Christian Bernard Matthijs Poulie

Christian Bernard Matthijs Poulie

Guest Researcher


  1. 2024
  2. Published

    Development and Preclinical Evaluation of [211At]PSAt-3-Ga: An Inhibitor for Targeted α-Therapy of Prostate Cancer.

    El Fakiri, M., Ayada, N., Müller, Marius, Hvass, Lars, Gamzov, T. H., Clausen, Anne Skovsbo, Geis, N. M., Steinacker, N., Hansson, E., Lindegren, S., Aneheim, E., Jensen, H., Eder, A., Jensen, Andreas, Poulie, Christian Bernard Matthijs, Kjær, Andreas, Eder, M. & Herth, Matthias Manfred, 2024, In: Journal of nuclear medicine : official publication, Society of Nuclear Medicine. 65, 4, p. 593-599

    Research output: Contribution to journalJournal articleResearchpeer-review

  3. 2023
  4. Published

    Editorial: Prof. Frank Rösch's legacy in the radiopharmaceutical chemistry field

    Poulie, Christian Bernard Matthijs, Piel, M., Neumaier, B., Ross, T. & Herth, Matthias Manfred, 2023, In: Frontiers in Nuclear Medicine. 3, 1336481.

    Research output: Contribution to journalEditorialResearchpeer-review

  5. Published

    In Vitro and In Vivo Evaluation of Pellotine: A Hypnotic Lophophora Alkaloid

    Poulie, C. B. M., Chan, C. B., Parka, A., Lettorp, M., Vos, J., Raaschou, A., Pottie, E., Bundgaard, M. S., Sørensen, L. M. E., Cecchi, C. R., Märcher-Rørsted, E., Bach, A., Herth, M. M., Decker, A., Jensen, A. A., Elfving, B., Kretschmann, A. C., Stove, C. P., Kohlmeier, K. A., Cornett, C. & 3 others, Janfelt, Christian, Kornum, Birgitte Rahbek & Kristensen, Jesper Langgaard, 2023, In: ACS Pharmacology & Translational Science. 6, 10, p. 1492-1507

    Research output: Contribution to journalJournal articleResearchpeer-review

  6. Published

    Next generation fibroblast activation protein (FAP) targeting PET tracers : The tetrazine ligation allows an easy and convenient way to 18F-labeled (4-quinolinoyl)glycyl-2-cyanopyrrolidines

    Poulie, Christian Bernard Matthijs, Shalgunov, Vladimir, Elvas, F., Van Rymenant, Y., Moon, E. S., Battisti, Umberto Maria, De Loose, J., De Meester, I., Rösch, F., Van Der Veken, P. & Herth, Matthias Manfred, 2023, In: European Journal of Medicinal Chemistry. 262, 10 p., 115862.

    Research output: Contribution to journalJournal articleResearchpeer-review

  7. Published

    Structure–Activity Assessment and In-Depth Analysis of Biased Agonism in a Set of Phenylalkylamine 5-HT2A Receptor Agonists

    Pottie, E., Poulie, Christian Bernard Matthijs, Simon, Ícaro Ariel, Harpsøe, Kasper, D’Andrea, L., Komarov, I. V., Gloriam, David E., Jensen, Anders A., Kristensen, Jesper Langgaard & Stove, C. P., 2023, In: ACS Chemical Neuroscience. 14, 15, p. 2727–2742

    Research output: Contribution to journalJournal articleResearchpeer-review

  8. Published

    Synthesis and radiolabeling of a polar [125 I]I-1,2,4,5-tetrazine

    Bidesi, N., Shalgunov, Vladimir, Battisti, Umberto Maria, Hvass, Lars, Jørgensen, Jesper Tranekjær, Poulie, Christian Bernard Matthijs, Jensen, A. I., Kjær, Andreas & Herth, Matthias Manfred, 2023, In: Journal of Labelled Compounds and Radiopharmaceuticals. 66, 1, p. 22-30

