Darryl S Pickering

Darryl S Pickering

Associate Professor


  1. 2016
  2. Published

    γ-Glutamyl-dipeptides: Easy tools to rapidly probe the stereoelectronic properties of ionotropic glutamate receptor binding pocket

    Tamborini, L., Nicosia, V., Conti, P., Dall'Oglio, F., De Micheli, C., Nielsen, Birgitte, Jensen, Anders A., Pickering, Darryl S & Pinto, A., 1 Dec 2016, In: Tetrahedron. 72, 51, p. 8586-8492 7 p.

    Research output: Contribution to journalJournal articlepeer-review

  3. Published

    Effects of sertraline, duloxetine, vortioxetine, and idazoxan in the rat affective bias test

    Refsgaard, L. K., Haubro, K., Pickering, Darryl S, Stuart, S., Robinson, E. & Andreasen T., Jesper, 14 Oct 2016, In: Psychopharmacology. 233, 21, p. 3763-3770 8 p.

    Research output: Contribution to journalJournal articlepeer-review

  4. Published

    Positive allosteric modulation of AMPA receptors differentially modulates the behavioural effects of citalopram in mouse models of antidepressant and anxiolytic action

    Fitzpatrick, C. M., Larsen, M., Madsen, L., Pickering, Darryl S, Clausen, Rasmus Prætorius & Andreasen T., Jesper, 26 Jun 2016, In: Behavioural Pharmacology. 27, 6, p. 549-555 7 p.

    Research output: Contribution to journalJournal articlepeer-review

  5. Published

    Effects of the dimeric PSD-95 inhibitor UCCB01-144 in mouse models of pain, cognition and motor function

    Andreasen T., Jesper, Nasser, A., Caballero-Puntiverio, M., Sahlholt, M., Bach, Anders, Gynther, M., Strømgaard, Kristian & Pickering, Darryl S, 5 Jun 2016, In: European Journal of Pharmacology. 780, p. 166-73 8 p.

    Research output: Contribution to journalJournal articlepeer-review

  6. Published

    Investigation of the presence and antinociceptive function of muscarinic acetylcholine receptors in the African naked mole-rat (Heterocephalus glaber)

    Jørgensen, K. B., Krogh-Jensen, K., Pickering, Darryl S, Kanui, T. & Abelson, Klas, 1 Jan 2016, In: Journal of Comparative Physiology A. Sensory, neural, and behavioral physiology. 202, 1, p. 7-15 9 p.

    Research output: Contribution to journalJournal articlepeer-review

  7. Published

    A pharmacological profile of the high-affinity GluK5 kainate receptor

    Møllerud, S., Kastrup, Jette Sandholm Jensen & Pickering, Darryl S, 2016, In: European Journal of Pharmacology. 788, p. 315-320 6 p.

    Research output: Contribution to journalJournal articlepeer-review

  8. Published

    Design, synthesis and structure-activity relationships of novel phenylalanine-based amino acids as kainate receptors ligands

    Szymańska, E., Chałupnik, P., Szczepańska, K., Moral, A. M. C., Pickering, Darryl S, Nielsen, Birgitte, Johansen, Tommy Nørskov & Kieć-Kononowicz, K., 2016, In: Bioorganic & Medicinal Chemistry Letters. 26, 22, p. 5568-5572 5 p.

    Research output: Contribution to journalJournal articlepeer-review

  9. Published

    Enthalpy-Entropy Compensation in the Binding of Modulators at Ionotropic Glutamate Receptor GluA2

    Krintel, C., Francotte, P., Pickering, Darryl S, Juknaite, L., Pøhlsgaaard, J., Olsen, L., Frydenvang, Karla Andrea, Goffin, E., Pirotte, B. & Kastrup, Jette Sandholm Jensen, 2016, In: Biophysical Journal. 110, 11, p. 2397-2406 10 p.

