Kristian Strømgaard

Kristian Strømgaard

Professor


  1. 1999
  2. Published

    Analogues of neuroactive polyamine wasp toxins that lack inner basic sites exhibit enhanced antagonism toward a muscle-type mammalian nicotinic acetylcholine receptor

    Strømgaard, Kristian, Brierley, M. J., Andersen, K., Sløk, F. A., Mellor, I. R., Usherwood, P. N., Krogsgaard-Larsen, Povl & Jaroszewski, J. W., 16 Dec 1999, In: Journal of Medicinal Chemistry. 42, 25, p. 5224-5234 11 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  3. 2000
  4. Published

    Solid phase synthesis and biological evaluation of enantiomerically pure wasp toxin analogues PhTX-343 and PhTX-12

    Strømgaard, Kristian, Bjørnsdottir, I., Andersen, K., Brierley, M. J., Rizoli, S., Eldursi, N., Mellor, I. R., Usherwood, P. N., Hansen, S. H., Krogsgaard-Larsen, Povl & Jaroszewski, J. W., Feb 2000, In: Chirality. 12, 2, p. 93-102 10 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  5. Published

    Solid-phase synthesis and biological evaluation of a combinatorial library of philanthotoxin analogues

    Strømgaard, Kristian, Brier, T. J., Andersen, K., Mellor, I. R., Saghyan, A., Tikhonov, D., Usherwood, P. N., Krogsgaard-Larsen, Povl & Jaroszewski, J. W., 16 Nov 2000, In: Journal of Medicinal Chemistry. 43, 23, p. 4526-4533 8 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  6. 2001
  7. Published

    Recent advances in the medicinal chemistry of polyamine toxins

    Strømgaard, Kristian, Andersen, K., Krogsgaard-Larsen, Povl & Jaroszewski, J. W., Nov 2001, In: Mini - Reviews in Medicinal Chemistry. 1, 4, p. 317-338 22 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  8. Published

    A versatile method for solid phase synthesis of polyamines: neuroactive polyamine toxins as example

    Strømgaard, Kristian, Andersen, K., Ruhland, T., Krogsgaard-Larsen, Povl & Jaroszewski, J. W., 2001, In: Synthesis. 6, p. 877-884 8 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  9. 2002
  10. Ginkgolides: selective acetylations, translactonization, and biological evaluation

    Jaracz, S., Strømgaard, Kristian & Nakanishi, K., 28 Jun 2002, In: Journal of Organic Chemistry. 67, 13, p. 4623-4626 4 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  11. Published

    Solid-phase synthesis of polyamine toxin analogues: potent and selective antagonists of Ca2+-permeable AMPA receptors

    Kromann, H., Krikstolaityte, S., Andersen, A. J., Andersen, K., Krogsgaard-Larsen, Povl, Jaroszewski, J. W., Egebjerg, J. & Strømgaard, Kristian, 19 Dec 2002, In: Journal of Medicinal Chemistry. 45, 26, p. 5745-5754 10 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  12. Ginkgolide derivatives for photolabeling studies: preparation and pharmacological evaluation

    Strømgaard, Kristian, Saito, D. R., Shindou, H., Ishii, S., Shimizu, T. & Nakanishi, K., 29 Aug 2002, In: Journal of Medicinal Chemistry. 45, 18, p. 4038-4046 9 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  13. Published

    Solid-phase synthesis and pharmacological evaluation of analogues of PhTX-12-A potent and selective nicotinic acetylcholine receptor antagonist

    Strømgaard, Kristian, Mellor, I. R., Andersen, K., Neagoe, I., Pluteanu, F., Usherwood, P. N. R., Krogsgaard-Larsen, Povl & Jaroszewski, J. W., 22 Apr 2002, In: Bioorganic & Medicinal Chemistry Letters. 12, 8, p. 1159-1162 4 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  14. 2003
  15. Published

    Contrasting actions of philanthotoxin-343 and philanthotoxin-(12) on human muscle nicotinic acetylcholine receptors

    Brier, T. J., Mellor, I. R., Tikhonov, D. B., Neagoe, I., Shao, Z., Brierley, M. J., Strømgaard, Kristian, Jaroszewski, J. W., Krogsgaard-Larsen, Povl & Usherwood, P. N. R., Oct 2003, In: Molecular Pharmacology. 64, 4, p. 954-964 11 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

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ID: 1302559