    Research output: Contribution to journalJournal articleResearchpeer-review

  9. 2022
  10. Published

    (S)-2-Mercaptohistidine: A First Selective Orthosteric GluK3 Antagonist

    Poulie, Christian Bernard Matthijs, Larsen, Y., Leteneur, C., Barthet, G., Bjørn-Yoshimoto, Walden, Malhaire, F., Nielsen, Birgitte, Pin, J. P., Mulle, C., Pickering, Darryl S & Bunch, Lennart, 2022, In: ACS Chemical Neuroscience. 13, 10, p. 1580–1587

    Research output: Contribution to journalJournal articleResearchpeer-review

  11. Published

    Bioorthogonal Click of Colloidal Gold Nanoparticles to Antibodies In vivo

    Poulie, Christian Bernard Matthijs, Sporer, E., Hvass, Lars, Jørgensen, Jesper Tranekjær, Kempen, Paul Joseph, Lopes van den Broek, S. I., Shalgunov, Vladimir, Kjær, Andreas, Jensen, A. I. & Herth, Matthias Manfred, 2022, In: Chemistry - A European Journal. 28, 61, 10 p., e202201847.

    Research output: Contribution to journalJournal articleResearchpeer-review

  12. Published

    Covalent core-radiolabeling of polymeric micelles with125I/211At for theranostic radiotherapy

    Sporer, E., Poulie, Christian Bernard Matthijs, Bäck, T., Lindegren, S., Jensen, H., Kempen, Paul Joseph, Kjær, Andreas, Herth, Matthias Manfred & Jensen, A. I., 2022, In: Nanotheranostics. 6, 4, p. 388-399

    Research output: Contribution to journalJournal articleResearchpeer-review

  13. Published

    Discovery of β-Arrestin-Biased 25CN-NBOH-Derived 5-HT2A Receptor Agonists

    Poulie, Christian Bernard Matthijs, Pottie, E., Simon, I. A., Harpsøe, Kasper, D’andrea, L., Komarov, I. V., Gloriam, David E., Jensen, Anders A., Stove, C. P. & Kristensen, Jesper Langgaard, 2022, In: Journal of Medicinal Chemistry. 65, 18, p. 12031–12043

    Research output: Contribution to journalJournal articleResearchpeer-review

  14. 2021
  15. Published

    Evaluation of [Cu-64]Cu-NOTA-PEG7-H-Tz for Pretargeted Imaging in LS174T Xenografts-Comparison to [111In-111]In-DOTA-PEG11-BisPy-Tz

    Poulie, Christian Bernard Matthijs, Jørgensen, Jesper Tranekjær, Shalgunov, Vladimir, Kougioumtzoglou, G., Jeppesen, T. E., Kjær, Andreas & Herth, Matthias Manfred, 2021, In: Molecules. 26, 3, 9 p., 544.

    Research output: Contribution to journalJournal articleResearchpeer-review

  16. Published

    Lipophilicity and Click Reactivity Determine the Performance of Bioorthogonal Tetrazine Tools in Pretargeted In Vivo Chemistry

    Steen, E. J. L., Jørgensen, Jesper Tranekjær, Denk, C., Battisti, Umberto Maria, Norregaard, K., Edem, P. E., Bratteby, K., Shalgunov, Vladimir, Wilkovitsch, M., Svatunek, D., Poulie, Christian Bernard Matthijs, Hvass, Lars, Simon, M., Wanek, T., Rossin, R., Robillard, M., Kristensen, Jesper Langgaard, Mikula, H., Kjær, Andreas & Herth, Matthias Manfred, 2021, In: ACS Pharmacology & Translational Science. 4, 2, p. 824-833 10 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  17. Published

    Surface Adsorption of the Alpha-Emitter Astatine-211 to Gold Nanoparticles Is Stable In Vivo and Potentially Useful in Radionuclide Therapy

    Sporer, E., Poulie, Christian Bernard Matthijs, Lindegren, S., Aneheim, E., Jensen, H., Bäck, T., Kempen, Paul Joseph, Kjær, Andreas, Herth, Matthias Manfred & Jensen, A. I., 2021, In: Journal of Nanotheranostics. 2, 4, p. 196-207