    Research output: Contribution to journalJournal articlepeer-review

  10. Published

    Modelling Affective Pain in Mice: Effects of Inflammatory Hypersensitivity on Place Escape/Avoidance Behaviour, Anxiety and Hedonic State

    Refsgaard, L. K., Hoffmann-Petersen, J., Sahlholt, M., Pickering, Darryl S & Andreasen T., Jesper, 2016, In: Journal of Neuroscience Methods. 262, p. 85-92 8 p.

    Research output: Contribution to journalJournal articlepeer-review

  11. Published

    Neto2 influences on kainate receptor pharmacology and function

    Han, L., Howe, J. & Pickering, Darryl S, 2016, In: Basic & Clinical Pharmacology & Toxicology. 119, p. 141-148 8 p.

    Research output: Contribution to journalJournal articlepeer-review

  12. Published

    Structural rearrangement of the intracellular domains during AMPA receptor activation

    Zachariassen, L. G., Katchan, L., Jensen, A. G., Pickering, Darryl S, Plested, A. & Kristensen, Anders Skov, 2016, In: Proceedings of the National Academy of Sciences USA (PNAS). 113, 27, p. E3950-E3959 10 p.

    Research output: Contribution to journalJournal articlepeer-review

  13. Published

    Structure of a High-Affinity Kainate Receptor: GluK4 Ligand-Binding Domain Crystallized with Kainate

    Kristensen, O., Kristensen, L. B., Møllerud, S., Frydenvang, Karla Andrea, Pickering, Darryl S & Kastrup, Jette Sandholm Jensen, 2016, In: Structure. 24, 9, p. 1582-1589 8 p.

    Research output: Contribution to journalJournal articlepeer-review

  14. Published

    Studies on Aryl-Substituted Phenylalanines: Synthesis, Activity, and Different Binding Modes at AMPA Receptors

    Szymanska, E., Frydenvang, Karla Andrea, Pickering, Darryl S, Krintel, C., Nielsen, Birgitte, Kooshki, A., Zachariassen, L. G., Olsen, L., Kastrup, Jette Sandholm Jensen & Johansen, Tommy Nørskov, 2016, In: Journal of Medicinal Chemistry. 59, 1, p. 448-461 14 p.

    Research output: Contribution to journalJournal articlepeer-review

  15. Published

    Synthesis and Pharmacological Characterization of the Selective GluK1 Radioligand (S)-2-Amino-3-(6-[3H]-2,4-dioxo-3,4-dihydrothieno[3,2-d]pyrimidin-1(2H)-yl)propanoic acid ([3H]-NF608)

    Alcaide, A., Marconi, L., Marek, A., Haym, I., Nielsen, Birgitte, Møllerud, S., Jensen, M., Conti, P., Pickering, Darryl S & Bunch, Lennart, 2016, In: MedChemComm. 7, p. 2136-2144 9 p.

    Research output: Contribution to journalJournal articlepeer-review

  16. Published

    Systemic and Brain Pharmacokinetics of Perforin Inhibitor Prodrugs

    Gynther, M., Pickering, Darryl S, Spicer, J., Denny, W. & Huttunen, K., 2016, In: Molecular Pharmaceutics. 13, 7, p. 2484-2491 8 p.

    Research output: Contribution to journalJournal articlepeer-review

  17. Published

    Tweaking subtype-selectivity and agonist efficacy at (S)-2-amino-3-(3-hydroxy-5-methyl-isoxazol-4-yl)propionic acid (AMPA) receptors in a small series of BnTetAMPA analogues

    Wang, S., Larsen, Y., Navarrete, C. V., Jensen, Anders A., Nielsen, Birgitte, Al-Musaed, A., Frydenvang, Karla Andrea, Kastrup, Jette Sandholm Jensen, Pickering, Darryl S & Clausen, Rasmus Prætorius, 2016, In: Journal of Medicinal Chemistry. 59, 5, p. 2244-2254 11 p.

    Research output: Contribution to journalJournal articlepeer-review

ID: 1299533