Birgitte Holst

Birgitte Holst

Guest Researcher


  1. 2008
  2. Published

    A second disulfide bridge from the N-terminal domain to extracellular loop 2 dampens receptor activity in GPR39

    Storjohann, L., Holst, Birgitte & Schwartz, Thue W., 2008, In: Biochemistry. 47, 35, p. 9198-207 9 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  3. Published

    Molecular mechanism of Zn2+ agonism in the extracellular domain of GPR39

    Storjohann, L., Holst, Birgitte & Schwartz, Thue W., 2008, In: FEBS Letters. 582, 17, p. 2583-8 5 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  4. Published

    Overlapping binding site for the endogenous agonist, small-molecule agonists, and ago-allosteric modulators on the ghrelin receptor

    Holst, Birgitte, Frimurer, T. M., Mokrosinski, J., Halkjaer, T., Cullberg, K. B., Underwood, C. R. & Schwartz, Thue W., 2008, In: Molecular Pharmacology. 75, 1, p. 44-59 15 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  5. 2007
  6. Published

    Allosteric enhancers, allosteric agonists and ago-allosteric modulators: where do they bind and how do they act?

    Schwartz, Thue W. & Holst, Birgitte, 2007, In: TIPS - Trends in Pharmacological Sciences. 28, 8, p. 366-73 7 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  7. Published

    GPR39 splice variants versus antisense gene LYPD1: expression and regulation in gastrointestinal tract, endocrine pancreas, liver, and white adipose tissue.

    Egerod, Kristoffer Lihme, Holst, Birgitte, Petersen, P. S., Hansen, Jacob B., Mulder, J., Hökfelt, T. & Schwartz, Thue W., 2007, In: Molecular Endocrinology. 21, 7, p. 1685-98 13 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  8. Published

    Identification of an efficacy switch region in the ghrelin receptor responsible for interchange between agonism and inverse agonism

    Holst, Birgitte, Mokrosinski, J., Lang, M., Brandt, E., Nygaard, R., Frimurer, T. M., Beck-Sickinger, A. G. & Schwartz, Thue W., 2007, In: Journal of Biological Chemistry. 282, 21, p. 15799-811 12 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  9. Published

    Importance of constitutive activity and arrestin-independent mechanisms for intracellular trafficking of the ghrelin receptor

    Holliday, N. D., Holst, Birgitte, Rodionova, E. A., Schwartz, Thue W. & Cox, H. M., 2007, In: Molecular Endocrinology. 21, 12, p. 3100-12 12 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  10. Published

    Melanocortin 4 receptor mutations in obese Czech children: Studies of prevalence, phenotype development, weight reduction response, and functional analysis

    Hainerova, I., Larsen, L. H., Holst, Birgitte, Finkova, M., Hainer, V., Lebl, J., Hansen, T. & Pedersen, O., 2007, In: Journal of Clinical Endocrinology and Metabolism. 92, 9, p. 3689-3696 7 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  11. 2006
  12. Published

    Ago-allosteric modulation and other types of allostery in dimeric 7TM receptors

    Schwartz, Thue W. & Holst, Birgitte, 2006, In: Journal of Receptors and Signal Transduction. 26, 1-2, p. 107-28 21 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

  13. Published

    GPR39 signaling is stimulated by zinc ions but not by obestatin

    Holst, Birgitte, Egerod, Kristoffer Lihme, Schild, E., Vickers, S. P., Cheetham, S., Gerlach, L., Storjohann, L., Stidsen, C. E., Jones, R., Beck-Sickinger, A. G. & Schwartz, Thue W., 2006, In: Endocrinology. 148, 1, p. 13-20 7 p.

    Research output: Contribution to journalJournal articleResearchpeer-review

ID: 9886