    Research output: Contribution to journalJournal articleResearchpeer-review

  18. Published

    The Alkaloids from Lophophora diffusa and Other “False Peyotes”

    Chan, Camilla Bachmand, Poulie, Christian Bernard Matthijs, Wismann, S. S., Soelberg, Jens & Kristensen, Jesper Langgaard, 2021, In: Journal of Natural Products. 84, 8, p. 2398–2407

    Research output: Contribution to journalJournal articleResearchpeer-review

  19. 2020
  20. Published

    A Diversity Oriented Synthesis Approach to New 2,3-trans-Substituted l-Proline Analogs as Potential Ligands for the Ionotropic Glutamate Receptors

    Kayser, S., Temperini, Piero, Poulie, Christian Bernard Matthijs, Staudt, Markus, Nielsen, Birgitte, Pickering, Darryl S & Bunch, Lennart, 4 Mar 2020, In: ACS Chemical Neuroscience. 11, p. 702-714 13 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  21. Published

    Dark Classics in Chemical Neuroscience: NBOMes

    Poulie, Christian Bernard Matthijs, Jensen, Anders A., Halberstadt, A. & Kristensen, Jesper Langgaard, 2020, In: ACS Chemical Neuroscience. p. 3860–3869 10 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  22. Published

    Design, Synthesis, and Pharmacological Characterization of Heterobivalent Ligands for the Putative 5-HT2A/mGlu2 Receptor Complex

    Poulie, Christian Bernard Matthijs, Liu, N., Jensen, Anders A. & Bunch, Lennart, 2020, In: Journal of Medicinal Chemistry. 63, 17, p. 9928-9949 22 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  23. Published

    Fragment-based labeling using condensation reactions of six potential 5-HT7R PET tracers

    Tampio L'Estrade, E., Shalgunov, Vladimir, Lehel, S., Nymann Petersen, I., Poulie, Christian Bernard Matthijs, Edgar, F. G., Volk, B., Ohlsson, T., Erlandsson, M., Knudsen, Gitte Moos & Herth, Matthias Manfred, 2020, In: Journal of Radioanalytical and Nuclear Chemistry. 326, p. 1749-1762 14 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  24. 2019
  25. Published

    One-step synthesis of N-succinimidyl-4-[18F]Fluorobenzoate ([18F]SFB)

    Petersen, I. N., Madsen, J., Poulie, Christian Bernard Matthijs, Kjær, Andreas & Herth, Matthias Manfred, 22 Sep 2019, In: Molecules. 24, 19, 7 p., 3436.

    Research output: Contribution to journalJournal articleResearchpeer-review

  26. Published

    Design and Synthesis of 2,3-trans-Proline Analogs as Ligands for the Ionotropic Glutamate Receptors and the Excitatory Amino Acid Transporters

    Poulie, Christian Bernard Matthijs, Alcaide Lopez, A., Krell-Jørgensen, M. P., Larsen, Y., Astier, E., Bjørn-Yoshimoto, Walden, Yi, F., Syrenne, J. T., Storgaard, M., Nielsen, Birgitte, Frydenvang, Karla Andrea, Jensen, Anders A., Hansen, K. B., Pickering, Darryl S & Bunch, Lennart, 19 Jun 2019, In: A C S Chemical Neuroscience. 10, 6, p. 2989-3007 19 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  27. 2017
  28. Published

    Tetrabutylammonium Fluoride (TBAF) as a Mild and Versatile Reagent for Cleaving Boroxazolidones to their Corresponding Free α-Amino Acids

    Poulie, Christian Bernard Matthijs & Bunch, Lennart, Mar 2017, In: European Journal of Organic Chemistry. 11, p. 1475-1478

    Research output: Contribution to journalJournal articleResearchpeer-review

  29. 2013
  30. Published

    Heterocycles as nonclassical bioisosteres of alpha-amino acids

    Poulie, Christian Bernard Matthijs & Bunch, Lennart, Feb 2013, In: ChemMedChem. 8, 2, p. 205-215

    Research output: Contribution to journalJournal articleResearchpeer-review

ID: 43877477