsøe, Kasper, Jørgensen, Flemming Steen & Olsen, L., 2012, In: Journal of Chemical Information and Modeling. 52, 2, p. 409-419Research output: Contribution to journal › Journal article › Research › peer-review
- Published
A steered molecular dynamics study of binding and translocation processes in the GABA transporter
Skovstrup, S., David, L., Taboureau, O. & Jørgensen, Flemming Steen, 2012, In: P L o S One. 7, 6, p. e39360Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Biostructure-based drug design
Jørgensen, Flemming Steen & Kastrup, Jette Sandholm Jensen, 2010, Textbook of drug design and discovery. Krogsgaard-Larsen, P., Strømgaard, K. & Madsen, U. (eds.). 4 ed. Boca Raton: CRC Press, p. 29-42Research output: Chapter in Book/Report/Conference proceeding › Book chapter › Education
- Published
Classification of cytochrome P450 1A2 inhibitors and noninhibitors by machine learning techniques
Poongavanam, V., Taboureau, O., Oostenbrink, C., Vermeulen, N. P. E., Olsen, L. & Jørgensen, Flemming Steen, 2009, In: Drug Metabolism and Disposition. 37, 3, p. 658-664Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Computational prediction of binding affinity for CYP1A2-ligand complexes using empirical free energy calculations
Poongavanam, V., Olsen, L., Jørgensen, Flemming Steen, Vermeulen, N. P. E. & Oostenbrink, C., 2010, In: Drug Metabolism and Disposition. 38, 8, p. 1347-1354Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Computational prediction of solubilizers' effect on partitioning
Høst, J., Christensen, I. T., Jørgensen, Flemming Steen, Frøkjær, Sven & Hovgaard, L., 2007, In: Internation Journal of Pharmaceutics. 329, 1-2, p. 46-52Research output: Contribution to journal › Journal article › Research › peer-review
- Published
Computeren er medicinalkemikerens arbejdshest
Larsen, S. B., Olsen, L. & Jørgensen, Flemming Steen, 2009, In: Lægemiddelforskning. p. 7-9Research output: Contribution to journal › Journal article › Communication
ID: 1302104
Most downloads
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2006
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Synthesis and antiangiogenic activity of N-alkylated levamisole derivatives
Research output: Contribution to journal › Journal article › Research › peer-review
Published -
1967
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Forbedret optagelse af lægemidler i organismen: computeren viser vejen
Research output: Contribution to journal › Journal article › Research
Published -
1525
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Design of prodrugs targeting the intestinal di/tri‐peptide transporter hPEPT1 (SLC15A1
Research output: Contribution to conference › Conference abstract for conference › Research › peer-review
Published